共 50 条
- [41] Conjugation of a brain-penetrant peptide with neurotensin provides antinociceptive propertiesJOURNAL OF CLINICAL INVESTIGATION, 2014, 124 (03): : 1199 - 1213Demeule, Michel论文数: 0 引用数: 0 h-index: 0机构: Angiochem Inc, Montreal, PQ, Canada Angiochem Inc, Montreal, PQ, Canada论文数: 引用数: h-index:机构:Regina, Anthony论文数: 0 引用数: 0 h-index: 0机构: Angiochem Inc, Montreal, PQ, Canada Angiochem Inc, Montreal, PQ, CanadaBesserer-Offroy, Elie论文数: 0 引用数: 0 h-index: 0机构: Univ Sherbrooke, Fac Med & Hlth Sci, Dept Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Univ Sherbrooke, Inst Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Angiochem Inc, Montreal, PQ, CanadaMurza, Alexandre论文数: 0 引用数: 0 h-index: 0机构: Univ Sherbrooke, Fac Med & Hlth Sci, Dept Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Univ Sherbrooke, Inst Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Angiochem Inc, Montreal, PQ, CanadaTetreault, Pascal论文数: 0 引用数: 0 h-index: 0机构: Univ Sherbrooke, Fac Med & Hlth Sci, Dept Physiol & Biophys, Sherbrooke, PQ J1H 5N4, Canada Angiochem Inc, Montreal, PQ, CanadaBelleville, Karine论文数: 0 引用数: 0 h-index: 0机构: Univ Sherbrooke, Fac Med & Hlth Sci, Dept Physiol & Biophys, Sherbrooke, PQ J1H 5N4, Canada Angiochem Inc, Montreal, PQ, CanadaChe, Christian论文数: 0 引用数: 0 h-index: 0机构: Angiochem Inc, Montreal, PQ, Canada Angiochem Inc, Montreal, PQ, CanadaLarocque, Alain论文数: 0 引用数: 0 h-index: 0机构: Angiochem Inc, Montreal, PQ, Canada Angiochem Inc, Montreal, PQ, CanadaThiot, Carine论文数: 0 引用数: 0 h-index: 0机构: Angiochem Inc, Montreal, PQ, Canada Angiochem Inc, Montreal, PQ, CanadaBeliveau, Richard论文数: 0 引用数: 0 h-index: 0机构: Univ Quebec, Mol Med Lab, Montreal, PQ H3C 3P8, Canada Angiochem Inc, Montreal, PQ, CanadaLongpre, Jean-Michel论文数: 0 引用数: 0 h-index: 0机构: Univ Sherbrooke, Fac Med & Hlth Sci, Dept Physiol & Biophys, Sherbrooke, PQ J1H 5N4, Canada Univ Sherbrooke, Fac Med & Hlth Sci, Dept Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Univ Sherbrooke, Inst Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Angiochem Inc, Montreal, PQ, CanadaMarsault, Eric论文数: 0 引用数: 0 h-index: 0机构: Univ Sherbrooke, Fac Med & Hlth Sci, Dept Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Univ Sherbrooke, Inst Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Angiochem Inc, Montreal, PQ, CanadaLeduc, Richard论文数: 0 引用数: 0 h-index: 0机构: Univ Sherbrooke, Fac Med & Hlth Sci, Dept Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Univ Sherbrooke, Inst Pharmacol, Sherbrooke, PQ J1H 5N4, Canada Angiochem Inc, Montreal, PQ, CanadaLachowicz, Jean E.论文数: 0 引用数: 0 h-index: 0机构: Angiochem Inc, Montreal, PQ, Canada Angiochem Inc, Montreal, PQ, CanadaGonias, Steven L.论文数: 0 引用数: 0 h-index: 0机构: UCSD, Sch Med, Dept Pathol, La Jolla, CA USA Angiochem Inc, Montreal, PQ, CanadaCastaigne, Jean-Paul论文数: 0 引用数: 0 h-index: 0机构: Angiochem Inc, Montreal, PQ, Canada Angiochem Inc, Montreal, PQ, CanadaSarret, Philippe论文数: 0 引用数: 0 h-index: 0机构: Univ Sherbrooke, Fac Med & Hlth Sci, Dept Physiol & Biophys, Sherbrooke, PQ J1H 5N4, Canada Angiochem Inc, Montreal, PQ, Canada
- [42] N-Aromatic-Substituted Indazole Derivatives as Brain-Penetrant and Orally Bioavailable JNK3 InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2021, 12 (10): : 1546 - 1552Feng, Yangbo论文数: 0 引用数: 0 h-index: 0机构: React Biol Corp, Malvern, PA 19355 USA Univ Miami, Miller Sch Med, Dept Mol & Cellular Pharmacol, Sylvester Comprehens Canc Ctr, Miami, FL 33136 USA Scripps Res, Crystallog Core Facil, Jupiter, FL 33458 USAPark, HaJeung论文数: 0 引用数: 0 h-index: 0机构: Scripps Res, Crystallog Core Facil, Jupiter, FL 33458 USA Scripps Res, Crystallog Core Facil, Jupiter, FL 33458 USARyu, Jae Cheon论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Biol Chem & Pharmacol, Coll Med, Columbus, OH 43210 USA Scripps Res, Crystallog Core Facil, Jupiter, FL 33458 USAYoon, Sung Ok论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Biol Chem & Pharmacol, Coll Med, Columbus, OH 43210 USA Scripps Res, Crystallog Core Facil, Jupiter, FL 33458 USA
- [43] Discovery of a Hydroxylamine-Based Brain-Penetrant EGFR Inhibitor for Metastatic Non-Small-Cell Lung CancerJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (22) : 15477 - 15492Hill, Jarvis论文数: 0 引用数: 0 h-index: 0机构: Univ Georgia, Dept Pharmaceut & Biomed Sci, Athens, GA 30602 USA Univ Georgia, Dept Chem, Athens, GA 30602 USA Univ Georgia, Dept Pharmaceut & Biomed Sci, Athens, GA 30602 USAJones, Robert M.论文数: 0 引用数: 0 h-index: 0机构: Univ Georgia, Complex Carbohydrate Res Ctr, Athens, GA 30602 USA Univ Georgia, Dept Pharmaceut & Biomed Sci, Athens, GA 30602 USA论文数: 引用数: h-index:机构:
- [44] Discovery of orally active, brain-penetrant C6-substituted aminothiazine BACE1 inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248Wu, Yong-Jin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAGuernon, Jason论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USARamkumar, Rajamani论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAMarcin, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAHiggins, Mendi论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAYang, Fukang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USASnyder, Lawrence论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAShi, Jianliang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAMcClure, Andrea论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAChang, ChiehYing论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAZhuo, Xiaoliang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAToyn, Jeremy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAAhlijanian, Michael K.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAMacor, John E.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USAThompson, Lorin A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USALewis, Hal论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Wallingford, CT 06492 USA
- [45] Volumetric Response of Brain Metastases in EGFR-Positive NSCLC Treated with CNS-Penetrant Tyrosine Kinase Inhibitors with or without Radiation TherapyINTERNATIONAL JOURNAL OF RADIATION ONCOLOGY BIOLOGY PHYSICS, 2022, 114 (03): : E60 - E60Ni, L.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USAPhuong, C.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USAChen, J. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USAChen, W. S.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USADaras, M.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Neurol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USARaleigh, D.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USANakamura, J. L.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USABoreta, L.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USASneed, P. K.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USABraunstein, S. E.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA Univ Calif San Francisco, Dept Radiat Oncol, San Francisco, CA USA
- [46] Design of a brain-penetrant CDK4/6 inhibitor for glioblastomaBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (16) : 2294 - 2301Bronner, Sarah M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAMerrick, Karl A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAMurray, Jeremy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USASalphati, Laurent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAMoffat, John G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAPang, Jodie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USASneeringer, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USADompe, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USACyr, Patrick论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAPurkey, Hans论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USABoenig, Gladys de Leon论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USALi, Jun论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAKolesnikov, Aleksandr论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USALarouche-Gauthier, Robin论文数: 0 引用数: 0 h-index: 0机构: Paraza Pharma Inc, 2525 Ave Marie Curie, Montreal, PQ H45 2E1, Canada Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USALai, Kwong Wah论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAShen, Xiaoli论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAAubert-Nicol, Samuel论文数: 0 引用数: 0 h-index: 0机构: Paraza Pharma Inc, 2525 Ave Marie Curie, Montreal, PQ H45 2E1, Canada Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAChen, Yi-Chen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USACheong, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USACrawford, James J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAHafner, Marc论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAHaghshenas, Pouyan论文数: 0 引用数: 0 h-index: 0机构: Paraza Pharma Inc, 2525 Ave Marie Curie, Montreal, PQ H45 2E1, Canada Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAJakalian, Araz论文数: 0 引用数: 0 h-index: 0机构: Paraza Pharma Inc, 2525 Ave Marie Curie, Montreal, PQ H45 2E1, Canada Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USALeclerc, Jean-Philippe论文数: 0 引用数: 0 h-index: 0机构: Paraza Pharma Inc, 2525 Ave Marie Curie, Montreal, PQ H45 2E1, Canada Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USALim, Ngiap-Kie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAO'Brien, Tom论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAPlise, Emile G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAShalan, Hadil论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USASturino, Claudio论文数: 0 引用数: 0 h-index: 0机构: Paraza Pharma Inc, 2525 Ave Marie Curie, Montreal, PQ H45 2E1, Canada Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAWai, John论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, 288 Fute Zhong Rd, Shanghai 200131, Peoples R China Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAXiao, Yang论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAYin, Jianping论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAZhao, Liang论文数: 0 引用数: 0 h-index: 0机构: Paraza Pharma Inc, 2525 Ave Marie Curie, Montreal, PQ H45 2E1, Canada Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAGould, Stephen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAOlivero, Alan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USAHeffron, Timothy P.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA Genentech Inc, 1 DNA Way, San Francisco, CA 94080 USA
- [47] Discovery of Preclinical Candidate AD1058 as a Highly Potent, Selective, and Brain-Penetrant ATR Inhibitor for the Treatment of Advanced MalignanciesJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (15) : 12735 - 12759Liu, Zhi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaJiang, Kailong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaLiu, Yan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Sch Pharm, Beijing 100049, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaLi, Junfei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Southern Med Univ, Sch Pharmaceut Sci, Guangzhou 510515, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaHuang, Siqi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaLi, Ping论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaXu, Lei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaXu, Xiaomin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaHu, Xiaobei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Chem Biol, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaZeng, Xia论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaHuang, Zehui论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaZhou, Yubo论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Chem Biol, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaLi, Jia论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Southern Med Univ, Sch Pharmaceut Sci, Guangzhou 510515, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Chem Biol, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaLong, Kai论文数: 0 引用数: 0 h-index: 0机构: Shanghai Annova Biotechnol Co Ltd, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R ChinaWang, Mingliang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Sch Pharm, Beijing 100049, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Peoples R China
- [48] NST-628 is a potent, fully brain-penetrant, RAS/MAPK pathway molecular glue inhibitor with efficacy in CNS tumor modelsMOLECULAR CANCER THERAPEUTICS, 2023, 22 (12)Ryan, Meagan B.论文数: 0 引用数: 0 h-index: 0Li, Chun论文数: 0 引用数: 0 h-index: 0Han, Yongxin论文数: 0 引用数: 0 h-index: 0Hoeflich, Klaus P.论文数: 0 引用数: 0 h-index: 0Hale, Michael R.论文数: 0 引用数: 0 h-index: 0Hagel, Margit论文数: 0 引用数: 0 h-index: 0
- [49] Development of a Novel Xenograft Pharmacokinetic/Pharmacodynamic Model for Assessing CNS Penetrant BTK inhibitorsMULTIPLE SCLEROSIS JOURNAL, 2022, 28 (1_SUPPL) : 108 - 109Basile, R.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USAHarp, C. Parker论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USARoach, A.论文数: 0 引用数: 0 h-index: 0机构: Gilead Sci, Foster City, CA USA Biogen, Cambridge, MA USABurns, J.论文数: 0 引用数: 0 h-index: 0机构: Abata Therapeut, Cambridge, MA USA Biogen, Cambridge, MA USATang, H.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USARyan, S.论文数: 0 引用数: 0 h-index: 0机构: Q32 Bio Inc, Cambridge, MA USA Biogen, Cambridge, MA USASchroeder, P.论文数: 0 引用数: 0 h-index: 0机构: FORMA Therapeut, Watertown, MA USA Biogen, Cambridge, MA USAKadakia, E.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USAGu, C.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USAPietrasiewicz, A.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USAD'Lima, N.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USAHamann, S.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USAJandreski, L.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USAReynolds, T. L.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USACameron, T.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USAMingueneau, M.论文数: 0 引用数: 0 h-index: 0机构: Biogen, Cambridge, MA USA Biogen, Cambridge, MA USA
- [50] Brain-Penetrant Macrocycles: Design Considerations, Future Prospects, and Call for PapersJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (10) : 7665 - 7667Malinky, Cori A.论文数: 0 引用数: 0 h-index: 0Bender, Aaron M.论文数: 0 引用数: 0 h-index: 0