Synthesis and evaluation of Schiff bases and 4-thiazolidinones as antibacterial agents

被引：0

作者：

Solankee, Anjani N. ^{[1
]}

机构：

[1] BKM Sci Coll, Dept Chem, Valsad 396001, Gujarat, India

来源：

JOURNAL OF THE INDIAN CHEMICAL SOCIETY | 2011年 / 88卷 / 11期

关键词：

Schiff bases; 4-thiazolidinones; thioglycolic acid; antibacterial activity; MANNICH REACTION-PRODUCTS; ANTIFUNGAL ACTIVITY; BIOLOGICAL-ACTIVITY; FUNGITOXICITY;

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

6-Methylpyridine-3-carbohydrazide (2) on condensation with different aromatic aldehydes (1) resulted in Schiff bases 3(a-i), which on cyclocondensation with thioglycolic acid resulted in 4-thiazolidinones 4(a-i). The newly synthesized compounds were characterized using IR, H-1 NMR, C-13 NMR and elemental analysis. Synthesized compounds were evaluated for their in vitro antibacterial activity against Gram-positive and Gram-negative strains.

引用

页码：1733 / 1738

页数：6

共 50 条

[41] CYANOETHYLATION OF SOME 4-THIAZOLIDINONES
HARHASH, AH
ELDINSOBHY, ME
ELNAGDI, MH
FODA, KM
EGYPTIAN JOURNAL OF CHEMISTRY, 1972, 15 (01): : 11 - 21
[42] Synthesis and biological evaluation of novel Indolyl 4-thiazolidinones bearing thiadiazine nucleus
Anekal, Doddappa Pralhad
Biradar, J. S.
ARABIAN JOURNAL OF CHEMISTRY, 2017, 10 : S2098 - S2105
[43] SYNTHESIS AND ANTIMICROBIAL ACTIVITY EVALUATION OF NOVEL 4-THIAZOLIDINONES CONTAINING A PYRONE MOIETY
Nechak, Rosa
Bouzroura, Samia Aichouche
Benmalek, Yamina
Salhi, Lydia
Martini, Sophie P.
Morizur, Vincent
Dunach, Elisabet
Kolli, Bellara Nedjar
SYNTHETIC COMMUNICATIONS, 2015, 45 (02) : 262 - 272
[44] 4-thiazolidinones: Synthesis and effect of chloro substituent on fungitoxicity
Upma, JR
Manrao, MR
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2004, 14 (02) : 177 - 178
[45] Structural design, synthesis and pharmacological evaluation of 4-thiazolidinones against Trypanosoma cruzi
de Oliveira Filho, Gevanio Bezerra
de Oliveira Cardoso, Marcos Verissimo
Pontes Espindola, Jose Wanderlan
Gomes Rebello Ferreira, Luiz Felipe
de Simone, Carlos Alberto
Ferreira, Rafaela Salgado
Coelho, Pollyanne Lacerda
Meira, Cassio Santana
Magalhaes Moreira, Diogo Rodrigo
Pereira Soares, Milena Botelho
Lima Leite, Ana Cristina
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 23 (23) : 7478 - 7486
[46] SYNTHESIS OF 4-THIAZOLIDINONES FROM RHODANINES BY THIOCARBONYL REMOVAL
HANSEN, MM
HARKNESS, AR
TETRAHEDRON LETTERS, 1994, 35 (38) : 6971 - 6974
[47] Synthesis of new pyrazolothiazole derivatives from 4-thiazolidinones
Turgut, Zuhal
Yolacan, Cigdem
Aydogan, Feray
Bagdatli, Emine
Ocal, Nuket
MOLECULES, 2007, 12 (09): : 2151 - 2159
[48] BRIDGED BIS(4-THIAZOLIDINONES) AND RELATED-COMPOUNDS WITH ANTIBACTERIAL ACTIVITY
PANDYA, D
NAIR, KB
PHARMAZIE, 1993, 48 (06): : 414 - 417
[49] Progress in the chemistry of 4-thiazolidinones
Hamama, Wafaa S.
Ismail, Mohamed A.
Shaaban, Saad
Zoorob, Hanafi H.
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2008, 45 (04) : 939 - 956
[50] 4-Thiazolidinones: The advances continue ...
Tripathi, Avinash C.
Gupta, Shiv Ji
Fatima, Gul Naz
Sonar, Pankaj Kumar
Verma, Amit
Saraf, Shailendra K.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 72 : 52 - 77

← 1 2 3 4 5 →