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- [31] Structure-Guided Discovery of Aminoquinazolines as Brain-Penetrant and Selective LRRK2 InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (01) : 838 - 856Keylor, Mitchell H.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAGulati, Anmol论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAKattar, Solomon D.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAJohnson, Rebecca E.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAChau, Ryan W.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAMargrey, Kaila A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAArdolino, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAZarate, Cayetana论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAPoremba, Kelsey E.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USASimov, Vladimir论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAMorriello, Gregori J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Kenilworth, NJ 07033 USA Merck & Co Inc, Boston, MA 02115 USAActon, John J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Kenilworth, NJ 07033 USA Merck & Co Inc, Boston, MA 02115 USAPio, Barbara论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Kenilworth, NJ 07033 USA Merck & Co Inc, Boston, MA 02115 USAYan, Xin论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAPalte, Rachel L.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAMcMinn, Spencer E.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USANogle, Lisa论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USALesburg, Charles A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAAdpressa, Donovon论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USALin, Shishi论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Kenilworth, NJ 07033 USA Merck & Co Inc, Boston, MA 02115 USANeelamkavil, Santhosh论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Kenilworth, NJ 07033 USA Janssen Pharmaceut Co Johnson & Johnson, 3470 Broadway, New York, NY 10031 USA Merck & Co Inc, Boston, MA 02115 USALiu, Ping论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USASu, Jing论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Kenilworth, NJ 07033 USA Merck & Co Inc, Boston, MA 02115 USAHegde, Laxminarayan G.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAWoodhouse, Janice D.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAFaltus, Robert论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAXiong, Tina论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USACiaccio, Paul J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAPiesvaux, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAOtte, Karin M.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAWood, Harold B.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Kenilworth, NJ 07033 USA Merck & Co Inc, Boston, MA 02115 USAKennedy, Matthew E.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USABennett, David Jonathan论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USADiMauro, Erin F.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAFell, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USAFuller, Peter H.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Boston, MA 02115 USA Merck & Co Inc, Boston, MA 02115 USA
- [32] Development of Novel Brain-Penetrant Radioligands for PET Imaging of GABA Transporter-1JOURNAL OF NUCLEAR MEDICINE, 2021, 62Wang, Chao论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USAGravel, Paul论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USAZheng, Ming-Qiang论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USAKapinos, Michael论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USAEmery, Paul论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USAHolden, Daniel论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USARopchan, Jim论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USABorroni, Edilio论文数: 0 引用数: 0 h-index: 0机构: Hoffmann La Roche AG, Basel, Switzerland Yale Univ, Radiol & Biomed Imaging, New Haven, CT USAHoner, Michael论文数: 0 引用数: 0 h-index: 0机构: Hoffmann La Roche AG, Basel, Switzerland Yale Univ, Radiol & Biomed Imaging, New Haven, CT USAGobbi, Luca论文数: 0 引用数: 0 h-index: 0机构: Hoffmann La Roche AG, Basel, Switzerland Yale Univ, Radiol & Biomed Imaging, New Haven, CT USATamagnan, Gilles论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Psychiat, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USACarson, Richard论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USAHuang, Henry论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA Yale Univ, Radiol & Biomed Imaging, New Haven, CT USA
- [33] ERAS-801 IS A SELECTIVE BRAIN-PENETRANT EGFR INHIBITOR WITH IMPROVED ACTIVITY AGAINST EGFR EXTRACELLULAR DOMAIN-MUTANT GLIOBLASTOMANEURO-ONCOLOGY, 2024, 26Okobi, Quincy论文数: 0 引用数: 0 h-index: 0机构: UCLA, Los Angeles, CA USA UCLA, Los Angeles, CA USACadet, Dimitri论文数: 0 引用数: 0 h-index: 0机构: UCLA, Los Angeles, CA USA UCLA, Los Angeles, CA USAUrner, Lorenz论文数: 0 引用数: 0 h-index: 0机构: UCLA, Los Angeles, CA USA UCLA, Los Angeles, CA USAJung, Michael论文数: 0 引用数: 0 h-index: 0机构: UCLA, Los Angeles, CA USA UCLA, Los Angeles, CA USACloughesy, Timothy论文数: 0 引用数: 0 h-index: 0机构: UCLA, Los Angeles, CA USA UCLA, Los Angeles, CA USANathanson, David论文数: 0 引用数: 0 h-index: 0机构: UCLA, Los Angeles, CA USA UCLA, Los Angeles, CA USA
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- [35] Discovery of Indoline-2-carboxamide Derivatives as a New Class of Brain-Penetrant Inhibitors of Trypanosoma bruceiJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (19) : 7695 - 7706Cleghorn, Laura A. T.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandAlbrecht, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandStojanovski, Laste论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandSimeons, Frederick R. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandNorval, Suzanne论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandKime, Robert论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandCollie, Iain T.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandDe Rycker, Manu论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandCampbell, Lorna论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland论文数: 引用数: h-index:机构:Frearson, Julie A.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandWyatt, Paul G.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandRead, Kevin D.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, ScotlandGilbert, Ian H.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland Univ Dundee, Coll Life Sci, Div Biol Chem & Drug Discovery, Drug Discovery Unit,Sir James Black Ctr, Dundee DD1 5EH, Scotland
- [36] DEVELOPMENT OF HIGHLY POTENT, SELECTIVE BET BROMODOMAIN INHIBITORS THAT ARE CNS PENETRANT AND EFFECTIVE IN RODENT MODELS OF BRAIN CANCERNEURO-ONCOLOGY, 2014, 16Johnstone, Shawn论文数: 0 引用数: 0 h-index: 0机构: IntelliSyn, Montreal, PQ, Canada IntelliSyn, Montreal, PQ, CanadaJohhnsone, Andrea论文数: 0 引用数: 0 h-index: 0机构: 2Miami Miller Sch Med, Miami, FL USA IntelliSyn, Montreal, PQ, CanadaPenas, Clara论文数: 0 引用数: 0 h-index: 0机构: 2Miami Miller Sch Med, Miami, FL USA IntelliSyn, Montreal, PQ, CanadaStathias, Vasileios论文数: 0 引用数: 0 h-index: 0机构: 2Miami Miller Sch Med, Miami, FL USA IntelliSyn, Montreal, PQ, CanadaBrothers, Shaun论文数: 0 引用数: 0 h-index: 0机构: 2Miami Miller Sch Med, Miami, FL USA IntelliSyn, Montreal, PQ, CanadaAyad, Nagi论文数: 0 引用数: 0 h-index: 0机构: 2Miami Miller Sch Med, Miami, FL USA IntelliSyn, Montreal, PQ, CanadaWahlestedt, Claes论文数: 0 引用数: 0 h-index: 0机构: 2Miami Miller Sch Med, Miami, FL USA IntelliSyn, Montreal, PQ, CanadaAlbert, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: IntelliSyn, Montreal, PQ, Canada IntelliSyn, Montreal, PQ, Canada
- [37] Development of highly potent, selective BET bromodomain inhibitors that are CNS penetrant and effective in rodent models of brain cancerABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250Albert, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: IntelliSyn Pharma, Chem, Montreal, PQ, Canada IntelliSyn Pharma, Chem, Montreal, PQ, CanadaJohnstone, Shawn论文数: 0 引用数: 0 h-index: 0机构: IntelliSyn Pharma, Chem, Montreal, PQ, Canada IntelliSyn Pharma, Chem, Montreal, PQ, CanadaBayrakdarian, Malken论文数: 0 引用数: 0 h-index: 0机构: IntelliSyn Pharma, Chem, Montreal, PQ, Canada IntelliSyn Pharma, Chem, Montreal, PQ, CanadaJohnstone, Andrea论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miller Sch Med, Psychiat & Behav Sci, Miami, FL 33136 USA IntelliSyn Pharma, Chem, Montreal, PQ, CanadaPenas, Clara论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miller Sch Med, Psychiat & Behav Sci, Miami, FL 33136 USA IntelliSyn Pharma, Chem, Montreal, PQ, CanadaStathias, Vasileios论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miller Sch Med, Psychiat & Behav Sci, Miami, FL 33136 USA IntelliSyn Pharma, Chem, Montreal, PQ, CanadaBrothers, Shaun论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miller Sch Med, Psychiat & Behav Sci, Miami, FL 33136 USA IntelliSyn Pharma, Chem, Montreal, PQ, CanadaAyad, Nagi论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miller Sch Med, Psychiat & Behav Sci, Miami, FL 33136 USA IntelliSyn Pharma, Chem, Montreal, PQ, CanadaWahlestedt, Claes论文数: 0 引用数: 0 h-index: 0机构: Univ Miami, Miller Sch Med, Psychiat & Behav Sci, Miami, FL 33136 USA IntelliSyn Pharma, Chem, Montreal, PQ, Canada
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