Optimization of synthetically novel agonists of the putative cannabinoid receptor, GPR55, using an activated state model

被引：0
|
作者：
Lingerfelt, Mary [1 ]
Alfakhori, Lara [2 ]
Hurst, Dow [1 ]
Zhao, Pingwei [3 ]
Croatt, Mitch [2 ]
Abood, Mary [3 ]
Reggio, Patricia [2 ]
机构：
[1] Univ North Carolina Greensboro, Chem & Biochem, Pleasant Garden, NC USA
[2] Univ North Carolina Greensboro, Chem & Biochem, Greensboro, NC USA
[3] Temple Univ, Anat & Cell Biol, Philadelphia, PA 19122 USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2015年 / 249卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
61
引用
收藏
页数：2
相关论文
共 50 条
  • [41] Potential Metabolic and Behavioural Roles of the Putative Endo-cannabinoid Receptors GPR18, GPR55 and GPR119 in Feeding
    Ramirez-Orozco, Ricardo E.
    Garcia-Ruiz, Ricardo
    Morales, Paula
    Villalon, Carlos M.
    Rafael Villafan-Bernal, J.
    Marichal-Cancino, Bruno A.
    CURRENT NEUROPHARMACOLOGY, 2019, 17 (10) : 947 - 960
  • [42] Identification of the GPR55 Agonist Binding Site Using a Novel Set of High-Potency GPR55 Selective Ligands
    Kotsikorou, Evangelia
    Madrigal, Karla E.
    Hurst, Dow P.
    Sharir, Haleli
    Lynch, Diane L.
    Heynen-Genel, Susanne
    Milan, Loribelle B.
    Chung, Thomas D. Y.
    Setzman, Herbert H.
    Bai, Yushi
    Caron, Marc G.
    Barak, Larry
    Abood, Mary E.
    Reggio, Patricia H.
    BIOCHEMISTRY, 2011, 50 (25) : 5633 - 5647
  • [43] Identification of the GPR55 Antagonist Binding Site Using a Novel Set of High-Potency GPR55 Selective Ligands
    Kotsikorou, Evangelia
    Sharir, Haleli
    Shore, Derek M.
    Hurst, Dow P.
    Lynch, Diane L.
    Madrigal, Karla E.
    Heynen-Genel, Susanne
    Milan, Loribelle B.
    Chung, Thomas D. Y.
    Seltzman, Herbert H.
    Bai, Yushi
    Caron, Marc G.
    Barak, Larry S.
    Croatt, Mitchell P.
    Abood, Mary E.
    Reggio, Patricia H.
    BIOCHEMISTRY, 2013, 52 (52) : 9456 - 9469
  • [44] Targeting Oxidative Stress: Novel Coumarin-Based Inverse Agonists of GPR55
    Apweiler, Matthias
    Saliba, Soraya Wilke
    Streyczek, Jana
    Hurrle, Thomas
    Graessle, Simone
    Braese, Stefan
    Fiebich, Bernd L.
    INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2021, 22 (21)
  • [45] Cannabinoid receptor GPR55 activation blocks nicotine use disorder by regulation of AMPAR phosphorylation
    Qingqing Liu
    Jiaoyan Yu
    Xi Li
    Yanyan Guo
    Ting Sun
    Li Luo
    Jing Ren
    Wei Jiang
    Ruitao Zhang
    Peng Yang
    Qi Yang
    Psychopharmacology, 2021, 238 : 3335 - 3346
  • [46] Erratum: GPR55 regulates cannabinoid 2 receptor-mediated responses in human neutrophils
    Nariman A B Balenga
    Elma Aflaki
    Julia Kargl
    Wolfgang Platzer
    Ralf Schröder
    Stefanie Blättermann
    Evi Kostenis
    Andrew J Brown
    Akos Heinemann
    Maria Waldhoer
    Cell Research, 2011, 21 : 1641 - 1641
  • [47] The Cannabinoid Receptor GPR55 Affects Osteoclast Function in vitro and Bone Mass in vivo.
    Whyte, L.
    Ryberg, E.
    Ridge, S.
    Mackie, K.
    Greasley, P.
    Ross, R.
    Rogers, M. J.
    JOURNAL OF BONE AND MINERAL RESEARCH, 2008, 23 : S62 - S62
  • [48] Cannabinoid receptor GPR55 activation blocks nicotine use disorder by regulation of AMPAR phosphorylation
    Liu, Qingqing
    Yu, Jiaoyan
    Li, Xi
    Guo, Yanyan
    Sun, Ting
    Luo, Li
    Ren, Jing
    Jiang, Wei
    Zhang, Ruitao
    Yang, Peng
    Yang, Qi
    PSYCHOPHARMACOLOGY, 2021, 238 (11) : 3335 - 3346
  • [49] GPR55: Current Knowledge and Future Perspectives of a Purported "Type-3" Cannabinoid Receptor
    Moriconi, A.
    Cerbara, I.
    Maccarrone, M.
    Topai, A.
    CURRENT MEDICINAL CHEMISTRY, 2010, 17 (14) : 1411 - 1429
  • [50] The novel cannabinoid receptor GPR55 mediates anxiolytic-like effects in the medial orbital cortex of mice with acute stress
    Qi-xin Shi
    Liu-kun Yang
    Wen-long Shi
    Lu Wang
    Shi-meng Zhou
    Shao-yu Guan
    Ming-gao Zhao
    Qi Yang
    Molecular Brain, 10
12345