共 50 条
- [21] Discovery of potent, selective, orally bioavailable Stearoyl-CoA desaturase 1 inhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2007, 50 (13) : 3086 - 3100Liu, Gang论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALynch, John K.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAFreeman, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALiu, Bo论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAXin, Zhili论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAZhao, Hongyu论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASerby, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAKym, Philip R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASuhar, Tom S.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASmith, Harriet T.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USACao, Ning论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAYang, Ruojing论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAJanis, Rich S.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAKrauser, Joel A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USACepa, Steven P.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USABeno, David W. A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASham, Hing L.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USACollins, Christine A.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASurowy, Teresa K.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USACamp, Heidi S.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Metab Dis Res, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA
- [22] Discovery of potent, selective and orally bioavailable phenylailanine based dipeptidyl peptioase IV inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U145 - U145Xu, JY论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAWei, L论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAMathvink, R论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAHe, JF论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAPark, YJ论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAHe, HB论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USALeiting, B论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USALyons, KA论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAMarsilio, F论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAPatel, RA论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAWu, JK论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAThornberry, NA论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USAWeber, AE论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, Rahway, NJ 07065 USA
- [23] Discovery of potent, selective, and orally bioavailable inhibitors of interleukin-1 receptor-associate kinase-4BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (23) : 5546 - 5550Wang, Zhulun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USASun, Daqing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAJohnstone, Sheree论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USACao, Zhaodan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAGao, Xiong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAJaen, Juan C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USALiu, Jingqian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USALively, Sarah论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAMiao, Shichang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USASudom, Athena论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USATomooka, Craig论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAWalker, Nigel P. C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAWright, Matthew论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAYan, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAYe, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAPowers, Jay P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USA
- [24] Discovery and optimization of orally bioavailable and potent plasma Kallikrein inhibitors bearing a quaternary carbonBIOORGANIC & MEDICINAL CHEMISTRY, 2022, 73Zhang, Weihe论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAVadlakonda, Satish论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAWu, Minwan论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAChintareddy, Venkat论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAVogeti, L. N.论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAJuarez, Luis论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAMuppa, Saritha论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Biol, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAParker, Cynthia论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Biol, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAKellogg-Yelder, Debra论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Anim Studies, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAWilliams, Jason论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Bioanalyt Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAPolach, Kevin论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Med Writing & Regulatory Commun, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAChen, Xilin论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Biol, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USARaman, Krishnan论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Computat Chem & Struct Biol, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USABabu, Y. S.论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Biol, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Anim Studies, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Bioanalyt Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Computat Chem & Struct Biol, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USAKotian, Pravin论文数: 0 引用数: 0 h-index: 0机构: BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Bioanalyt Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Computat Chem & Struct Biol, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA BioCryst Pharmaceut Inc, Discovery Ctr Excellence, Dept Discovery Chem, 2100 Riverchase Ctr,Bldg 200,Suite 200, Birmingham, AL 35244 USA
- [25] Discovery of potent and orally bioavailable 17β-hydroxysteroid dehydrogenase type 3 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY, 2012, 20 (10) : 3242 - 3254Harada, Koichiro论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanKubo, Hideki论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanAbe, Jun论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanHaneta, Mari论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanConception, Arnel论文数: 0 引用数: 0 h-index: 0机构: Sumika Technoserv Corp, Div Organ Synth, Takarazuka, Hyogo 6650051, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanInoue, Shinichi论文数: 0 引用数: 0 h-index: 0机构: Sumika Technoserv Corp, Div Organ Synth, Takarazuka, Hyogo 6650051, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanOkada, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Sumika Technoserv Corp, Div Organ Synth, Takarazuka, Hyogo 6650051, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanNishioka, Kazuhiko论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Crop Protect Div Int, Chuo Ku, Tokyo 1048260, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan
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