Novel synthesis of C-3-(hetero)aryl [1,2,3]triazolo[1,5-a]pyridines using the Stille reaction

被引：4
|
作者：
Germain, Herve [1 ]
Harris, Craig S. [1 ]
Lebraud, Honorine [1 ]
机构：
[1] AstraZeneca, Ctr Rech, ZI Pompelle, F-51689 Reims 2, France
来源：
TETRAHEDRON LETTERS | 2011年 / 52卷 / 48期
关键词：
1,2,3]Triazolo[1,5-a]pyridine; Stille cross-coupling reaction; Microwave-assisted organic synthesis (MAOS); TRIAZOLOPYRIDINES; HYDRAZONES; OXIDATION; HALOPYRIMIDINES;
D O I：
10.1016/j.tetlet.2011.09.052
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Herein, we report a novel and high yielding approach for the preparation of the first C-3-organometallic substituted [1,2,3]triazolo[1,5-a]pyridine and its application to the Stille reaction using MAOS. (C) 2011 Elsevier Ltd. All rights reserved.
引用
收藏
页码：6376 / 6378
页数：3
相关论文
共 50 条
  • [21] Synthesis and in vitro leishmanicidal activity of novel [1,2,3]triazolo[1,5-a] pyridine salts
    Martin-Montes, Alvaro
    Ballesteros-Garrido, Rafael
    Martin-Escolano, Ruben
    Marin, Clotilde
    Guitierrez-Sanchez, Ramon
    Abarca, Beier
    Ballesteros, Rafael
    Sanchez-Moreno, Manuel
    [J]. RSC ADVANCES, 2017, 7 (26) : 15715 - 15726
  • [22] Chemical reactivity of [1,2,3]triazolo[1,5-a]- and [1,5-c]-pyrimidinium salts
    Bátori, S
    Gács-Baitz, E
    Bokotey, S
    Messmer, A
    [J]. TETRAHEDRON, 2003, 59 (24) : 4297 - 4301
  • [23] STUDIES ON HETEROCYCLIC-COMPOUNDS .33. SYNTHESIS OF [1,2,3]-TRIAZOLO[1,5-A]PYRIDINES WITH NICKEL PEROXIDE
    OGURA, H
    MINEO, S
    NAKAGAWA, K
    SHIBA, S
    [J]. YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, 1981, 101 (04): : 329 - 335
  • [24] Triazolopyridines.: Part 25:: Synthesis of new chiral ligands from [1,2,3]triazolo[ 1,5-a]pyridines
    Abarca, Belen
    Ballesteros, Rafael
    Ballesteros-Garrido, Rafael
    Colobert, Francoise
    Leroux, Frederic R.
    [J]. TETRAHEDRON, 2007, 63 (42) : 10479 - 10485
  • [25] Evaluation of the Novel Antichagasic Activity of [1,2,3]Triazolo[1,5-a]pyridine Derivatives
    Lapier, Michel
    Zuniga-Lopez, Maria C.
    Aguilera-Venegas, Benjamin
    Adam, Rosa
    Abarca, Belen
    Ballesteros, Rafael
    Lopez-Munoz, Rodrigo
    Diego Maya, Juan
    Olea-Azar, Claudio
    [J]. CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2017, 17 (04) : 399 - 411
  • [26] Triazoloazine Diazomethylazine Valence Isomerization. [1,2,3]Triazolo[1,5-a]pyridines and 2-Diazomethylpyridines
    Aylward, Nigel
    Winter, Hans-Wilhelm
    Eckhardt, Ulrich
    Wentrup, Curt
    [J]. JOURNAL OF ORGANIC CHEMISTRY, 2016, 81 (02): : 667 - 672
  • [27] A new synthesis for 1,2,4-triazolo[1,5-a]-pyridines and 1,2,4-triazolo[1,5-a]isoquinolines
    Hussein, AM
    Sherif, SM
    Atalla, AA
    [J]. MONATSHEFTE FUR CHEMIE, 1996, 127 (11): : 1153 - 1160
  • [28] Efficient multicomponent synthesis of highly substituted [1,2,3]triazolo[1,5-a]pyrimidines
    Eugene S. Gladkov
    Svetlana N. Sirko
    Svetlana V. Shishkina
    Oleg V. Shishkin
    Irina V. Knyazeva
    Sergey M. Desenko
    Valentin A. Chebanov
    [J]. Monatshefte für Chemie - Chemical Monthly, 2010, 141 : 773 - 779
  • [29] Efficient multicomponent synthesis of highly substituted [1,2,3]triazolo[1,5-a]pyrimidines
    Gladkov, Eugene S.
    Sirko, Svetlana N.
    Shishkina, Svetlana V.
    Shishkin, Oleg V.
    Knyazeva, Irina V.
    Desenko, Sergey M.
    Chebanov, Valentin A.
    [J]. MONATSHEFTE FUR CHEMIE, 2010, 141 (07): : 773 - 779
  • [30] Synthesis of [1,2,3]Triazolo[1,5-a]quinoline-3-carboxamides Promoted by Organocatalyst and Base
    Da Costa, Gabriel P. P.
    Blodorn, Gustavo B. B.
    Barcellos, Thiago
    Silva, Marcio S.
    Luque, Rafael
    Alves, Diego
    [J]. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2023, 26 (30)
12345