Inhibition of big endothelin-1 (BIG ET-1) responses in endothelium-denuded human coronary artery by the selective endothelin-converting enzyme-1 (ECE-1) inhibitor PD159790

被引:0
|
作者
Maguire, JJ
Ahn, K
Davenport, AP
机构
[1] Univ Cambridge, Addenbrookes Hosp, Ctr Clin Investigat, Clin Pharmacol Unit, Cambridge CB2 2QQ, England
[2] Parke Davis Pharmaceut Res, Ann Arbor, MI 48105 USA
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
193P
引用
收藏
页码:U102 / U102
页数:1
相关论文
共 50 条
  • [31] Endothelin-converting enzyme-1 (ECE-1) is a downstream target of the homeobox transcription factor Nkx2-5
    Funke-Kaiser, H
    Lemmer, J
    von Langsdorff, C
    Thomas, A
    Kovacevic, SD
    Strasdat, M
    Behrouzi, T
    Zollmann, FS
    Paul, M
    Orzechowski, HD
    HYPERTENSION, 2003, 42 (04) : 636 - 636
  • [32] Role for chymase in the conversion of big endothelin-1 to biologically active endothelin peptides by endothelium-denuded human umbilical vein in vitro
    Maguire, JJ
    Telyatnikova, N
    Davenport, AP
    BRITISH JOURNAL OF PHARMACOLOGY, 2000, 129 : U108 - U108
  • [33] Human endothelin-converting enzyme (ECE-1):: three isoforms with distinct subcellular localizations
    Schweizer, A
    Valdenaire, O
    Nelböck, P
    Deuschle, U
    Edwards, JBDM
    Stumpf, JG
    Löffler, BM
    BIOCHEMICAL JOURNAL, 1997, 328 : 871 - 877
  • [34] Endothelin-converting enzyme-1 inhibition and growth of human glioblastoma cells
    Berger, Y
    Delmilow, HI
    Blum-Kaelin, D
    Kitas, EA
    Löffler, BM
    Aebi, JD
    Juillerat-Jeanneret, L
    JOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (02) : 483 - 498
  • [35] D-VAL(22) CONTAINING HUMAN BIG ENDOTHELIN-1 ANALOG, [D-VAL(22)]BIG ET-1[16-38], INHIBITS THE ENDOTHELIN-CONVERTING ENZYME
    MORITA, A
    NOMIZU, M
    OKITSU, M
    HORIE, K
    YOKOGOSHI, H
    ROLLER, PP
    FEBS LETTERS, 1994, 353 (01) : 84 - 88
  • [36] [PHE(22)]-BIG ENDOTHELIN-1[19-37] - A NEW AND POTENT INHIBITOR OF THE ENDOTHELIN-CONVERTING ENZYME
    CLAING, A
    NEUGEBAUER, W
    YANO, M
    RAE, GA
    DORLEANSJUSTE, P
    JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1995, 26 : S72 - S74
  • [37] Effect of Endothelin-Converting Enzyme Inhibitors on big Endothelin-1 Induced Contraction in Isolated rat Basilar Artery
    M. Zimmermann
    C. S. Jung
    H. Vatter
    A. Raabe
    V. Seifert
    Acta Neurochirurgica, 2002, 144 : 1213 - 1219
  • [38] Effect of Endothelin-Converting Enzyme Inhibitors on big Endothelin-1 Induced Contraction in Isolated rat Basilar Artery
    Zimmermann, M
    Jung, CS
    Vatter, H
    Raabe, A
    Seifert, V
    ACTA NEUROCHIRURGICA, 2002, 144 (11) : 1213 - 1219
  • [39] Endothelin-converting enzyme-1 (ECE-1)-dependent trafficking of corticotropin-releasing factor receptor 1 (CRF-R1)
    Bhargava, Aditi
    Bunnett, Nigel W.
    Hasdemir, Burcu
    FASEB JOURNAL, 2010, 24
  • [40] PHARMACOLOGICAL EVIDENCE FOR THE SPECIFICITY OF THE PHOSPHORAMIDON-SENSITIVE ENDOTHELIN-CONVERTING ENZYME FOR BIG ENDOTHELIN-1
    TELEMAQUE, S
    GRATTON, JP
    CLAING, A
    DORLEANSJUSTE, P
    JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1993, 22 : S85 - S89