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- [21] FGFR2/3 in urothelial carcinomaPATHOLOGIE, 2024, 45 (06): : 409 - 411Rose, Michael论文数: 0 引用数: 0 h-index: 0机构: Uniklin Ulm, Inst Pathol, Albert Einstein Allee 23, D-89081 Ulm, Germany Uniklin RWTH Aachen, Inst Pathol, Aachen, Germany Uniklin Ulm, Inst Pathol, Albert Einstein Allee 23, D-89081 Ulm, GermanyGaisa, Nadine T.论文数: 0 引用数: 0 h-index: 0机构: Uniklin Ulm, Inst Pathol, Albert Einstein Allee 23, D-89081 Ulm, Germany Uniklin RWTH Aachen, Inst Pathol, Aachen, Germany Uniklin Ulm, Inst Pathol, Albert Einstein Allee 23, D-89081 Ulm, Germany
- [22] Alofanib, a novel allosteric FGFR2 inhibitor, shows potent antitumor activity in ovarian cancer with FGFR2 expressionCANCER RESEARCH, 2015, 75Tjulandin, Sergei论文数: 0 引用数: 0 h-index: 0机构: NN Blokhin Russian Canc Res Ctr, Moscow, Russia NN Blokhin Russian Canc Res Ctr, Moscow, RussiaByakhov, Mikhail论文数: 0 引用数: 0 h-index: 0机构: Moscow Clin Res Ctr, Moscow, Russia NN Blokhin Russian Canc Res Ctr, Moscow, RussiaStepanova, Evgenia论文数: 0 引用数: 0 h-index: 0机构: NN Blokhin Russian Canc Res Ctr, Moscow, Russia NN Blokhin Russian Canc Res Ctr, Moscow, RussiaKhochenkov, Dmitry论文数: 0 引用数: 0 h-index: 0机构: NN Blokhin Russian Canc Res Ctr, Moscow, Russia NN Blokhin Russian Canc Res Ctr, Moscow, RussiaHarrison, Daniel论文数: 0 引用数: 0 h-index: 0机构: Altogen Labs, Austin, TX USA NN Blokhin Russian Canc Res Ctr, Moscow, RussiaTsimafeyeu, Ilya论文数: 0 引用数: 0 h-index: 0机构: Russian Pharmaceut Technol, Moscow, Russia NN Blokhin Russian Canc Res Ctr, Moscow, Russia
- [23] From Fragment to Lead: De Novo Design and Development toward a Selective FGFR2 InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (02) : 1481 - 1504Turner, Lewis D.论文数: 0 引用数: 0 h-index: 0机构: Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, England Biosplice Therapeut Inc, 9360 Towne Ctr Dr, San Diego, CA 92121 USA Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, England论文数: 引用数: h-index:机构:Hubball, Ryan A.论文数: 0 引用数: 0 h-index: 0机构: Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, England Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, EnglandOrritt, Kyle M.论文数: 0 引用数: 0 h-index: 0机构: Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, England Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, EnglandLin, Chi-Chuan论文数: 0 引用数: 0 h-index: 0机构: Univ Leeds, Astbury Ctr Struct Mol Biol, Inst Mol & Cellular Biol, Leeds LS2 9JT, W Yorkshire, England Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, EnglandBurns, Julie E.论文数: 0 引用数: 0 h-index: 0机构: Univ Leeds, Leeds Inst Med Res St Jamess, Leeds LS9 7TF, W Yorkshire, England Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, EnglandKnowles, Margaret A.论文数: 0 引用数: 0 h-index: 0机构: Univ Leeds, Leeds Inst Med Res St Jamess, Leeds LS9 7TF, W Yorkshire, England Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, EnglandFishwick, Colin W. G.论文数: 0 引用数: 0 h-index: 0机构: Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, England Univ Leeds, Sch Chem, Leeds LS2 9JT, W Yorkshire, England
- [24] Identifying FGFR2 fusions/rearrangements in cholangiocarcinoma patients using a novel cfDNA algorithm for treatment with RLY-4008, a highly selective irreversible FGFR2 inhibitorEUROPEAN JOURNAL OF CANCER, 2022, 174 : S116 - S116Schram, A.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USABorad, M.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin Scottsdale, Med Oncol, PPDS, Phoenix, AZ USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USASahai, V.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Gastrointestinal Med Oncol, Ann Arbor, MI USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAKamath, S.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Hematol & Med Oncol, Taussig Canc Inst, Cleveland, OH USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAKim, R.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Med Gastrointestinal Oncol, Tampa, FL USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USALiao, C. Y. A.论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Hematol & Oncol, Med Ctr, Chicago, IL USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAOh, D. Y.论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ Hosp, Hemato Oncol, Seoul, South Korea Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAPonz-Sarvise, M.论文数: 0 引用数: 0 h-index: 0机构: Univ Navarra Clin, Med Oncol, Pamplona, Spain Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAYachnin, J.论文数: 0 引用数: 0 h-index: 0机构: Karolinska Univ Solna, Early Clin, Trial Unit, Stockholm, Sweden Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAShell, S. A.论文数: 0 引用数: 0 h-index: 0机构: Biopharma Collaborat, Guardant Hlth, Palo Alto, CA USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USACassier, P.论文数: 0 引用数: 0 h-index: 0机构: Ctr Leon Berard, Med Oncol, Lyon, France Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USADotan, E.论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Gastrointestinal Med Oncol, Philadelphia, PA USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAFlorou, V.论文数: 0 引用数: 0 h-index: 0机构: Univ Utah, Oncol, Huntsman Canc Inst, PPDS, Salt Lake City, UT USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAMoreno, V.论文数: 0 引用数: 0 h-index: 0机构: START MADRID Hosp Univ Fdn Jimenez Diaz, Clin Res, Madrid, Spain Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAPark, J. O.论文数: 0 引用数: 0 h-index: 0机构: Samsung Med Ctr, Hematol Oncol, PPDS, Seoul, South Korea Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USATai, D.论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Med Oncol, Singapore, Singapore Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USASchmidt-Kittler, O.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut, Translat Med, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAFerte, C.论文数: 0 引用数: 0 h-index: 0机构: Relay Therapeut, Clin Dev, Cambridge, MA USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USAGoyal, L.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Hematol Oncol, Boston, MA USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USASubbiah, V.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Invest Canc Therapeut, Houston, TX USA Mem Sloan Kettering Canc Ctr, Med Oncol, New York, NY USA
- [25] Preclinical Combination Studies of an FGFR2 Targeted Thorium-227 Conjugate and the ATR Inhibitor BAY 1895344INTERNATIONAL JOURNAL OF RADIATION ONCOLOGY BIOLOGY PHYSICS, 2019, 105 (02): : 410 - 422Wickstroem, Katrine论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwayHagemann, Urs B.论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Pharma, Preclin Res, Berlin, Germany Bayer AS, Thorium Conjugate Res, Oslo, NorwayKristian, Alexander论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwayEllingsen, Christine论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwaySommer, Anette论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Pharma, Preclin Res, Berlin, Germany Bayer AS, Thorium Conjugate Res, Oslo, NorwayEllinger-Ziegelbauer, Heidrun论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Pharma, Translat Sci, Wuppertal, Germany Bayer AS, Thorium Conjugate Res, Oslo, NorwayWirnitzer, Uta论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Pharma, Translat Sci, Wuppertal, Germany Bayer AS, Thorium Conjugate Res, Oslo, NorwayHagelin, Else-Marie论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwayLarsen, Aasmund论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwaySmeets, Roger论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwayBjerke, Roger M.论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwayKarlsson, Jenny论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwayRyan, Olav B.论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, NorwayWengner, Antje M.论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Pharma, Preclin Res, Berlin, Germany Bayer AS, Thorium Conjugate Res, Oslo, NorwayLinden, Lars论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Pharma, Preclin Res, Wuppertal, Germany Bayer AS, Thorium Conjugate Res, Oslo, NorwayMumberg, Dominik论文数: 0 引用数: 0 h-index: 0机构: Bayer AG, Pharma, Preclin Res, Berlin, Germany Bayer AS, Thorium Conjugate Res, Oslo, NorwayCuthbertson, Alan S.论文数: 0 引用数: 0 h-index: 0机构: Bayer AS, Thorium Conjugate Res, Oslo, Norway Bayer AS, Thorium Conjugate Res, Oslo, Norway
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- [29] Discovery of LHQ490 as a highly selective fibroblast growth factor receptor 2 (FGFR2) inhibitorEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 272Li, Huiqiong论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaKe, Ran论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, 345 Lingling Rd, Shanghai 200032, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaZhou, Yang论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Chinese Minist Educ MOE,Coll Pharm, 855 Xingye Ave East, Guangzhou 511400, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaChang, Shaohua论文数: 0 引用数: 0 h-index: 0机构: Kinoteck Therapeut CO LTD, 6 Lane 333,Huaxia East Rd, Shanghai 202110, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaWang, Jie论文数: 0 引用数: 0 h-index: 0机构: Jinan Univ, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Chinese Minist Educ MOE,Coll Pharm, 855 Xingye Ave East, Guangzhou 511400, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaSu, Chen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Adv Res Inst, Natl Facil Prot Sci Shanghai, Shanghai 201210, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaWu, Pinglian论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaYang, Bowen论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaWang, Zhen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, 345 Lingling Rd, Shanghai 200032, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaDing, Ke论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, 345 Lingling Rd, Shanghai 200032, Peoples R China Jinan Univ, Int Cooperat Lab Tradit Chinese Med Modernizat & I, Guangzhou City Key Lab Precis Chem Drug Dev, Chinese Minist Educ MOE,Coll Pharm, 855 Xingye Ave East, Guangzhou 511400, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R ChinaMa, Dawei论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R China Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Chem Biol, 345 Lingling Rd, Shanghai 200032, Peoples R China East China Normal Univ, Chang Kung Chuang Inst, Sch Chem & Mol Engn, 500 Dongchuan Rd, Shanghai 200241, Peoples R China
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