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- [21] Discovery of novel HIV integrase inhibitors part 2: Selection and evaluation of an azabicyclic carbamoyl pyridone inhibitor as a pre-clinical candidateABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 245Akiyama, Toshiyuki论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, JapanJohns, Brian A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC USA Shionogi & Co Ltd, Osaka, JapanTaoda, Yoshiyuki论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, JapanYoshida, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, JapanTaishi, Teruhiko论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, JapanKawasuji, Takashi论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, JapanMurai, Hitoshi论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, JapanYoshinaga, Tomokazu论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, JapanSato, Akihiko论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, JapanFujiwara, Tamio论文数: 0 引用数: 0 h-index: 0机构: Shionogi & Co Ltd, Osaka, Japan Shionogi & Co Ltd, Osaka, Japan
- [22] Pre-clinical characterization of CX-4945, a potent and selective small molecule inhibitor of CK2 for the treatment of cancerMOLECULAR AND CELLULAR BIOCHEMISTRY, 2011, 356 (1-2) : 37 - 43Pierre, Fabrice论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAChua, Peter C.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAO'Brien, Sean E.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USASiddiqui-Jain, Adam论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USABourbon, Pauline论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAHaddach, Mustapha论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAMichaux, Jerome论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USANagasawa, Johnny论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USASchwaebe, Michael K.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAStefan, Eric论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAVialettes, Anne论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAWhitten, Jeffrey P.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAChen, Ta Kung论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USADarjania, Levan论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAStansfield, Ryan论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USABliesath, Joshua论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USADrygin, Denis论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAHo, Caroline论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAOmori, May论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAProffitt, Chris论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAStreiner, Nicole论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USARice, William G.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USARyckman, David M.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USAAnderes, Kenna论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut, San Diego, CA 92121 USA Cylene Pharmaceut, San Diego, CA 92121 USA
- [23] Pre-clinical characterization of CX-4945, a potent and selective small molecule inhibitor of CK2 for the treatment of cancerMolecular and Cellular Biochemistry, 2011, 356 : 37 - 43Fabrice Pierre论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Peter C. Chua论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Sean E. O’Brien论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Adam Siddiqui-Jain论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Pauline Bourbon论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Mustapha Haddach论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Jerome Michaux论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Johnny Nagasawa论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Michael K. Schwaebe论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Eric Stefan论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Anne Vialettes论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Jeffrey P. Whitten论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Ta Kung Chen论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Levan Darjania论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Ryan Stansfield论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Joshua Bliesath论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Denis Drygin论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Caroline Ho论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,May Omori论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Chris Proffitt论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Nicole Streiner论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,William G. Rice论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,David M. Ryckman论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,Kenna Anderes论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceuticals,
- [24] Discovery of Novel 2,4,5-Trisubstituted Pyrimidine Derivatives as Potent and Selective FGFR Inhibitors against Gatekeeper Mutants for the Treatment of NSCLCJOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (05) : 5907 - 5925Zhang, Jianxia论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaWang, Yi论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaWang, Mengying论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaWang, Peipei论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaYan, Hao论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaWang, Dalong论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaZheng, Jiahao论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaLi, Bin论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaChen, Chaoyue论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaCao, Di论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaZheng, Xiaohui论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaLi, Xiaokun论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaWang, Kun论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R ChinaLiu, Zhiguo论文数: 0 引用数: 0 h-index: 0机构: Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China Wenzhou Med Univ, Sch Pharmaceut Sci, State Key Lab Macromol Drugs & Large scale Prepara, Wenzhou 325035, Zhejiang, Peoples R China
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- [26] Is CNS availability for oncology a no-brainer? Discovery of PF-06463922, a novel small molecule inhibitor of ALK/ROS1 with pre-clinical brain availability and broad spectrum potency against ALK-resistant mutationsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 247Johnson, Ted W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USABailey, Simon论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USABurke, Benjamin J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USACollins, Michael R.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USACui, J. Jean论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USADeal, Judy论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USADeng, Ye-Li论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAGukasyan, Hovhannes论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAHe, Mingying论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAHoffman, Jacqui论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAHoffman, Robert L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAHuang, Qinhua论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAKania, Robert S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAKath, John C.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USALe, Phuong T.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAMcTigue, Michele论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAPalmer, Cynthia L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USARichardson, Paul F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USASach, Neal W.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAShen, Hong论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USASmith, Graham L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USASrirangam, Jay论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAZhu, Huichun论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAZhu, Jinjiang论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USADinh, Dac论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAEngstrom, Lars论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAHu, Wenyue论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USALam, Hieu论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USALam, Justine L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USALi, Qiuhua论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USASmeal, Tod论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USATimofeevski, Sergei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USALu, Melissa West论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAYamazaki, Shinji论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAZou, Helen Y.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USAEdwards, Martin P.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, San Diego, CA USA Pfizer Inc, San Diego, CA USA
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