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- [21] Preclinical characterization of tunlametinib, a novel, potent, and selective MEK inhibitorFRONTIERS IN PHARMACOLOGY, 2023, 14Liu, Yahong论文数: 0 引用数: 0 h-index: 0机构: Shanghai Kechow Pharm Inc, Shanghai, Peoples R China Shanghai Kechow Pharm Inc, Shanghai, Peoples R ChinaCheng, Ying论文数: 0 引用数: 0 h-index: 0机构: Shanghai Kechow Pharm Inc, Shanghai, Peoples R China Shanghai Kechow Pharm Inc, Shanghai, Peoples R ChinaHuang, Gongchao论文数: 0 引用数: 0 h-index: 0机构: Shanghai Kechow Pharm Inc, Shanghai, Peoples R China Shanghai Kechow Pharm Inc, Shanghai, Peoples R ChinaXia, Xiangying论文数: 0 引用数: 0 h-index: 0机构: Shanghai Kechow Pharm Inc, Shanghai, Peoples R China Shanghai Kechow Pharm Inc, Shanghai, Peoples R ChinaWang, Xingkai论文数: 0 引用数: 0 h-index: 0机构: Shanghai Kechow Pharm Inc, Shanghai, Peoples R China Shanghai Kechow Pharm Inc, Shanghai, Peoples R ChinaTian, Hongqi论文数: 0 引用数: 0 h-index: 0机构: Shanghai Kechow Pharm Inc, Shanghai, Peoples R China Shanghai Kechow Pharm Inc, Shanghai, Peoples R China
- [22] The Chk1 inhibitor AZD7762 sensitises p53 mutant breast cancer cells to radiation in vitro and in vivoMOLECULAR MEDICINE REPORTS, 2012, 6 (04) : 897 - 903Ma, Zhikun论文数: 0 引用数: 0 h-index: 0机构: Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R China Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R ChinaYa, Guoliang论文数: 0 引用数: 0 h-index: 0机构: Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Gen Surg, Luoyang 471003, Henan, Peoples R China Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R ChinaZhou, Bo论文数: 0 引用数: 0 h-index: 0机构: Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R China Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R ChinaFan, Yonggang论文数: 0 引用数: 0 h-index: 0机构: Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Gen Surg, Luoyang 471003, Henan, Peoples R China Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R ChinaGao, Shegan论文数: 0 引用数: 0 h-index: 0机构: Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R China Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R ChinaFeng, Xiaoshan论文数: 0 引用数: 0 h-index: 0机构: Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R China Henan Univ Sci & Technol, Affiliated Hosp 1, Dept Oncol, Luoyang 471003, Henan, Peoples R China
- [23] Chk1/2 inhibitor AZD7762 enhances the susceptibility of IDH-mutant brain cancer cells to temozolomideMedical Oncology, 39Erkin Ozgiray论文数: 0 引用数: 0 h-index: 0机构: Ege University,Department of Neurosurgery, Medicine FacultyFatma Sogutlu论文数: 0 引用数: 0 h-index: 0机构: Ege University,Department of Neurosurgery, Medicine FacultyCigir Biray Avci论文数: 0 引用数: 0 h-index: 0机构: Ege University,Department of Neurosurgery, Medicine Faculty
- [24] Gemcitabine and Chk1 Inhibitor AZD7762 Synergistically Suppress the Growth of Lkb1-Deficient Lung AdenocarcinomaCANCER RESEARCH, 2017, 77 (18) : 5068 - 5076Liu, Yan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USALi, Yuyang论文数: 0 引用数: 0 h-index: 0机构: Shandong Univ, Shandong Prov Hosp, Jinan, Shandong, Peoples R China Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAWang, Xiaoen论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USALiu, Feiyang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Hefei, Anhui, Peoples R China Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAGao, Peng论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAQuinn, Max M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USALi, Fei论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAMerlino, Ashley A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USABenes, Cyril论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Ctr Canc Res, Boston, MA 02114 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USALiu, Qingsong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Hefei, Anhui, Peoples R China Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USAWong, Kwok-Kin论文数: 0 引用数: 0 h-index: 0机构: NYU, Langone Med Ctr New York, Laura & Isaac Perlmutter Canc Ctr, New York, NY 10016 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02115 USA
- [25] Chk1/2 inhibitor AZD7762 enhances the susceptibility of IDH-mutant brain cancer cells to temozolomideMEDICAL ONCOLOGY, 2022, 39 (11)论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Avci, Cigir Biray论文数: 0 引用数: 0 h-index: 0机构: Ege Univ, Med Fac, Dept Med Biol, Izmir, Turkey Ege Univ, Med Fac, Dept Neurosurg, Izmir, Turkey
- [26] Preclinical pharmacokinetics of CASC-578, a novel, selective, potent, and orally bioavailable small molecule checkpoint kinase 1 inhibitorCANCER RESEARCH, 2017, 77Leviten, Dina论文数: 0 引用数: 0 h-index: 0Sierra, Teresa论文数: 0 引用数: 0 h-index: 0Dozier, Ashley论文数: 0 引用数: 0 h-index: 0Boyce, Richard论文数: 0 引用数: 0 h-index: 0Boyle, Bob论文数: 0 引用数: 0 h-index: 0Peterson, Scott论文数: 0 引用数: 0 h-index: 0Vo, Alex C.论文数: 0 引用数: 0 h-index: 0
- [27] Discovery of the Potent and Selective Inhaled Janus Kinase 1 Inhibitor AZD4604 and Its Preclinical CharacterizationJOURNAL OF MEDICINAL CHEMISTRY, 2023, : 13400 - 13415Nilsson, Magnus论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenBerggren, Kristina论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenBerglund, Susanne论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenCerboni, Silvia论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenCollins, Mia论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenDahl, Goran论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Struct & Biophys Res & Early Dev, Discovery Sci, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenElmqvist, David论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Pharmaceut Sci, Early Prod Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenGrimster, Neil P.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Oncol R&D, Waltham, MA 02451 USA AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenHendrickx, Ramon论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Res & Early Dev, Resp & Immunol,DMPK, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenJohansson, Johan R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenKettle, Jason G.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Oncol R&D, Waltham, MA 02451 USA AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenLepisto, Matti论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenRhedin, Magdalena论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenSmailagic, Amir论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenSu, Qibin论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Oncol R&D, Waltham, MA 02451 USA AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenWennberg, Tiiu论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenWu, Allan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Discovery Sci, R&D, Waltham, MA 02451 USA AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenOsterlund, Torben论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Res & Early Dev, Discovery Sci,Mechanist Biol & Profiling, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenNaessens, Thomas论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenMitra, Suman论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden
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