Synthesis of Novel Polyazinyl-Substituted Triazolopyridines from [1,2,3]Triazolo[1,5-a]pyridines

被引：4
|
作者：
Adam, Rosa [1 ]
Abarca, Belen [1 ]
Ballesteros, Rafael [1 ]
机构：
[1] Univ Valencia, Fac Farm, Dept Quim Organ, Avda Vicente Andres Estelles S-N, Valencia 46100, Spain
来源：
SYNTHESIS-STUTTGART | 2017年 / 49卷 / 22期
关键词：
triazolopyridines; diazines; triazines; lithiation reactions; polynitrogenated ligands; RING-CHAIN ISOMERIZATION; ANTILEISHMANIAL ACTIVITY; ANTIBACTERIAL ACTIVITY; COORDINATION POLYMERS; BETA-CYCLODEXTRIN; AQUEOUS-SOLUTION; THEORETICAL DFT; LIGANDS; CHEMISTRY; 1,2,3-TRIAZOLES;
D O I：
10.1055/s-0036-1588525
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A series of 7-azinyl-substituted triazolopyridines and 3-(6-azinyl-substituted 2-pyridyl)triazolopyridines were synthesized by addition of the corresponding 3-substituted 7-lithiotriazolopyridine to pyrimidine, pyrazine, pyridazine, and 1,3,5-triazine respectively, followed by hydrolysis and oxidation.
引用
收藏
页码：5059 / 5066
页数：8
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