Novel synthesis of C-3-(hetero)aryl [1,2,3]triazolo[1,5-a]pyridines using the Stille reaction

被引：4

作者：

Germain, Herve ^{[1
]}

Harris, Craig S. ^{[1
]}

Lebraud, Honorine ^{[1
]}

机构：

[1] AstraZeneca, Ctr Rech, ZI Pompelle, F-51689 Reims 2, France

来源：

TETRAHEDRON LETTERS | 2011年 / 52卷 / 48期

关键词：

1,2,3]Triazolo[1,5-a]pyridine; Stille cross-coupling reaction; Microwave-assisted organic synthesis (MAOS); TRIAZOLOPYRIDINES; HYDRAZONES; OXIDATION; HALOPYRIMIDINES;

D O I：

10.1016/j.tetlet.2011.09.052

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Herein, we report a novel and high yielding approach for the preparation of the first C-3-organometallic substituted [1,2,3]triazolo[1,5-a]pyridine and its application to the Stille reaction using MAOS. (C) 2011 Elsevier Ltd. All rights reserved.

引用

页码：6376 / 6378

页数：3

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