共 46 条
- [1] Pre-clinical characterization of a novel series of FGFR2 selective inhibitors with potency against clinically relevant mutationsCANCER RESEARCH, 2022, 82 (12)Fischer, John论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USABouhana, Karyn论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAChicarelli, Mark J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USADahlke, Josh论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAFell, Brad论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAFulton, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAGuarnieri, Anna论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAJalluri, Ravi论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAJohnson, Amber论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAMclean, Brent论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAMejia, Max论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USARieger, Rob论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USARobinson, John论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USARodriguez, Mareli论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USASullivan, Francis论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAWang, Yang论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAWinski, Shannon论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAZhou, Yeyun论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USA
- [2] In vivo characterization of a selective FGFR2 inhibitor with potency against gatekeeper and molecular brake mutationsCANCER RESEARCH, 2023, 83 (07)Fischer, John论文数: 0 引用数: 0 h-index: 0Bouhana, Karyn论文数: 0 引用数: 0 h-index: 0Chicarelli, Mark论文数: 0 引用数: 0 h-index: 0Fell, Brad论文数: 0 引用数: 0 h-index: 0Fulton, Jennifer论文数: 0 引用数: 0 h-index: 0Guarnieri, Anna论文数: 0 引用数: 0 h-index: 0Haygood, Leyla论文数: 0 引用数: 0 h-index: 0Jalluri, Ravi论文数: 0 引用数: 0 h-index: 0Johnson, Amber论文数: 0 引用数: 0 h-index: 0Mclean, Brent论文数: 0 引用数: 0 h-index: 0Mejia, Max论文数: 0 引用数: 0 h-index: 0Rieger, Rob论文数: 0 引用数: 0 h-index: 0Robinson, John论文数: 0 引用数: 0 h-index: 0Rodriguez, Mareli论文数: 0 引用数: 0 h-index: 0Sullivan, Francis论文数: 0 引用数: 0 h-index: 0Wang, Yang论文数: 0 引用数: 0 h-index: 0Winski, Shannon论文数: 0 引用数: 0 h-index: 0Zhou, YeYun论文数: 0 引用数: 0 h-index: 0
- [3] Identification of a reversible selective FGFR2 clinical development candidate with potency against gatekeeper and molecular brake mutationsMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Fischer, John论文数: 0 引用数: 0 h-index: 0Bouhana, Karyn论文数: 0 引用数: 0 h-index: 0Brizendine, Richard论文数: 0 引用数: 0 h-index: 0Chicarelli, Mark论文数: 0 引用数: 0 h-index: 0Fell, Brad论文数: 0 引用数: 0 h-index: 0Fulton, Jennifer论文数: 0 引用数: 0 h-index: 0Guarnieri, Anna论文数: 0 引用数: 0 h-index: 0Haygood, Leyla论文数: 0 引用数: 0 h-index: 0Jalluri, Ravi论文数: 0 引用数: 0 h-index: 0Johnson, Amber论文数: 0 引用数: 0 h-index: 0Koch, Keith论文数: 0 引用数: 0 h-index: 0Koslov-Davino, Erika论文数: 0 引用数: 0 h-index: 0Mejia, Max论文数: 0 引用数: 0 h-index: 0Rieger, Rob论文数: 0 引用数: 0 h-index: 0Robinson, John论文数: 0 引用数: 0 h-index: 0Rodriguez, Mareli论文数: 0 引用数: 0 h-index: 0Sullivan, Francis论文数: 0 引用数: 0 h-index: 0Wang, Yang论文数: 0 引用数: 0 h-index: 0Winski, Shannon论文数: 0 引用数: 0 h-index: 0Wood, Silas论文数: 0 引用数: 0 h-index: 0Zhou, Yeyun论文数: 0 引用数: 0 h-index: 0
- [4] Discovery and characterization of selective, FGFR1 sparing, inhibitors of FGFR2/3 oncogenic mutations for the treatment of cancersMOLECULAR CANCER THERAPEUTICS, 2021, 20 (12)Dardenne, Etienne论文数: 0 引用数: 0 h-index: 0Padilla, Fernando论文数: 0 引用数: 0 h-index: 0Rasmussen, Sara论文数: 0 引用数: 0 h-index: 0Yang, Shao Ning论文数: 0 引用数: 0 h-index: 0Mentes, Ahmet论文数: 0 引用数: 0 h-index: 0Ogawa, Luisa Shin论文数: 0 引用数: 0 h-index: 0Trombino, Anthony论文数: 0 引用数: 0 h-index: 0Romashko, Darlene论文数: 0 引用数: 0 h-index: 0Chevtsova, Maria论文数: 0 引用数: 0 h-index: 0Thakur, Shalabh论文数: 0 引用数: 0 h-index: 0Buck, Elisabeth论文数: 0 引用数: 0 h-index: 0Roberts, Christopher论文数: 0 引用数: 0 h-index: 0Lucas, Matthew论文数: 0 引用数: 0 h-index: 0Lin, Tai-An论文数: 0 引用数: 0 h-index: 0
- [5] Discovery and characterization of selective, FGFR1-sparing, inhibitors of FGFR2/3 oncogenic mutations for the treatment of cancersANNALS OF ONCOLOGY, 2021, 32 : S15 - S15Dardenne, E.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USAPadilla, F.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USARasmussen, S.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USAYang, S. N.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USAMentes, A.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USAOgawa, L. S.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USAFiorenza, R.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USATrombino, A.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USASmith, S.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USARomashko, D.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USAIshiyama, N.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USAChevtsova, M.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USAThakur, S.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USARosfjord, E.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USABuck, E.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USARoberts, C.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USALucas, M.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, Cambridge, MA USA Black Diamond Therapeut, R&D, New York, NY USALin, T-A.论文数: 0 引用数: 0 h-index: 0机构: Black Diamond Therapeut, R&D, New York, NY USA Black Diamond Therapeut, R&D, New York, NY USA
- [6] Pre-clinical In Vitro and In Vivo Characterization of a Novel EGFR Sparing ErbB2 Inhibitor with Activity Against Oncogenic ErbB2 MutationsEUROPEAN JOURNAL OF CANCER, 2022, 174 : S81 - S81Chicarelli, M. J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USABouhana, K.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USACable, L.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USACrow, M.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAFell, B.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAFischer, J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAFulton, J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAGuarnieri, A.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAJalluri, R.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USARobinson, J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USASullivan, F.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAWinski, S.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAZhou, Y.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USA
- [7] Characterization of two novel oncogenic FGFR2 fusions sensitive to the FGFR-selective inhibitor Debio 1347 in cholangiocarcinomaCANCER RESEARCH, 2015, 75Vaslin, Anne论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandRigotti, Stefania论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandLembrez, Nathalie论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandVuagniaux, Gregoire论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandMoulon, Corinne论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandTanaka, Hiroaki论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, Switzerland
- [8] Pre-clinical characterization of potent and selective next-generation RET inhibitors.CANCER RESEARCH, 2021, 81 (13)Kolakowski, Gabrielle R.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USAAnderson, Erin D.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USABallard, Joshua A.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USABrandhuber, Barbara J.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USACondroski, Kevin R.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USAGomez, Eliana B.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USAIrvin, Thomas C.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USAKumar, Manoj论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USAPatel, Nisha A.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USAWatson, Faith D.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USAAndrews, Steven W.论文数: 0 引用数: 0 h-index: 0机构: Loxo Oncol Lilly, Boulder, CO USA Loxo Oncol Lilly, Boulder, CO USA
- [9] Discovery of highly selective DUB inhibitors with in vivo pre-clinical anti-tumor activityCANCER RESEARCH, 2015, 75Jacq, Xavier论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandMartin, Niall M. B.论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandSmith, Lisa论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandHarrigan, Jeanine论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandKnights, Charlotte论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandRobinson, Helen论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandOfir-Rosenfeld, Yaara论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandCranston, Aaron论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandKemp, Mark I.论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, EnglandJackson, Stephen P.论文数: 0 引用数: 0 h-index: 0机构: MISSION Therapeut Ltd, Cambridge, England MISSION Therapeut Ltd, Cambridge, England
- [10] Genomic and clinical characterization of non-small cell lung cancer (NSCLC) patients harboring mutations in FGFR2 and FGFR3ANNALS OF ONCOLOGY, 2019, 30Scheffler, M.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyChanra, T.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyKron, A.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyKoleczko, S.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyAbdulla, D. S. Y.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyIhle, M. A.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Pathol, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyHolzem, A.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyRiedel, R.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyMichels, S.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyFischer, R. N.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyMerkelbach-Bruse, S.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Pathol, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyBuettner, R.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Pathol, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyNogova, L.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, GermanyWolf, J.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Koln, Ctr Integrated Oncol, Dept Internal Med 1, Cologne, Germany Uniklin Koln, Dept Internal Med 1, Cologne, Germany