Microwave assisted synthesis of 4-thiazolidinones and its 5-arylidene derivatives: Screening of antimicrobial activity with various microorganisms

被引：0

作者：

Upadhyay, Apoorva ^{[1
]}

Srivastava, S. K. ^{[1
]}

Srivastava, S. D. ^{[1
]}

Upadhyay, Navneeta ^{[2
]}

机构：

[1] Dr Hari Singh Gour Vishwavidyalaya, Synthet Organ Chem Lab, Dept Chem, Sagar 470003, Madhya Pradesh, India

[2] Chameli Devi Inst Technol, Dept Chem, Indore, Madhya Pradesh, India

来源：

JOURNAL OF THE INDIAN CHEMICAL SOCIETY | 2011年 / 88卷 / 07期

关键词：

Isonicotinamide; thiazolidinone; microwave synthesis; antimicrobial agents; ANTI-HIV AGENTS; ORGANIC-SYNTHESIS; CANCER; DESIGN; ACID;

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Several new ethyl(isonicotinamid-4-yl)acetate (1), 2-(isonicotinamid-4-yl)acetohydrazide (2), 2-(isonicotinamid-4-yl)acetylhydrazino arylidenes (3a-j), 2-aryl-3-[(isonicotinamid-4-yl)acetamido]-4-oxo-1,3-thiazolidines (4a-j) and 5-arylidene-2-aryl-3-[(isonicotinamid-4-yl)acetamido]-4-oxo-1,3-thiazolidines (5a-j) have been synthesized. The structures of all the newly synthesized compounds were confirmed by IR, (1)H NMR, (13)C NMR, FAB-Mass spectra and by microanalytical data. Compounds 4a-j and 5a-j have been screened for their antibacterial and antifungal activity against some selected microorganisms.

引用

页码：1025 / 1031

页数：7

共 50 条

[41] Synthesis and antimicrobial activity of 5-arylidene-4-oxo-thiazolidines
Desai, N. C.
Bhavsar, A. M.
Shavalia, Alpesh
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2007, 16 (03) : 271 - 274
[42] 5-arylidene derivatives of Meldrum's acid as synthons in pyrano[4,3-b]pyran synthesis
Palasz, Aleksandra
Jelska, Katarzyna
Ozog, Monika
Serda, Pawel
MONATSHEFTE FUR CHEMIE, 2007, 138 (05): : 481 - 488
[43] One-pot synthesis of 5-arylidene-2-imino-4-thiazolidinones under microwave irradiation
Kasmi-Mir, Souad
Djafri, Ayada
Paquin, Ludovic
Hamelin, Jack
Rahmouni, Mustapha
MOLECULES, 2006, 11 (08): : 597 - 602
[44] Synthesis and fungicidal activity of 2-imino-3-(4-arylthiazol-2-yl)-thiazolidin-4-ones and their 5-arylidene derivatives
Liu, HL
Li, ZC
Anthonsen, T
MOLECULES, 2000, 5 (09) : 1055 - 1061
[45] 5-Arylidene Derivatives of Meldrum’s Acid as Synthons in Pyrano[4,3-b]pyran Synthesis
Aleksandra Pałasz
Katarzyna Jelska
Monika Ożóg
Paweł Serda
Monatshefte für Chemie - Chemical Monthly, 2007, 138 : 481 - 488
[46] STUDIES ON 4-THIAZOLIDINONES .5. SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 2-ARYL-3(2',4'-DIPHENYLAMINO-SYM-TRIAZIN-6'-YL)-5-H/METHYL/CARBOXYMETHYL-4-THIAZOLIDINONES
MEHTA, L
PAREKH, H
JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 1988, 65 (09) : 648 - 650
[47] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 4-THIAZOLIDINONES, 2-AZETIDINONES, 4-IMIDAZOLINONE DERIVATIVES HAVING THYMOL MOIETY
VASHI, BS
MEHTA, DS
SHAH, VH
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1995, 34 (09): : 802 - 808
[48] STUDIES ON 4-THIAZOLIDINONES .8. PREPARATION AND ANTIMICROBIAL ACTIVITY OF 2-ARYL-3-ACRIDIN-9-YLAMINO-5-METHYL CARBOXYMETHYL-4-THIAZOLIDINONES
PATEL, CL
PAREKH, H
JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 1988, 65 (04) : 282 - 284
[49] Microwave assisted synthesis and antimicrobial activity of some novel pyrimidine derivatives
Vaghasia, S. J.
Shah, V. H.
JOURNAL OF THE SERBIAN CHEMICAL SOCIETY, 2007, 72 (02) : 109 - 117
[50] Microwave assisted synthesis and antimicrobial screening of pyrazoline-5-ones
Shiradkar, Mahendra
Kale, Rajesh
Baviskar, Bhushan
Dighe, Rajendra
ASIAN JOURNAL OF CHEMISTRY, 2007, 19 (01) : 449 - 453

← 1 2 3 4 5 →