Microwave assisted synthesis of 4-thiazolidinones and its 5-arylidene derivatives: Screening of antimicrobial activity with various microorganisms

被引：0

作者：

Upadhyay, Apoorva ^{[1
]}

Srivastava, S. K. ^{[1
]}

Srivastava, S. D. ^{[1
]}

Upadhyay, Navneeta ^{[2
]}

机构：

[1] Dr Hari Singh Gour Vishwavidyalaya, Synthet Organ Chem Lab, Dept Chem, Sagar 470003, Madhya Pradesh, India

[2] Chameli Devi Inst Technol, Dept Chem, Indore, Madhya Pradesh, India

来源：

JOURNAL OF THE INDIAN CHEMICAL SOCIETY | 2011年 / 88卷 / 07期

关键词：

Isonicotinamide; thiazolidinone; microwave synthesis; antimicrobial agents; ANTI-HIV AGENTS; ORGANIC-SYNTHESIS; CANCER; DESIGN; ACID;

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Several new ethyl(isonicotinamid-4-yl)acetate (1), 2-(isonicotinamid-4-yl)acetohydrazide (2), 2-(isonicotinamid-4-yl)acetylhydrazino arylidenes (3a-j), 2-aryl-3-[(isonicotinamid-4-yl)acetamido]-4-oxo-1,3-thiazolidines (4a-j) and 5-arylidene-2-aryl-3-[(isonicotinamid-4-yl)acetamido]-4-oxo-1,3-thiazolidines (5a-j) have been synthesized. The structures of all the newly synthesized compounds were confirmed by IR, (1)H NMR, (13)C NMR, FAB-Mass spectra and by microanalytical data. Compounds 4a-j and 5a-j have been screened for their antibacterial and antifungal activity against some selected microorganisms.

引用

页码：1025 / 1031

页数：7

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