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- [21] Discovery of AG-120: A first-in-class inhibitor of IDH1 mutant enzymes for the treatment of cancers harboring IDH1 mutationsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 252Popovici-Muller, Janeta论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USALemieux, Rene论文数: 0 引用数: 0 h-index: 0机构: KSQ Therapeut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USASaunders, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Resilience Therapeut, Boston, MA USA Agios Pharmaceut, Cambridge, MA USASalituro, Francesco论文数: 0 引用数: 0 h-index: 0机构: Sage Therapeut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAYen, Katharine论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAStraley, Kimberly论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut, Boston, MA USA Agios Pharmaceut, Cambridge, MA USATobin, Erica论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAWang, Fang论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAGross, Stefan论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAArtin, Erin论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USADang, Lenny论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAYang, Hua论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAUtley, Luke论文数: 0 引用数: 0 h-index: 0机构: Alnylam Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAChen, Yue论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAOlaharski, Andrew论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USASilverman, Lee论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAAgresta, Sam论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USASu, Michael论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USABiller, Scott论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USA
- [22] A phase I study of the first-in-class mitochondrial metabolism inhibitor CPI-613 in patients with advanced hematologic malignancies.JOURNAL OF CLINICAL ONCOLOGY, 2013, 31 (15)Pardee, Timothy S.论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USALevitan, Denise A.论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USAHurd, David Duane论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USAEllis, Leslie R.论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USAIsom, Scott论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USAHarrelson, Robin论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USAManuel, Megan论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USADralle, Sarah论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USALyerly, Susan论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USAPowell, Bayard L.论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ Hlth Sci, Winston Salem, NC USA
- [23] Longitudinal Pharmacokinetic/Pharmacodynamic Profile of AG-120, a Potent Inhibitor of the IDH1 Mutant Protein, in a Phase 1 Study of IDH1-Mutant Advanced Hematologic MalignanciesBLOOD, 2015, 126 (23)Fan, Bin论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USALe, Kha论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAManyak, Erika论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USALiu, Hua论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAPrahl, Malia论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USABowden, Chris J.论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USABiller, Scott论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAAgresta, Sam论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USAYang, Hua论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut, Cambridge, MA USA Agios Pharmaceut, Cambridge, MA USA
- [24] FIRST-IN-CLASS, ORAL MUTANT IDH2 INHIBITOR REVERSES DIFFERENTIATION BLOCK IN ACUTE MYELOID LEUKAEMIA TO PRODUCE CLINICALLY MEANINGFUL RESPONSESEXPERIMENTAL HEMATOLOGY, 2017, 53 : S38 - S38论文数: 引用数: h-index:机构:
- [25] First-in-Human Phase 1 Trial of VT3989, a First-in-Class YAP/TEAD Inhibitor in Patients with Advanced MesotheliomaJOURNAL OF THORACIC ONCOLOGY, 2023, 18 (11) : S384 - S384Yap, T.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USADesai, J.论文数: 0 引用数: 0 h-index: 0机构: Peter MacCallum Canc Ctr, Melbourne, Vic, Australia Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USADagogo-Jack, I.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Canc Ctr, Boston, MA USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAMillward, M.论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth II Med Ctr, Linear Canc Trials, Perth, WA, Australia Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAKindler, H. L.论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Chicago, IL 60637 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USATolcher, A. W.论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, San Antonio, TX USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAFrentzas, S.论文数: 0 引用数: 0 h-index: 0机构: Monash Med Ctr, Clayton, Vic, Australia Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USABody, A. L.论文数: 0 引用数: 0 h-index: 0机构: Monash Med Ctr, Clayton, Vic, Australia Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAThurston, A.论文数: 0 引用数: 0 h-index: 0机构: Toxicol Solut, Marana, AZ USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAPost, L.论文数: 0 引用数: 0 h-index: 0机构: Vivace Therapeut, San Mateo, TX USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USADorr, F. A.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAKwiatkowski, D. J.论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, Boston, MA USA Dana Farber Canc Inst, Boston, MA 02115 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA
- [26] AG-120, A FIRST-IN-CLASS MUTANT IDH1 INHIBITOR IN PATIENTS WITH RECURRENT OR PROGRESSIVE IDH1 MUTANT GLIOMA: UPDATED RESULTS FROM THE PHASE 1 NON-ENHANCING GLIOMA POPULATIONNEURO-ONCOLOGY, 2017, 19 : 10 - 11Mellinghoff, Ingo K.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USATouat, Mehdi论文数: 0 引用数: 0 h-index: 0机构: Gustave Roussy, Villejuif, France Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMaher, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dallas, TX 75390 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USADe la Fuente, Macarena论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miami, FL USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USACloughesy, Timothy F.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Los Angeles, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAHoldhoff, Matthias论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Baltimore, MD USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USACote, Gregory M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Harvard Canc Ctr, Boston, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABurris, Howard论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAJanku, Filip论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAHuang, Ray论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Harvard Canc Ctr, Boston, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAYoung, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAEllingson, Benjamin论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Los Angeles, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USANimkar, Tara论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAJiang, Liewen论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut Inc, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAIshii, Yuko论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut Inc, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAChoe, Sung论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut Inc, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAFan, Bin论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut Inc, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USASteelman, Lori论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut Inc, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAYen, Katharine论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut Inc, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABowden, Chris论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut Inc, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAPandya, Susan论文数: 0 引用数: 0 h-index: 0机构: Agios Pharmaceut Inc, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAWen, Patrick Y.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Harvard Canc Ctr, Boston, MA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA
- [27] Trial in Progress: A Phase 1 Study of KTX-1001, an Oral, First-in-Class, Selective MMSET Inhibitor in Patients with Relapsed and Refractory Multiple MyelomaBLOOD, 2023, 142Berdeja, Jesus G.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USA Sarah Cannon Res Inst, Nashville, TN USADingli, David论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Sarah Cannon Res Inst, Nashville, TN USA论文数: 引用数: h-index:机构:Yee, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Ctr Canc, Boston, MA USA Sarah Cannon Res Inst, Nashville, TN USAChung, Alfred论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, San Francisco, CA USA Sarah Cannon Res Inst, Nashville, TN USAGasparetto, Cristina论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Duke Canc Inst, Med Ctr, Durham, NC USA Mayo Clin, Phoenix, AZ USA Sarah Cannon Res Inst, Nashville, TN USALeif Bergsagel, P.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USARoy, Vivek论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Div Hematol Oncol, Jacksonville, FL USA Sarah Cannon Res Inst, Nashville, TN USAAbdallah, Al-Ola论文数: 0 引用数: 0 h-index: 0机构: Univ Kansas, Med Ctr, Kansas City, KS USA US Myeloma Innovat Res Collaborat USMIRC, Kansas City, KS USA Sarah Cannon Res Inst, Nashville, TN USAThanendrarajan, Sharmilan论文数: 0 引用数: 0 h-index: 0机构: Univ Arkansas Med Sci, Winthrop P Rockefeller Canc Inst, Myeloma Ctr, Little Rock, AR USA Sarah Cannon Res Inst, Nashville, TN USAAfrough, Aimaz论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Hematol Malignancies & Cellular Therapy, Dallas, TX USA Sarah Cannon Res Inst, Nashville, TN USARosinol, Laura论文数: 0 引用数: 0 h-index: 0机构: Hosp Clin Barcelona, Hematopoiet Cell Transplantat Unit, IDIBAPS, Barcelona, Spain Sarah Cannon Res Inst, Nashville, TN USATrudel, Suzanne论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Div Med Oncol & Hematol, Toronto, ON, Canada Sarah Cannon Res Inst, Nashville, TN USARodriguez Otero, Paula论文数: 0 引用数: 0 h-index: 0机构: Ctr Invest Biomed Red Canc CIBERONC, Madrid, Spain Sarah Cannon Res Inst, Nashville, TN USATouzeau, Cyrille论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Nantes, Nantes, France Sarah Cannon Res Inst, Nashville, TN USABories, Pierre论文数: 0 引用数: 0 h-index: 0机构: Toulouse Univ, Inst Canc, Toulouse, France Sarah Cannon Res Inst, Nashville, TN USABang, Soo论文数: 0 引用数: 0 h-index: 0机构: K36 Therapeut, Cambridge, MA USA Sarah Cannon Res Inst, Nashville, TN USAConnolly, Terry论文数: 0 引用数: 0 h-index: 0机构: K36 Therapeut, Cambridge, MA USA Sarah Cannon Res Inst, Nashville, TN USAKim, Michelle论文数: 0 引用数: 0 h-index: 0机构: K36 Therapeut, Cambridge, MA USA Sarah Cannon Res Inst, Nashville, TN USALewis, Chad A.论文数: 0 引用数: 0 h-index: 0机构: K36 Therapeut, Cambridge, MA USA Sarah Cannon Res Inst, Nashville, TN USALinberg, Bao-Van Tran论文数: 0 引用数: 0 h-index: 0机构: K36 Therapeut, Cambridge, MA USA Sarah Cannon Res Inst, Nashville, TN USATravis Quigley, M.论文数: 0 引用数: 0 h-index: 0机构: K36 Therapeut, Cambridge, MA USA Sarah Cannon Res Inst, Nashville, TN USALandgren, Ola论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Myeloma Div, Sylvester Comprehens Canc Ctr, Miami, FL USA Sarah Cannon Res Inst, Nashville, TN USAUsmani, Saad Z.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Div Hematol Oncol, Dept Med, Myeloma Serv, New York, NY USA Sarah Cannon Res Inst, Nashville, TN USAMateos, Maria-Victoria论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Salamanca, IBSAL, Salamanca, Spain Sarah Cannon Res Inst, Nashville, TN USASiegel, David S.论文数: 0 引用数: 0 h-index: 0机构: Hackensack Univ, Multiple Myeloma Div, Med Ctr, Hackensack, NJ USA Sarah Cannon Res Inst, Nashville, TN USA
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