A convenient method for the synthesis of 2-trichloromethyl-4-p-substituted-phenyl-3H-1,5-benzodiazepines.

被引：56
|
作者：
Bonacorso, HG
Bittencourt, ST
Wastowski, AD
Wentz, AP
Zanatta, N
Martins, MAP
机构：
[1] Departamento de Química, Univ. Federal de Santa Maria(UFSM), 97119-900 Santa Maria, RS
来源：
TETRAHEDRON LETTERS | 1996年 / 37卷 / 51期
关键词：
D O I：
10.1016/S0040-4039(96)02145-4
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A convenient method to obtain a new series of 2-trichloromethyl-4-aryl-3H-1,5-benzodiazepines from the reaction of beta-methoxyvinyl trichloromethyl ketones derived from acetals and o-phenylenediamine is reported. Copyright (C) 1996 Elsevier Science Ltd
引用
收藏
页码：9155 / 9156
页数：2
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