Structure-based design of HIV protease inhibitors: Sulfonamide-containing 5,6-dihydro-4-hydroxy-2-pyrones as non-peptidic inhibitors

被引：89
|
作者：
Thaisrivongs, S
Skulnick, HI
Turner, SR
Strohbach, JW
Tommasi, RA
Johnson, PD
Aristoff, PA
Judge, TM
Gammill, RB
Morris, JK
Romines, KR
Chrusciel, RA
Hinshaw, RR
Chong, KT
Tarpley, WG
Poppe, SM
Slade, DE
Lynn, JC
Horng, MM
Tomich, PK
Seest, EP
Dolak, LA
Howe, WJ
Howard, GM
Schwende, FJ
Toth, LN
Padbury, GE
Wilson, GJ
Shiou, LH
Zipp, GL
Wilkinson, KF
Rush, BD
Ruwart, MJ
Koeplinger, KA
Zhao, ZY
Cole, S
Zaya, RM
Kakuk, TJ
Janakiraman, MN
Watenpaugh, KD
机构：
[1] SAMC, Pharmacia and Upjohn, Inc., Kalamazoo
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1996年 / 39卷 / 22期
关键词：
D O I：
10.1021/jm960541s
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
[No abstract available]
引用
收藏
页码：4349 / 4353
页数：5
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