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- [1] Novel Orally Active Antimalarial ThiazolesJOURNAL OF MEDICINAL CHEMISTRY, 2011, 54 (21) : 7713 - 7719Cabrera, Diego Gonzalez论文数: 0 引用数: 0 h-index: 0机构: Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South Africa Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaDouelle, Frederic论文数: 0 引用数: 0 h-index: 0机构: Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South Africa Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaFeng, Tzu-Shean论文数: 0 引用数: 0 h-index: 0机构: Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South Africa Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaNchinda, Aloysius T.论文数: 0 引用数: 0 h-index: 0机构: Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South Africa Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaYounis, Yassir论文数: 0 引用数: 0 h-index: 0机构: Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South Africa Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaWhite, Karen L.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Ctr Drug Candidate Optimisat, Parkville, Vic 3052, Australia Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaWu, Quoc论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Ctr Drug Candidate Optimisat, Parkville, Vic 3052, Australia Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaRyan, Eileen论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Ctr Drug Candidate Optimisat, Parkville, Vic 3052, Australia Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaBurrows, Jeremy N.论文数: 0 引用数: 0 h-index: 0机构: ICC, CH-1215 Geneva, Switzerland Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaWaterson, David论文数: 0 引用数: 0 h-index: 0机构: ICC, CH-1215 Geneva, Switzerland Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South AfricaWitty, Michael J.论文数: 0 引用数: 0 h-index: 0机构: ICC, CH-1215 Geneva, Switzerland Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South Africa论文数: 引用数: h-index:机构:Charman, Susan A.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Ctr Drug Candidate Optimisat, Parkville, Vic 3052, Australia Univ Cape Town, Dept Chem, ZA-7701 Rondebosch, South Africa论文数: 引用数: h-index:机构:
- [2] Structure-activity relationships of orally active antimalarial acridones: Synthesis, optimization, and biological activityAMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, 2006, 75 (05): : 251 - 251Kelly, Jane X.论文数: 0 引用数: 0 h-index: 0机构: Portland VA Med Ctr, Portland, OR USA Portland VA Med Ctr, Portland, OR USASmilkstein, Martin论文数: 0 引用数: 0 h-index: 0机构: Portland VA Med Ctr, Portland, OR USA Portland VA Med Ctr, Portland, OR USAWinter, Rolf论文数: 0 引用数: 0 h-index: 0机构: Portland VA Med Ctr, Portland, OR USA Portland VA Med Ctr, Portland, OR USADodean, Rosie论文数: 0 引用数: 0 h-index: 0机构: Portland VA Med Ctr, Portland, OR USA Portland VA Med Ctr, Portland, OR USARiscoe, Mike论文数: 0 引用数: 0 h-index: 0机构: Portland VA Med Ctr, Portland, OR USA Portland VA Med Ctr, Portland, OR USA
- [3] Aminoazabenzimidazoles, a Novel Class of Orally Active Antimalarial AgentsJOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (13) : 5702 - 5713Hameed, Shahul P.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaChinnapattu, Murugan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaShanbag, Gajanan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaManjrekar, Praveena论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, India AstraZeneca India Pvt Ltd, Dept Med Chem, Bangalore 560024, Karnataka, IndiaKoushik, Krishna论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca India Pvt 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- [4] Potent Plasmodium falciparum Gametocytocidal Activity of Diaminonaphthoquinones, Lead Antimalarial Chemotypes Identified in an Antimalarial Compound ScreenANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2015, 59 (03) : 1389 - 1397Tanaka, Takeshi Q.论文数: 0 引用数: 0 h-index: 0机构: NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USAGuiguemde, W. Armand论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USABarnett, David S.论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USAMaron, Maxim I.论文数: 0 引用数: 0 h-index: 0机构: Loyola Univ Chicago, Dept Biol, Chicago, IL USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USAMin, Jaeki论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USAConnelly, Michele C.论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USASuryadevara, Praveen Kumar论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USAGuy, R. Kiplin论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USAWilliamson, Kim C.论文数: 0 引用数: 0 h-index: 0机构: NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USA Loyola Univ Chicago, Dept Biol, Chicago, IL USA NIAID, Lab Malaria & Vector Res, Bethesda, MD 20892 USA
- [5] ANTIMALARIAL PROPERTIES OF ORALLY ACTIVE IRON CHELATORSCLINICAL RESEARCH, 1988, 36 (03): : A411 - A411HEPPNER, DG论文数: 0 引用数: 0 h-index: 0机构: UNIV MINNESOTA,DEPT LAB MED & PATHOL,MINNEAPOLIS,MN 55455HALLAWAY, PE论文数: 0 引用数: 0 h-index: 0机构: UNIV MINNESOTA,DEPT LAB MED & PATHOL,MINNEAPOLIS,MN 55455KONTOGHIORGHES, GJ论文数: 0 引用数: 0 h-index: 0机构: UNIV MINNESOTA,DEPT LAB MED & PATHOL,MINNEAPOLIS,MN 55455EATON, JW论文数: 0 引用数: 0 h-index: 0机构: UNIV MINNESOTA,DEPT LAB MED & PATHOL,MINNEAPOLIS,MN 55455
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- [10] Arylmethoxypyridines as novel, potent and orally active mGlu5 receptor antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (07) : 1892 - 1897Büttelmann, B论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandPeters, JU论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandCeccarelli, S论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandKolczewski, S论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandVieira, E论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandPrinssen, EP论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandSpooren, W论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandSchuler, F论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandHuwyler, J论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandPorter, RHP论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, SwitzerlandJaeschke, G论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche Ltd, Div Pharma, Discovery Chem, CH-4070 Basel, Switzerland