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- [1] DEVELOPMENT OF BRAIN-PENETRANT EGFR INHIBITORS FOR GLIOBLASTOMANEURO-ONCOLOGY, 2018, 20 : 70 - 70Tsang, Jonathan论文数: 0 引用数: 0 h-index: 0机构: UCLA Mol & Med Pharmacol, Los Angeles, CA USA UCLA Mol & Med Pharmacol, Los Angeles, CA USAUrner, Lorenz论文数: 0 引用数: 0 h-index: 0机构: UCLA Chem & Biochem, Los Angeles, CA USA UCLA Mol & Med Pharmacol, Los Angeles, CA USAKim, Gyudong论文数: 0 引用数: 0 h-index: 0机构: UCLA Chem & Biochem, Los Angeles, CA USA UCLA Mol & Med Pharmacol, Los Angeles, CA USAChow, Kingsley论文数: 0 引用数: 0 h-index: 0机构: UCLA Chem & Biochem, Los Angeles, CA USA UCLA Mol & Med Pharmacol, Los Angeles, CA USAClark, Peter论文数: 0 引用数: 0 h-index: 0机构: UCLA Mol & Med Pharmacol, Los Angeles, CA USA UCLA Mol & Med Pharmacol, Los Angeles, CA USACloughesy, Timothy论文数: 0 引用数: 0 h-index: 0机构: UCLA Neurooncol, Los Angeles, CA USA UCLA Mol & Med Pharmacol, Los Angeles, CA USAJung, Michael论文数: 0 引用数: 0 h-index: 0机构: UCLA Chem & Biochem, Los Angeles, CA USA UCLA Mol & Med Pharmacol, Los Angeles, CA USANathanson, David论文数: 0 引用数: 0 h-index: 0机构: UCLA Mol & Med Pharmacol, Los Angeles, CA USA UCLA Mol & Med Pharmacol, Los Angeles, CA USA
- [2] Identification of Brain-Penetrant ATP-Competitive mTOR Inhibitors for CNS SyndromesJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (13) : 9095 - 9119Bonazzi, Simone论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAGray, Audrey论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAThomsen, Noel M.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USABiag, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USALabbe-Giguere, Nancy论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAKeaney, Erin P.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Kymera Therapeut, 200 Arsenal Yards Blvd, Watertown, MA 02472 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAMalik, Hasnain A.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USASun, Yingchuan论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA ImmunoGen, 830 Winter St, Waltham, MA 02451 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USANunez, Jill论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAKarki, Rajeshri G.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAKnapp, Mark论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAElling, Robert论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAFuller, John论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Chem Biol & Therapeut, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAPardee, Gwynn论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Chem Biol & Therapeut, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USACraig, Lucas论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USACapre, Ketthsy论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USASalas, Sarah论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAGorde, Aakruti论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Sana Biotechnol, 300 Technol Sq, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USALiang, Guiqing论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut, 50 Northern Ave, Boston, MA 02210 USA Novartis Inst Biomed Res, Pharmacokinet Sci, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USALubicka, Danuta论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Drug Dev Tech Res & Dev, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAMcTighe, Stephanie M.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Arkuda Therapeut, 200 Arsenal Yards Blvd, Watertown, MA 02472 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAGoold, Carleton论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Maze Therapeut, 171 Oyster Point Blvd South, San Francisco, CA 94080 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USALiu, Shanming论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Chem Biol & Therapeut, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USADeng, Lin论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Pharmacokinet Sci, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAHong, Jin论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Preclin Safety, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAFekete, Alexander论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Preclin Safety, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAStadelmann, Pascal论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Preclin Safety, CH-4056 Basel, Switzerland Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAFrieauff, Wilfried论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Preclin Safety, CH-4056 Basel, Switzerland Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAElhajouji, Azeddine论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Preclin Safety, CH-4056 Basel, Switzerland Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USABauer, Daniel论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Preclin Safety, CH-4056 Basel, Switzerland Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USALerchner, Andreas论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, CH-4056 Basel, Switzerland Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USARadetich, Branko论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Sonata Therapeut, 500 Arsenal St, Watertown, MA 02472 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAFuret, Pascal论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, CH-4056 Basel, Switzerland Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAPiizzi, Grazia论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USABurdette, Doug论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Pharmacokinet Sci, Cambridge, MA 02139 USA Moderna Therapeut, 200 Technol Sq, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAWilson, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Stylus Med, 1400 One Kendal Sq, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAPeukert, Stefan论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAHamann, Lawrence G.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Global Discovery Chem, Cambridge, MA 02139 USA Interdict Bio, 953 Indiana St, San Francisco, CA 94107 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USAMurphy, Leon O.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Chem Biol & Therapeut, Cambridge, MA 02139 USA Casma Therapeut Inc, 400 Technol Sq, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USACurtis, Daniel论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA Vesalius Therapeut, 100 Binney St, Cambridge, MA 02142 USA Novartis Inst Biomed Res, Neurosci, Cambridge, MA 02139 USA
- [3] Brain-penetrant kinase chemotherapeutics: Learning from CNS spaceABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2019, 257Mader, Mary论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Discovery Chem Res & Technol, Indianapolis, IN 46285 USA Eli Lilly & Co, Discovery Chem Res & Technol, Indianapolis, IN 46285 USAShi, Yuan论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Discovery Chem Res & Technol, Indianapolis, IN 46285 USA Eli Lilly & Co, Discovery Chem Res & Technol, Indianapolis, IN 46285 USA
- [4] Development of a Potent Brain-Penetrant EGFR Tyrosine Kinase Inhibitor against Malignant Brain TumorsACS MEDICINAL CHEMISTRY LETTERS, 2020, 11 (10): : 1799 - 1809Tsang, Jonathan E.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Med Pharmacol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USAUrner, Lorenz M.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Chem & Biochem, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USAKim, Gyudong论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Chem & Biochem, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USAChow, Kingsley论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Med Pharmacol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USABaufeld, Lynn论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Med Pharmacol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USAFaull, Kym论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Jane & Terry Semel Inst Neurosci & Human Behav, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Psychiat & Biobehav Sci, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USACloughesy, Timothy F.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Neurol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USAClark, Peter M.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Med Pharmacol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Crump Inst Mol Imaging, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USAJung, Michael E.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Chem & Biochem, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USANathanson, David A.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Med Pharmacol, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol, Los Angeles, CA 90095 USA
- [5] 18F-Labeled brain-penetrant EGFR tyrosine kinase inhibitors for PET imaging of glioblastomaCHEMICAL SCIENCE, 2023, 14 (47) : 13825 - 13831Narayanam, Maruthi Kumar论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Crump Inst Mol Imaging, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USATsang, Jonathan E.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USAXu, Shili论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Crump Inst Mol Imaging, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USANathanson, David A.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USAMurphy, Jennifer M.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Crump Inst Mol Imaging, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Calif Los Angeles, Dept Mol & Med Pharmacol, David Geffen Sch Med, Los Angeles, CA 90095 USA
- [6] Discovery of Brain-Penetrant COMT Inhibitors for the Treatment of Cognitive ImpairmentNEUROPSYCHOPHARMACOLOGY, 2016, 41 : S205 - S205Carr, Gregory论文数: 0 引用数: 0 h-index: 0机构: Lieber Inst Brain Dev, Baltimore, MD USA Lieber Inst Brain Dev, Baltimore, MD USALi, Cailian论文数: 0 引用数: 0 h-index: 0机构: Lieber Inst Brain Dev, Baltimore, MD USA Lieber Inst Brain Dev, Baltimore, MD USADePasquale, Michael论文数: 0 引用数: 0 h-index: 0机构: Lieber Inst Brain Dev, Baltimore, MD USA Lieber Inst Brain Dev, Baltimore, MD USATian, Qingjun论文数: 0 引用数: 0 h-index: 0机构: Lieber Inst Brain Dev, Baltimore, MD USA Lieber Inst Brain Dev, Baltimore, MD USAWeinberger, Daniel R.论文数: 0 引用数: 0 h-index: 0机构: Lieber Inst Brain Dev, Baltimore, MD USA Lieber Inst Brain Dev, Baltimore, MD USABarrow, James论文数: 0 引用数: 0 h-index: 0机构: Lieber Inst Brain Dev, Baltimore, MD USA Lieber Inst Brain Dev, Baltimore, MD USA
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- [8] Discovery of Brain-Penetrant Glucosylceramide Synthase Inhibitors with a Novel PharmacophoreJOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (05) : 4270 - 4290Tanaka, Yuta论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanSeto, Masaki论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanKakegawa, Keiko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanTakami, Kazuaki论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanKikuchi, Fumiaki论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanYamamoto, Takeshi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanNakamura, Minoru论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanDaini, Masaki论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanMurakami, Masataka论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanOhashi, Tomohiro论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanKasahara, Takahito论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanWang, Junsi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanIkeda, Zenichi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanWada, Yasufumi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanPuenner, Florian论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanFujii, Takahiro论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanInazuka, Masakazu论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanSato, Sho论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanSuzaki, Tomohiko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanOak, Jeong-Ho论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanTakai, Yuichi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanKohara, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanKimoto, Kouya论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanOki, Hideyuki论文数: 0 引用数: 0 h-index: 0机构: Axcelead Drug Discovery Partners, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanMikami, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanSasaki, Minoru论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, JapanTanaka, Yuta论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, Res, Fujisawa, Kanagawa 2518555, Japan
- [9] The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (01) : 658 - 665Graham, Thomas H.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAShen, Hong C.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALiu, Wensheng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAXiong, Yusheng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAVerras, Andreas论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USABleasby, Kelly论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USABhatt, Urmi R.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChabin, Renee M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Operat Res, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChen, Dunlu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChen, Qing论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGarcia-Calvo, Margarita论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAGeissler, Wayne M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHe, Huaibing论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALassman, Michael E.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAShen, Zhu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USATong, Xinchun论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USATung, Elaine C.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAXie, Dan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAXu, Suoyu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAColletti, Steven L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USATata, James R.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAHale, Jeffrey J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAPinto, Shirly论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAShen, Dong-Ming论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
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