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- [1] Preclinical characterization of alofanib, a novel allosteric FGFR2 inhibitorANNALS OF ONCOLOGY, 2016, 27Tsimafeyeu, I.论文数: 0 引用数: 0 h-index: 0机构: Kidney Canc Res Bur, Moscow Off, Moscow, Russia Kidney Canc Res Bur, Moscow Off, Moscow, RussiaStepanova, E.论文数: 0 引用数: 0 h-index: 0机构: NN Blokhin Russian Canc Res Ctr, Lab Biomarkers & Tumor Angiogenesis, Moscow, Russia Kidney Canc Res Bur, Moscow Off, Moscow, RussiaKhochenkov, D.论文数: 0 引用数: 0 h-index: 0机构: NN Blokhin Russian Canc Res Ctr, Lab Biomarkers & Tumor Angiogenesis, Moscow, Russia Kidney Canc Res Bur, Moscow Off, Moscow, RussiaMurillo, G.论文数: 0 引用数: 0 h-index: 0机构: IIT, Res Inst, Chicago, IL 60616 USA Kidney Canc Res Bur, Moscow Off, Moscow, RussiaLapina, N.论文数: 0 引用数: 0 h-index: 0机构: Fed Med Biol Agcy, Inst Toxicol, Lab Toxicol & Pharmacol, St Petersburg, Russia Kidney Canc Res Bur, Moscow Off, Moscow, RussiaGavrilova, E.论文数: 0 引用数: 0 h-index: 0机构: Ruspharmtech LLC, Spb Off, St Petersburg, Russia Kidney Canc Res Bur, Moscow Off, Moscow, RussiaByakhov, M.论文数: 0 引用数: 0 h-index: 0机构: Moscow Clin & Res Ctr, Dept Chemotherapy, Moscow, Russia Kidney Canc Res Bur, Moscow Off, Moscow, RussiaTjulandin, S.论文数: 0 引用数: 0 h-index: 0机构: NN Blokhin Russian Canc Res Ctr, Dept Clin Pharmacol & Chemotherapy, Moscow, Russia Kidney Canc Res Bur, Moscow Off, Moscow, Russia
- [2] Toxicity of selective allosteric FGFR2 inhibition in preclinical studiesCANCER RESEARCH, 2016, 76Lapina, Nataliya V.论文数: 0 引用数: 0 h-index: 0Melikhova, Marina V.论文数: 0 引用数: 0 h-index: 0Vakunenkova, Olga A.论文数: 0 引用数: 0 h-index: 0Kashuro, Vadim A.论文数: 0 引用数: 0 h-index: 0
- [3] Preclinical characterization of the selective FGFR inhibitor INCB054828CANCER RESEARCH, 2015, 75Liu, Phillip C. C.论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAWu, Liangxing论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAKoblish, Holly论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USABowman, Kevin论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAZhang, Yue论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAKlabe, Ronald论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USALeffet, Lynn论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USADiMatteo, Darlise论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USARupar, Mark论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAGallagher, Karen论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAHansbury, Michael论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAZhang, Colin论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAHe, Chunhong论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USACollier, Paul论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USACovington, Maryanne论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAWynn, Richard论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAYeleswaram, Swamy论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAVaddi, Kris论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USABurn, Timothy论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAYao, Wenqing论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAHuber, Reid论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAScherle, Peggy论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USAHollis, Gregory论文数: 0 引用数: 0 h-index: 0机构: Incyte Corp, Wilmington, DE USA Incyte Corp, Wilmington, DE USA
- [4] Discovery of a highly potent and selective FGFR2 inhibitor for FGFR2-driven cancersCANCER RESEARCH, 2024, 84 (06)Li, Wenqian论文数: 0 引用数: 0 h-index: 0Liu, Bin论文数: 0 引用数: 0 h-index: 0Wang, Junmei论文数: 0 引用数: 0 h-index: 0Yin, Tinggui论文数: 0 引用数: 0 h-index: 0Yu, Kuo-Long论文数: 0 引用数: 0 h-index: 0Kumar, Sanjeev论文数: 0 引用数: 0 h-index: 0Wen, Zhiming论文数: 0 引用数: 0 h-index: 0Zhao, Genshi论文数: 0 引用数: 0 h-index: 0Pan, Weitao论文数: 0 引用数: 0 h-index: 0
- [5] In vivo characterization of a selective FGFR2 inhibitor with potency against gatekeeper and molecular brake mutationsCANCER RESEARCH, 2023, 83 (07)Fischer, John论文数: 0 引用数: 0 h-index: 0Bouhana, Karyn论文数: 0 引用数: 0 h-index: 0Chicarelli, Mark论文数: 0 引用数: 0 h-index: 0Fell, Brad论文数: 0 引用数: 0 h-index: 0Fulton, Jennifer论文数: 0 引用数: 0 h-index: 0Guarnieri, Anna论文数: 0 引用数: 0 h-index: 0Haygood, Leyla论文数: 0 引用数: 0 h-index: 0Jalluri, Ravi论文数: 0 引用数: 0 h-index: 0Johnson, Amber论文数: 0 引用数: 0 h-index: 0Mclean, Brent论文数: 0 引用数: 0 h-index: 0Mejia, Max论文数: 0 引用数: 0 h-index: 0Rieger, Rob论文数: 0 引用数: 0 h-index: 0Robinson, John论文数: 0 引用数: 0 h-index: 0Rodriguez, Mareli论文数: 0 引用数: 0 h-index: 0Sullivan, Francis论文数: 0 引用数: 0 h-index: 0Wang, Yang论文数: 0 引用数: 0 h-index: 0Winski, Shannon论文数: 0 引用数: 0 h-index: 0Zhou, YeYun论文数: 0 引用数: 0 h-index: 0
- [6] Characterization of two novel oncogenic FGFR2 fusions sensitive to the FGFR-selective inhibitor Debio 1347 in cholangiocarcinomaCANCER RESEARCH, 2015, 75Vaslin, Anne论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandRigotti, Stefania论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandLembrez, Nathalie论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandVuagniaux, Gregoire论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandMoulon, Corinne论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, SwitzerlandTanaka, Hiroaki论文数: 0 引用数: 0 h-index: 0机构: Debiopharm Int SA, Lausanne, Switzerland Debiopharm Int SA, Lausanne, Switzerland
- [7] RLY-4008, the First Highly Selective FGFR2 Inhibitor with Activity across FGFR2 Alterations and Resistance MutationsCANCER DISCOVERY, 2023, 13 (09) : 2012 - 2031Subbiah, Vivek论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASahai, Vaibhav论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ann Arbor, MI 48109 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAMaglic, Dejan论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USABruderek, Kamil论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAToure, B. Barry论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAZhao, Songping论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAValverde, Roberto论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAO'Hearn, Patrick J.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAMoustakas, Demetri T.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASchoenherr, Heike论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAGerami-Moayed, Nastaran论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USATaylor, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAHudson, Brandi M.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAHoude, Damian J.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAPal, Debjani论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAFoster, Lindsey论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAGunaydin, Hakan论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAAyaz, Pelin论文数: 0 引用数: 0 h-index: 0机构: DE Shaw Res, New York, NY USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASharon, Dina A.论文数: 0 引用数: 0 h-index: 0机构: DE Shaw Res, New York, NY USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAGoyal, Lipika论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA 02114 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASchram, Alison M.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAKamath, Suneel论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Taussig Canc Inst, Cleveland, OH 44106 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASherwin, Cori Ann论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USASchmidt-Kittler, Oleg论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAJen, Kai Yu论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USARicard, Fabien论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAWolf, Beni B.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAShaw, David E.论文数: 0 引用数: 0 h-index: 0机构: DE Shaw Res, New York, NY USA Columbia Univ, Dept Biochem & Mol Biophys, New York, NY USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USABergstrom, Donald A.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAWatters, James论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USACasaletto, Jessica B.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut Inc, 399 Binney St, Cambridge, MA 02139 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA
- [8] Discovery and preclinical characterization of ISM8001, a covalent and selective FGFR2/FGFR3 dual inhibitor with strong monotherapy anti-tumor activity against advanced solid tumorsCANCER RESEARCH, 2024, 84 (06)Zhang, Yihong论文数: 0 引用数: 0 h-index: 0Wang, Yazhou论文数: 0 引用数: 0 h-index: 0Cai, Xin论文数: 0 引用数: 0 h-index: 0Liu, Jinxin论文数: 0 引用数: 0 h-index: 0Cui, Hui论文数: 0 引用数: 0 h-index: 0Qiao, Junwen论文数: 0 引用数: 0 h-index: 0Lin, Xiaoxia论文数: 0 引用数: 0 h-index: 0Ding, Xiao论文数: 0 引用数: 0 h-index: 0Bavadekar, Supriya论文数: 0 引用数: 0 h-index: 0Rao, Sujata论文数: 0 引用数: 0 h-index: 0Zhang, Man论文数: 0 引用数: 0 h-index: 0Ren, Feng论文数: 0 引用数: 0 h-index: 0Zhavoronkov, Alex论文数: 0 引用数: 0 h-index: 0
- [9] Preclinical activity of the VEGFR, FGFR and PDGFR inhibitor lucitanib in FGFR2 aberrant endometrial and gastric cancer modelsEUROPEAN JOURNAL OF CANCER, 2014, 50 : 110 - 110Guffanti, F.论文数: 0 引用数: 0 h-index: 0机构: IRCCS Mario Negri Inst Pharmacol Res, Milan, Italy IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalyChila, R.论文数: 0 引用数: 0 h-index: 0机构: IRCCS Mario Negri Inst Pharmacol Res, Milan, Italy IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalyBello, E.论文数: 0 引用数: 0 h-index: 0机构: IRCCS Mario Negri Inst Pharmacol Res, Milan, Italy IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalyCeriani, L.论文数: 0 引用数: 0 h-index: 0机构: IRCCS Mario Negri Inst Pharmacol Res, Milan, Italy IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalyZangarini, M.论文数: 0 引用数: 0 h-index: 0机构: IRCCS Mario Negri Inst Pharmacol Res, Milan, Italy IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalyZucchetti, M.论文数: 0 引用数: 0 h-index: 0机构: IRCCS Mario Negri Inst Pharmacol Res, Milan, Italy IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalySaba, C.论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Int Servier, Suresnes, France IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalyJacquet-Bescond, A.论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Int Servier, Suresnes, France IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalyPierrat, M.论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Int Servier, Suresnes, France IRCCS Mario Negri Inst Pharmacol Res, Milan, ItalyDamia, G.论文数: 0 引用数: 0 h-index: 0机构: IRCCS Mario Negri Inst Pharmacol Res, Milan, Italy IRCCS Mario Negri Inst Pharmacol Res, Milan, Italy
- [10] Design and preclinical profile of CH5183284/Debio 1347, a novel orally available and selective FGFR inhibitor acting on a gatekeeper mutant of FGFR2CANCER RESEARCH, 2014, 74 (19)Ebiike, Hirosato论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanTaka, Naoki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanNakanishi, Yoshito论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanAkiyama, Nukinori论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanSawamura, Fumie论文数: 0 引用数: 0 h-index: 0机构: Chugai Res Inst Med Sci Inc, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanMorikami, Kenji论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanMatsushita, Masayuki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanOhmori, Masayuki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanTakami, Kyouko论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanHyohdoh, Ikumi论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanKohchi, Masami论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanHayase, Tadakatsu论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanNishii, Hiroki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanIshii, Nobuya论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, JapanMatsuoka, Hiroharu论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Shizuoka, Japan Chugai Pharmaceut Co Ltd, Shizuoka, Japan