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- [31] Discovery of SPH3127: A Novel, Highly Potent, and Orally Active Direct Renin InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (16) : 10882 - 10897Iijima, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaSugama, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaTakahashi, Yoichi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaHirai, Miki论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaTogashi, Yuko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaXie, Jianshu论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaShen, Jingkang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaKe, Ying论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaAkatsuka, Hidenori论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaKawaguchi, Takayuki论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaTakedomi, Kei论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaKashima, Akiko论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaNishio, Masashi论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaInui, Yosuke论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaYoneda, Hikaru论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaXia, Guangxin论文数: 0 引用数: 0 h-index: 0机构: Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R ChinaIijima, Toru论文数: 0 引用数: 0 h-index: 0机构: Mitsubishi Tanabe Pharm Corp, Sohyaku Innovat Res Div, Yokohama 2270033, Japan Univ Tokyo, Grad Sch Pharmaceut Sci, Lead Explorat Unit, Drug Discovery Initiat, Tokyo 1130033, Japan Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China
- [32] Discovery of novel quinoline sulphonamide derivatives as potent, selective and orally active RORγ inverse agonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (14) : 1799 - 1806Amaudrut, Jerome论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceArgiriadi, Maria A.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBarth, Martine论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBreinlinger, Eric C.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBressac, Didier论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBroqua, Pierre论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceCalderwood, David J.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceChatar, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceCusack, Kevin P.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceGauld, Stephen B.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 1 North Waukegan Rd, N Chicago, IL 60064 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceJacquet, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceKamath, Rajesh, V论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceKort, Michael E.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 1 North Waukegan Rd, N Chicago, IL 60064 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceLepais, Valerie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceLuccarini, Jean-Michel论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMasson, Philippe论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMontalbetti, Christian论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMounier, Laurent论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FrancePotin, Dominique论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FrancePoupardin, Olivia论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceRouaud, Sylvie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceSpitzer, Luc论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceWallace, Craig D.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, France
- [33] Novel pyrimidine-5-carboxylic acid as a potent and orally active PPARγ partial agonistABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 233 : 517 - 517Seto, Shigeki论文数: 0 引用数: 0 h-index: 0机构: Kyorin Pharmaceut Co Ltd, Discovery Res Labs, Dept Chem, Nogi, Tochigi 3290114, Japan Kyorin Pharmaceut Co Ltd, Discovery Res Labs, Dept Chem, Nogi, Tochigi 3290114, JapanOkada, Kyoko论文数: 0 引用数: 0 h-index: 0机构: Kyorin Pharmaceut Co Ltd, Discovery Res Labs, Dept Chem, Nogi, Tochigi 3290114, Japan Kyorin Pharmaceut Co Ltd, Discovery Res Labs, Dept Chem, Nogi, Tochigi 3290114, JapanKiyota, Koichi论文数: 0 引用数: 0 h-index: 0机构: Kyorin Pharmaceut Co Ltd, Discovery Res Labs, Dept Chem, Nogi, Tochigi 3290114, Japan Kyorin Pharmaceut Co Ltd, Discovery Res Labs, Dept Chem, Nogi, Tochigi 3290114, Japan
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