One-pot synthesis of polysubstituted pyrimidines

被引：30
|
作者：
Kiselyov, AS [1 ]
机构：
[1] Chem Divers, Small Mol Drug Discovery, San Diego, CA 92121 USA
来源：
TETRAHEDRON LETTERS | 2005年 / 46卷 / 10期
关键词：
pyrimidines; amidines; condensations;
D O I：
10.1016/j.tetlet.2005.01.068
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A series of polysubstituted pyrimidines were synthesized from in situ generated alpha,beta-unsaturated imines and the corresponding amidine or guanidine derivatives in a convenient one-pot procedure. (C) 2005 Elsevier Ltd. All rights reserved.
引用
收藏
页码：1663 / 1665
页数：3
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