A convenient method for the synthesis of 2-trichloromethyl-4-p-substituted-phenyl-3H-1,5-benzodiazepines.

被引：56
|
作者：
Bonacorso, HG
Bittencourt, ST
Wastowski, AD
Wentz, AP
Zanatta, N
Martins, MAP
机构：
[1] Departamento de Química, Univ. Federal de Santa Maria(UFSM), 97119-900 Santa Maria, RS
来源：
TETRAHEDRON LETTERS | 1996年 / 37卷 / 51期
关键词：
D O I：
10.1016/S0040-4039(96)02145-4
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A convenient method to obtain a new series of 2-trichloromethyl-4-aryl-3H-1,5-benzodiazepines from the reaction of beta-methoxyvinyl trichloromethyl ketones derived from acetals and o-phenylenediamine is reported. Copyright (C) 1996 Elsevier Science Ltd
引用
收藏
页码：9155 / 9156
页数：2
相关论文
共 50 条
  • [41] Synthesis of 1H-3-ferrocenyl-1-phenyl-4-substituted pyrazoles
    Joksovic, Milan
    Ratkovic, Zoran
    Vukicevic, Mirjana
    Vukicevic, Rastko D.
    SYNLETT, 2006, (16) : 2581 - 2584
  • [42] A CONVENIENT SYNTHESIS OF 3-CHLORO-3,4-DIHYDRO-4-HYDROXY-3-NITRO-2-PHENYL-2H-1-BENZOPYRANS
    DAUZONNE, D
    DEMERSEMAN, P
    SYNTHESIS-STUTTGART, 1990, (01): : 66 - 70
  • [43] SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 1-(P-SUBSTITUTED)PHENYL-3-(P-ALKOXY)PHENYL-4-PHENYL-AZETIDIN-2-ONES
    DIURNO, MV
    CRISTINZIANO, A
    MAZZONI, O
    PISCOPO, E
    BOLOGNESE, A
    FARMACO, 1995, 50 (02): : 143 - 148
  • [44] CONVENIENT SYNTHESIS OF 2-SUBSTITUTED 3-NITRO-2H-CHROMENE DERIVATIVES
    SAKAKIBARA, T
    KOEZUKA, M
    SUDOH, R
    BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, 1978, 51 (10) : 3095 - 3096
  • [45] A CONVENIENT SYNTHESIS OF NOVEL 3-QUINOXALINYL-1,5-BENZODIAZEPINES - STABLE TAUTOMERS IN 1,5-BENZODIAZEPIN-2-ONE RING-SYSTEM
    KURASAWA, Y
    SATOH, J
    OGURA, M
    OKAMOTO, Y
    TAKADA, A
    HETEROCYCLES, 1984, 22 (07) : 1531 - 1535
  • [46] Reaction of 4-aryl-2,3-dihydro-2-phenyl-1H-1,5-benzodiazepines with 2-chloroacetyl chloride.: Synthesis of N-acyl- and azeto[1,2-a]-1,5-benzodiazepines
    Insuasty, Braulio
    Quiroga, Jairo
    Abonia, Rodrigo
    Insuasty, Henry
    Escobar, Henry
    Diaz, Emilso
    Nogueras, Manuel
    HETEROCYCLIC COMMUNICATIONS, 2006, 12 (05) : 347 - 354
  • [47] Synthesis and Herbicidal Activity of 2-Substituted-6-methyl-4-phenyl-3(2H)-pyridazinone
    Xu, Han
    Zhang, Mingzhe
    Liu, Bin
    Yang, Huazheng
    CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2014, 34 (04) : 722 - 728
  • [48] A convenient synthesis of 2-Substituted 3-Nitro-2H-chromene Derivatives
    Sakakibara, Tohru
    Koezuica, Masaru
    Sudoh, Rokuro
    Bulletin of the Chemical Society of Japan, 1978, 51 (10): : 3095 - 3096
  • [49] A convenient general synthesis of 3-substituted 2H-chromene derivatives
    Kaye, PT
    Nocanda, XW
    JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 2002, (10): : 1318 - 1323
  • [50] STUDIES ON 4(1H)-QUINAZOLINONES .1. A CONVENIENT SYNTHESIS AND SOME REACTIONS OF 1-PHENYL-2-SUBSTITUTED-4(1H)-QUINAZOLINONES
    OZAKI, K
    YAMADA, Y
    OINE, T
    CHEMICAL & PHARMACEUTICAL BULLETIN, 1980, 28 (03) : 702 - 707
12345