Practical and Efficient Synthesis of 3-Aryl-2H-benzo[1,4]thiazine Derivatives Catalyzed by KHSO4

被引:14
|
作者
Baghernejad, Bita [1 ]
Heravi, Majid M. [1 ]
Oskooie, Hossein A. [1 ]
机构
[1] Alzahra Univ, Dept Chem, Sch Sci, Tehran, Iran
关键词
o-Aminothiophenols; 3-aryl-2H-benzo[1; 4]thiazine; KHSO4; INHIBITORS; ALDEHYDES; POTENT; ACID;
D O I
10.1080/00397911003629465
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
[image omitted] KHSO4 efficiently catalyzes the condensation of o-aminothiophenols and 2-bromo-1-aryl-ethanones to yield 3-aryl-2H-benzo[1,4]thiazines in good yields.
引用
收藏
页码:589 / 593
页数:5
相关论文
共 50 条
  • [21] A KHSO4 promoted tandem synthesis of 1,3,4-thiadiazoles from thiohydrazides and DMF derivatives
    Gan, Zongjie
    Tian, Binghua
    Yuan, Jianyong
    Ran, Dongzhi
    Zhang, Lin
    Dong, Gang
    Pan, Tao
    Zeng, Yixin
    Yu, Yu
    TETRAHEDRON LETTERS, 2020, 61 (31)
  • [22] Sustainable synthesis of antibacterial 3-aryl-2H-benzo[b,1,4]oxazin-2-ones via SNAr Csp2-Csp2 coupling
    Salehzadeh, Fatemeh
    Esmkhani, Maryam
    Noori, Milad
    Javanshir, Shahrzad
    Iraji, Aida
    Mahdavi, Mohammad
    FRONTIERS IN CHEMISTRY, 2024, 12
  • [23] In(OTf)3-catalyzed tandem aza-Piancatelli rearrangement/Michael reaction for the synthesis of 3,4-dihydro-2H-benzo[b][1,4]thiazine and oxazine derivatives
    Reddy, B. V. Subba
    Reddy, Y. Vikram
    Lakshumma, P. Subba
    Narasimhulu, G.
    Yadav, J. S.
    Sridhar, B.
    Reddy, P. Purushotham
    Kunwar, A. C.
    RSC ADVANCES, 2012, 2 (28): : 10661 - 10666
  • [24] Samarium diiodide catalyzed synthesis of 2,3-dihydro-1H-benzo[b][1,4]-diazepine derivatives
    Luo, YQ
    Xu, F
    Han, XY
    Shen, Q
    CHINESE JOURNAL OF CHEMISTRY, 2005, 23 (10) : 1417 - 1420
  • [25] Efficient synthesis of 2,2-disubstituted 4H-benzo[1,4]oxazin-3-ones or 4H-benzo[1,4]thiazin-3-ones by nucleophilic aromatic substitution
    Powell, Noel A.
    Ciske, Fred L.
    Cai, Cuiman
    Holsworth, Daniel D.
    Van Huis, Chad
    Edmunds, Jeremy J.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 231
  • [26] Efficient synthesis of novel benzo-[e]-[1,4]-diazepine derivatives
    Messeri, T
    Pentassuglia, G
    Di Fabio, R
    TETRAHEDRON LETTERS, 2001, 42 (18) : 3227 - 3230
  • [27] Synthesis of (Z)-hetarylmethylene and (Z)-substituted benzylidene derivatives of 4H-benzo[1,4]thiazine-3-thiones and their subsequent conversion to benzothiopyrano-[3,2-b][1,4]benzothiazines
    Kamila, S
    Koh, B
    Zhang, HM
    Biehl, ER
    ARKIVOC, 2006, : 1 - 14
  • [28] Synthesis of 3-methyl-4H-benzo[b][1,4]thiazine-2-carboxylates Using CAN as a Catalyst and Its Conversion Into Guanidines
    Jawale, Dhanaji, V
    Wagare, Devendra
    Lingampalle, Dinesh L.
    Netankar, Prashant D.
    CURRENT ORGANOCATALYSIS, 2021, 8 (02) : 258 - 263
  • [29] A Straightforward Approach for the Synthesis of Novel Derivatives of Benzo[b]pyrazolo[5,1:2,3]pyrimido[4,5-e][1,4]thiazine
    Sheikhi-Mohammareh, Seddigheh
    Shiri, Ali
    Bakavoli, Mehdi
    Mague, Joel
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2016, 53 (04) : 1231 - 1235
  • [30] Solid-phase synthesis of 2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine derivatives
    Liu, Zhang
    Chen, Wenteng
    Giulianotti, Marc A.
    Houghten, Richard A.
    TETRAHEDRON LETTERS, 2011, 52 (32) : 4112 - 4113