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- [1] Identification of a reversible selective FGFR2 clinical development candidate with potency against gatekeeper and molecular brake mutationsMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Fischer, John论文数: 0 引用数: 0 h-index: 0Bouhana, Karyn论文数: 0 引用数: 0 h-index: 0Brizendine, Richard论文数: 0 引用数: 0 h-index: 0Chicarelli, Mark论文数: 0 引用数: 0 h-index: 0Fell, Brad论文数: 0 引用数: 0 h-index: 0Fulton, Jennifer论文数: 0 引用数: 0 h-index: 0Guarnieri, Anna论文数: 0 引用数: 0 h-index: 0Haygood, Leyla论文数: 0 引用数: 0 h-index: 0Jalluri, Ravi论文数: 0 引用数: 0 h-index: 0Johnson, Amber论文数: 0 引用数: 0 h-index: 0Koch, Keith论文数: 0 引用数: 0 h-index: 0Koslov-Davino, Erika论文数: 0 引用数: 0 h-index: 0Mejia, Max论文数: 0 引用数: 0 h-index: 0Rieger, Rob论文数: 0 引用数: 0 h-index: 0Robinson, John论文数: 0 引用数: 0 h-index: 0Rodriguez, Mareli论文数: 0 引用数: 0 h-index: 0Sullivan, Francis论文数: 0 引用数: 0 h-index: 0Wang, Yang论文数: 0 引用数: 0 h-index: 0Winski, Shannon论文数: 0 引用数: 0 h-index: 0Wood, Silas论文数: 0 引用数: 0 h-index: 0Zhou, Yeyun论文数: 0 引用数: 0 h-index: 0
- [2] TYRA-200: Potent Against FGFR2 Fusions, Molecular Brake Mutations and Gatekeeper ResistanceEUROPEAN JOURNAL OF CANCER, 2022, 174 : S16 - S16Allen, E.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USABalcer, A.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USABensen, D.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USABurn, T.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USAHoffman, I.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USAHudkins, R.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Chem, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USAIyer, S.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USANeal, M.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USANelson, K.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USAOcchino, C.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Chem, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USAPatel, P.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Chem, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USAStarrett, J.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USASwanson, R.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USAYe, Q.论文数: 0 引用数: 0 h-index: 0机构: Tyra Biosci, Biol, Carlsbad, CA USA Tyra Biosci, Biol, Carlsbad, CA USA
- [3] In Vivo Pre-clinical characterization of a Novel Series of FGFR2 Selective Inhibitors with Potency Against Clinically Relevant MutationsEUROPEAN JOURNAL OF CANCER, 2022, 174 : S81 - S81Fischer, J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USABouhana, K.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAChicarelli, M. J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USADahlke, J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAFell, B.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAFulton, J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAGuarnieri, A.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAHaygood, L.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAJalluri, R.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAJohnson, A.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAMcLean, B.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAMax, M.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USARieger, R.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USARobinson, J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USARodriguez, M.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USASullivan, F.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAWang, Y.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAWinski, S.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USAZhou, Y.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Res Dev, Boulder, CO USA Cogent Biosci, Res Dev, Boulder, CO USA
- [4] ctDNA-based genomic landscape analysis to evaluate molecular brake and gatekeeper mutations in FGFR2 alterationsJOURNAL OF CLINICAL ONCOLOGY, 2023, 41 (16)Severson, Paul论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma, San Francisco, CA USASytnikova, Julia论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma, San Francisco, CA USAMohan, Adithi论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma, San Francisco, CA USAZhang, Nicole论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma, San Francisco, CA USADonderici, Elifnur Yay论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma, San Francisco, CA USAWilliams, Richard Thomas论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma, San Francisco, CA USA
- [5] Pre-clinical characterization of a novel series of FGFR2 selective inhibitors with potency against clinically relevant mutationsCANCER RESEARCH, 2022, 82 (12)Fischer, John论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USABouhana, Karyn论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAChicarelli, Mark J.论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USADahlke, Josh论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAFell, Brad论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAFulton, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAGuarnieri, Anna论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAJalluri, Ravi论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAJohnson, Amber论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAMclean, Brent论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAMejia, Max论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USARieger, Rob论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USARobinson, John论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USARodriguez, Mareli论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USASullivan, Francis论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAWang, Yang论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAWinski, Shannon论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USAZhou, Yeyun论文数: 0 引用数: 0 h-index: 0机构: Cogent Biosci, Cambridge, MA USA Cogent Biosci, Cambridge, MA USA
- [6] Regulation of the Molecular Brake Region in FGFR2 KinaseBIOPHYSICAL JOURNAL, 2015, 108 (02) : 530A - 530AKarp, Jerome M.论文数: 0 引用数: 0 h-index: 0机构: Yeshiva Univ, Albert Einstein Coll Med, Biochem, Bronx, NY USA Yeshiva Univ, Albert Einstein Coll Med, Biochem, Bronx, NY USACowburn, David论文数: 0 引用数: 0 h-index: 0机构: Yeshiva Univ, Albert Einstein Coll Med, Biochem, Bronx, NY USA Yeshiva Univ, Albert Einstein Coll Med, Biochem, Bronx, NY USA
- [7] RLY-4008, the First Highly Selective FGFR2 Inhibitor with Activity across FGFR2 Alterations and Resistance MutationsCANCER DISCOVERY, 2023, 13 (09) : 2012 - 2031Subbiah, Vivek论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASahai, Vaibhav论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ann Arbor, MI 48109 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAMaglic, Dejan论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USABruderek, Kamil论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAToure, B. Barry论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAZhao, Songping论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAValverde, Roberto论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAO'Hearn, Patrick J.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAMoustakas, Demetri T.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASchoenherr, Heike论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAGerami-Moayed, Nastaran论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USATaylor, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAHudson, Brandi M.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAHoude, Damian J.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAPal, Debjani论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAFoster, Lindsey论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAGunaydin, Hakan论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAAyaz, Pelin论文数: 0 引用数: 0 h-index: 0机构: DE Shaw Res, New York, NY USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASharon, Dina A.论文数: 0 引用数: 0 h-index: 0机构: DE Shaw Res, New York, NY USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAGoyal, Lipika论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA 02114 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASchram, Alison M.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAKamath, Suneel论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Taussig Canc Inst, Cleveland, OH 44106 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASherwin, Cori Ann论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASchmidt-Kittler, Oleg论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAJen, Kai Yu论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USARicard, Fabien论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAWolf, Beni B.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAShaw, David E.论文数: 0 引用数: 0 h-index: 0机构: DE Shaw Res, New York, NY USA Columbia Univ, Dept Biochem & Mol Biophys, New York, NY USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USABergstrom, Donald A.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAWatters, James论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USACasaletto, Jessica B.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA
- [8] Regulation of the "molecular brake" region in FGFR2 kinase.MOLECULAR BIOLOGY OF THE CELL, 2014, 25Karp, J. M.论文数: 0 引用数: 0 h-index: 0机构: Albert Einstein Coll Med, Bronx, NY 10467 USA Albert Einstein Coll Med, Bronx, NY 10467 USACowburn, D.论文数: 0 引用数: 0 h-index: 0机构: Albert Einstein Coll Med, Bronx, NY 10467 USA Albert Einstein Coll Med, Bronx, NY 10467 USA
- [9] Activity of KIN-3248, a next-generation pan-FGFR inhibitor, against acquired FGFR-gatekeeper and molecular-brake drug resistance mutationsJOURNAL OF CLINICAL ONCOLOGY, 2022, 40 (04)Franovic, Aleksandra论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USAMohan, Adithi论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USAUryu, Sean论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USAWu, Qibiao论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USAJiang, Ping论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USAMiller, Nichol论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USATyhonas, John论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USATimple, Noelito论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USASeverson, Paul论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USAKania, Robert论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USAMurphy, Eric论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USABardeesy, Nabeel论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USAMartin, Eric论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharma Inc, San Diego, CA USA
- [10] Preclinical characterization of a Selective FGFR2/3 inhibitor, GSC000829EUROPEAN JOURNAL OF CANCER, 2024, 211 : S52 - S52Han, T.论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R ChinaFu, D.论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R ChinaCheng, T.论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R ChinaXia, Y.论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R ChinaHu, Z.论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R ChinaYang, F.论文数: 0 引用数: 0 h-index: 0机构: Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R China Changchun GeneSci Pharmaceut Co Ltd, Chem Drug Res & Dev, Shanghai, Peoples R China