Targeting WNT signaling in vivo via Tankyrase inhibition.

被引:0
|
作者
Schatoff, Emma M. [1 ]
Leach, Benjamin I. [1 ]
Foronda, Miguel [1 ]
Zafra, Maria Paz [1 ]
Dow, Lukas [1 ]
机构
[1] Weill Cornell Med, New York, NY USA
关键词
D O I
10.1158/1538-7445.MOUSEMODELS17-B32
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
B32
引用
收藏
页码:70 / 70
页数:1
相关论文
共 50 条
  • [1] Targeting WNT signaling in vivovia Tankyrase inhibition
    Schatoff, Emma M.
    Leach, Benjamin I.
    Foronda, Miguel
    Zafra, Maria Paz
    Goswami, Sukanya
    Dow, Lukas E.
    CANCER RESEARCH, 2018, 78 (13)
  • [2] Tankyrase inhibition represses Wnt signaling and lung cancer growth
    Busch, Alexander M.
    Johnson, Kevin C.
    Tacchelly, Ofelia
    Wang, Zhenghan
    Ahmed, Yashi F.
    Dmitrovsky, Ethan
    Freemantle, Sarah J.
    CANCER RESEARCH, 2012, 72
  • [3] Structural Basis and Selectivity of Tankyrase Inhibition by a Wnt Signaling Inhibitor WIKI4
    Haikarainen, Teemu
    Venkannagari, Harikanth
    Narwal, Mohit
    Obaji, Ezeogo
    Lee, Hao-Wei
    Nkizinkiko, Yves
    Lehtio, Lari
    PLOS ONE, 2013, 8 (06):
  • [4] Targeting Tankyrase to Fight WNT-dependent Tumours
    Thorvaldsen, Tor Espen
    BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, 2017, 121 (02) : 81 - 88
  • [5] Disruption of Wnt/β-Catenin Signaling and Telomeric Shortening Are Inextricable Consequences of Tankyrase Inhibition in Human Cells
    Kulak, Ozlem
    Chen, Hua
    Holohan, Brody
    Wu, Xiaofeng
    He, Huawei
    Borek, Dominika
    Otwinowski, Zbyszek
    Yamaguchi, Kiyoshi
    Garofalo, Lauren A.
    Ma, Zhiqiang
    Wright, Woodring
    Chen, Chuo
    Shay, Jerry W.
    Zhang, Xuewu
    Lum, Lawrence
    MOLECULAR AND CELLULAR BIOLOGY, 2015, 35 (14) : 2425 - 2435
  • [6] Triptolide has antitumor effects in lung cancer via Wnt pathway inhibition.
    Li, Youqiang
    Zheng, Li
    Shen, Binghui
    Kim, Jae
    Raz, Dan
    CLINICAL CANCER RESEARCH, 2014, 20
  • [7] Leukemia Stem Cells Are Resistant to In Vivo, Cell Non-Autonomous Wnt Inhibition.
    Lane, Steven W.
    Lo Celso, Cristina
    Sykes, Stephen M.
    Shterental, Sebastian
    Paktinat, Mahnaz
    Lin, Charles P.
    Williams, David A.
    Scadden, David T.
    Gilliland, D. Gary
    BLOOD, 2009, 114 (22) : 424 - 424
  • [8] Tankyrase inhibition stabilizes axin and antagonizes Wnt signalling
    Shih-Min A. Huang
    Yuji M. Mishina
    Shanming Liu
    Atwood Cheung
    Frank Stegmeier
    Gregory A. Michaud
    Olga Charlat
    Elizabeth Wiellette
    Yue Zhang
    Stephanie Wiessner
    Marc Hild
    Xiaoying Shi
    Christopher J. Wilson
    Craig Mickanin
    Vic Myer
    Aleem Fazal
    Ronald Tomlinson
    Fabrizio Serluca
    Wenlin Shao
    Hong Cheng
    Michael Shultz
    Christina Rau
    Markus Schirle
    Judith Schlegl
    Sonja Ghidelli
    Stephen Fawell
    Chris Lu
    Daniel Curtis
    Marc W. Kirschner
    Christoph Lengauer
    Peter M. Finan
    John A. Tallarico
    Tewis Bouwmeester
    Jeffery A. Porter
    Andreas Bauer
    Feng Cong
    Nature, 2009, 461 : 614 - 620
  • [9] Tankyrase inhibition stabilizes axin and antagonizes Wnt signalling
    Huang, Shih-Min A.
    Mishina, Yuji M.
    Liu, Shanming
    Cheung, Atwood
    Stegmeier, Frank
    Michaud, Gregory A.
    Charlat, Olga
    Wiellette, Elizabeth
    Zhang, Yue
    Wiessner, Stephanie
    Hild, Marc
    Shi, Xiaoying
    Wilson, Christopher J.
    Mickanin, Craig
    Myer, Vic
    Fazal, Aleem
    Tomlinson, Ronald
    Serluca, Fabrizio
    Shao, Wenlin
    Cheng, Hong
    Shultz, Michael
    Rau, Christina
    Schirle, Markus
    Schlegl, Judith
    Ghidelli, Sonja
    Fawell, Stephen
    Lu, Chris
    Curtis, Daniel
    Kirschner, Marc W.
    Lengauer, Christoph
    Finan, Peter M.
    Tallarico, John A.
    Bouwmeester, Tewis
    Porter, Jeffery A.
    Bauer, Andreas
    Cong, Feng
    NATURE, 2009, 461 (7264) : 614 - 620
  • [10] Tankyrase 1 inhibitior XAV939 increases chemosensitivity in colon cancer cell lines via inhibition of the Wnt signaling pathway
    Wu, Xuefang
    Luo, Feng
    Li, Jinbang
    Zhong, Xueyun
    Liu, Kunping
    INTERNATIONAL JOURNAL OF ONCOLOGY, 2016, 48 (04) : 1333 - 1340