Microwave assisted synthesis of 4-thiazolidinones and its 5-arylidene derivatives: Screening of antimicrobial activity with various microorganisms

被引：0

作者：

Upadhyay, Apoorva ^{[1
]}

Srivastava, S. K. ^{[1
]}

Srivastava, S. D. ^{[1
]}

Upadhyay, Navneeta ^{[2
]}

机构：

[1] Dr Hari Singh Gour Vishwavidyalaya, Synthet Organ Chem Lab, Dept Chem, Sagar 470003, Madhya Pradesh, India

[2] Chameli Devi Inst Technol, Dept Chem, Indore, Madhya Pradesh, India

来源：

JOURNAL OF THE INDIAN CHEMICAL SOCIETY | 2011年 / 88卷 / 07期

关键词：

Isonicotinamide; thiazolidinone; microwave synthesis; antimicrobial agents; ANTI-HIV AGENTS; ORGANIC-SYNTHESIS; CANCER; DESIGN; ACID;

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Several new ethyl(isonicotinamid-4-yl)acetate (1), 2-(isonicotinamid-4-yl)acetohydrazide (2), 2-(isonicotinamid-4-yl)acetylhydrazino arylidenes (3a-j), 2-aryl-3-[(isonicotinamid-4-yl)acetamido]-4-oxo-1,3-thiazolidines (4a-j) and 5-arylidene-2-aryl-3-[(isonicotinamid-4-yl)acetamido]-4-oxo-1,3-thiazolidines (5a-j) have been synthesized. The structures of all the newly synthesized compounds were confirmed by IR, (1)H NMR, (13)C NMR, FAB-Mass spectra and by microanalytical data. Compounds 4a-j and 5a-j have been screened for their antibacterial and antifungal activity against some selected microorganisms.

引用

页码：1025 / 1031

页数：7

共 50 条

[21] Ultrasound assisted, VOSO4 catalyzed synthesis of 4-thiazolidinones: Antimicrobial evaluation of indazole-4-thiazolidinone derivatives
Angapelly, Srinivas
Ramya, P. V. Sri
SunithaRani, Routhu
Kumar, C. Ganesh
Kamal, Ahmed
Arifuddin, Mohammed
TETRAHEDRON LETTERS, 2017, 58 (49) : 4632 - 4637
[22] Synthesis of alkoxyphthalimide derivatives of 5-arylidene-2-(6′-chlorobenzothiazol-2′-yl-imino)-4-thiazolidinones
Dixit, N
Talesara, GL
JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 2005, 82 (08) : 754 - 756
[23] SYNTHESIS AND ANTIMICROBIAL ACTIVITY EVALUATION OF NOVEL 4-THIAZOLIDINONES CONTAINING A PYRONE MOIETY
Nechak, Rosa
Bouzroura, Samia Aichouche
Benmalek, Yamina
Salhi, Lydia
Martini, Sophie P.
Morizur, Vincent
Dunach, Elisabet
Kolli, Bellara Nedjar
SYNTHETIC COMMUNICATIONS, 2015, 45 (02) : 262 - 272
[24] Synthesis of some novel fluorinated 4-thiazolidinones containing amide linkages and their antimicrobial screening
Shah, Tejaskumar J.
Desai, Vikas A.
ARKIVOC, 2007, : 218 - 228
[25] 4-Thiazolidinone Based 5-Arylidene Hybrids: Design, Synthesis, Antimicrobial Activity, and Molecular Docking Studies
Desai, Nisheeth C. C.
Jadeja, Dharmpalsinh J. J.
Khasiya, Ashvinkumar G. G.
Dave, Bharti P. P.
Khedkar, Vijay M. M.
POLYCYCLIC AROMATIC COMPOUNDS, 2024, 44 (04) : 2715 - 2732
[26] Synthesis and biological activity evaluation of 5-pyrazoline substituted 4-thiazolidinones
Havrylyuk, Dmytro
Zimenkovsky, Borys
Vasylenko, Olexandr
Day, Craig W.
Smee, Donald F.
Grellier, Philippe
Lesyk, Roman
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 66 : 228 - 237
[27] Microwave assisted synthesis and antimicrobial screening of substituted 2-aryl-5-H-(3′-chloro-5′-phenoxy benzo(b) thiophenoyl-2-amino)-4-thiazolidinones
Vasoya, SL
Thaker, KM
Popat, KH
Joshi, HS
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2003, 13 (01) : 65 - 68
[28] SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF N(10)-ARYLIDENEHYDRAZIDOPHENOTHIAZINE AND THEIR 4-THIAZOLIDINONES AND 2-AZETIDINONES
HOGALE, MB
UTHALE, AC
NIKAM, BP
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1991, 30 (07): : 717 - 720
[29] Synthesis and antibiofilm activity of marine natural product-based 4-thiazolidinones derivatives
Rane, Rajesh A.
Sahu, Niteshkumar U.
Shah, Chetan P.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (23) : 7131 - 7134
[30] Synthesis and antimicrobial activity of some new 4-thiazolidinones derived from heterocyclic Schiff bases
Kumar, D
Sharma, RC
JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 2002, 79 (03) : 284 - 285

← 1 2 3 4 5 →