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- [41] Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (03) : 1340 - 1354Tabrizi, Mojgan Aghazadeh论文数: 0 引用数: 0 h-index: 0机构: Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyBaraldi, Pier Giovanni论文数: 0 引用数: 0 h-index: 0机构: Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyBaraldi, Stefania论文数: 0 引用数: 0 h-index: 0机构: Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyRuggiero, Emanuela论文数: 0 引用数: 0 h-index: 0机构: Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyDe Stefano, Lucia论文数: 0 引用数: 0 h-index: 0机构: Univ Trieste, Grad Sch Chem, I-34127 Trieste, Italy Natl Canc Inst, Dept Mol Biol & Translat Res, Div Expt & Clin Pharmacol, I-33081 Aviano, Pordenone, Italy Ctr Mol Biomed, I-33081 Aviano, Pordenone, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyRizzolio, Flavio论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Inst, Dept Mol Biol & Translat Res, Div Expt & Clin Pharmacol, I-33081 Aviano, Pordenone, Italy Ctr Mol Biomed, I-33081 Aviano, Pordenone, Italy Ca Foscari Univ Venezia, Dept Mol Sci & Nanosyst, I-30172 Venice, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyMannelli, Lorenzo Di Cesare论文数: 0 引用数: 0 h-index: 0机构: Univ Firenze, Sect Pharmacol & Toxicol, Dept Neurosci Psychol Drug Res & Child Hlth, I-50139 Florence, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyGhelardini, Carla论文数: 0 引用数: 0 h-index: 0机构: Univ Firenze, Sect Pharmacol & Toxicol, Dept Neurosci Psychol Drug Res & Child Hlth, I-50139 Florence, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyChicca, Andrea论文数: 0 引用数: 0 h-index: 0机构: Univ Bern, NCCR TransCure, Inst Biochem & Mol Med, CH-3012 Bern, Switzerland Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyLapillo, Margherita论文数: 0 引用数: 0 h-index: 0机构: Univ Pisa, Dept Pharm, I-56126 Pisa, Italy Univ Bern, NCCR TransCure, Inst Biochem & Mol Med, CH-3012 Bern, Switzerland Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyGertsch, Jurg论文数: 0 引用数: 0 h-index: 0机构: Univ Bern, NCCR TransCure, Inst Biochem & Mol Med, CH-3012 Bern, Switzerland Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, Italy论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Martinelli, Adriano论文数: 0 引用数: 0 h-index: 0机构: Univ Pisa, Dept Pharm, I-56126 Pisa, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyGranchi, Carlotta论文数: 0 引用数: 0 h-index: 0机构: Univ Pisa, Dept Pharm, I-56126 Pisa, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyMinutolo, Filippo论文数: 0 引用数: 0 h-index: 0机构: Univ Pisa, Dept Pharm, I-56126 Pisa, Italy Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, ItalyTuccinardi, Tiziano论文数: 0 引用数: 0 h-index: 0机构: Univ Pisa, Dept Pharm, I-56126 Pisa, Italy Temple Univ, Coll Sci & Technol, Ctr Biotechnol, Sbarro Inst Canc Res & Mol Med, Philadelphia, PA 19122 USA Univ Ferrara, Dept Chem & Pharmaceut Sci, I-44121 Ferrara, Italy
- [42] Discovery of C-5 Pyrazole-Substituted Pyrrolopyridine Derivatives as Potent and Selective Inhibitors for Janus Kinase 1JOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (10) : 6725 - 6742Lang, Jia-Jia论文数: 0 引用数: 0 h-index: 0机构: Univ South China, Hengyang Med Coll, Sch Chem & Chem Engn, Hengyang 421001, Peoples R China Univ South China, Key Lab Prot Struct & Funct Univ Hunan Prov, Hengyang 421001, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaLv, You论文数: 0 引用数: 0 h-index: 0机构: Univ Sci & Technol, Coll Bioresources Chem & Mat Engn, Xian 710021, Shaanxi, Peoples R China Xian Amazinggene Co Ltd, Xian 710026, Shaanxi, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaKobe, Bostjan论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Inst Mol Biosci, Australian Infect Dis Res Ctr, Sch Chem & Mol Biosci, Brisbane, Qld 4072, Australia Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaChen, Hongfei论文数: 0 引用数: 0 h-index: 0机构: Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaTan, Yan论文数: 0 引用数: 0 h-index: 0机构: Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaChen, Limei论文数: 0 引用数: 0 h-index: 0机构: Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaWang, Xuechuan论文数: 0 引用数: 0 h-index: 0机构: Univ Sci & Technol, Coll Bioresources Chem & Mat Engn, Xian 710021, Shaanxi, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaMi, Pengbing论文数: 0 引用数: 0 h-index: 0机构: Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R China Univ South China, Hengyang Med Coll, Sch Chem & Chem Engn, Hengyang 421001, Peoples R China Univ South China, Key Lab Prot Struct & Funct Univ Hunan Prov, Hengyang 421001, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaZheng, Xing论文数: 0 引用数: 0 h-index: 0机构: Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R China Univ South China, Hengyang Med Coll, Sch Chem & Chem Engn, Hengyang 421001, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R ChinaLin, Ying-Wu论文数: 0 引用数: 0 h-index: 0机构: Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R China Univ South China, Hengyang Med Coll, Sch Chem & Chem Engn, Hengyang 421001, Peoples R China Univ South China, Key Lab Prot Struct & Funct Univ Hunan Prov, Hengyang 421001, Peoples R China Univ South China, Hengyang Med Sch, Dept Pharm, Hengyang 421001, Hunan, Peoples R China
- [43] Discovery of 5-substituent-N-arylbenzamide derivatives as potent, selective and orally bioavailable LRRK2 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 27 (17) : 4034 - 4038Ding, Xiao论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaDai, Xuedong论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaLong, Kai论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaPeng, Cheng论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaAndreotti, Daniele论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurosci CEDD, Verona, Italy GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaBamborough, Paul论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Platform Technol Sci, Med Res Ctr, Gunnels Wood Rd, Stevenage, Herts, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaEatherton, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurosci CEDD, New Frontiers Sci Pk, Harlow, Essex, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaEdge, Colin论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Platform Technol Sci, Med Res Ctr, Gunnels Wood Rd, Stevenage, Herts, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaJandu, Karamjit S.论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, Med Res Ctr, Gunnels Wood Rd, Stevenage, Herts, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaNichols, Paula L.论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurosci CEDD, New Frontiers Sci Pk, Harlow, Essex, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaPhilps, Oliver J.论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, Med Res Ctr, Gunnels Wood Rd, Stevenage, Herts, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaStasi, Luigi Piero论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaWan, Zehong论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaXiang, Jia-Ning论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaDong, Kelly论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Platform Technol Sci, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaDossang, Pamela论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Platform Technol Sci, Med Res Ctr, Gunnels Wood Rd, Stevenage, Herts, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaHo, Ming-Hsun论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Platform Technol Sci, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaLi, Yi论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Platform Technol Sci, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaMensah, Lucy论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Platform Technol Sci, Med Res Ctr, Gunnels Wood Rd, Stevenage, Herts, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaGuan, Xiaoming论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaReith, Alastair D.论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurosci CEDD, New Frontiers Sci Pk, Harlow, Essex, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, Med Res Ctr, Gunnels Wood Rd, Stevenage, Herts, England GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R ChinaRen, Feng论文数: 0 引用数: 0 h-index: 0机构: GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China GSK Pharmaceut R&D, Neurodegenerat DPU, Neurosci Therapeut Area Unit, 898 Halei Rd,Zhangjiang Hitech Pk, Shanghai 201203, Peoples R China
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- [45] Discovery of Thieno[3,2-d]pyrimidine derivatives as potent and selective inhibitors of ataxia telangiectasia mutated and Rad3 related (ATR) kinaseEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 255Duan, Yunxin论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaCheng, Haodong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China论文数: 引用数: h-index:机构:Xia, Jiawei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaXu, Yerong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaZhang, Ruyue论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaSun, Rui论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaLu, Tao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R ChinaChen, Yadong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Peoples R China
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