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- [1] Structure-based design of novel HIV protease inhibitors: Sulfonamide-containing 4-hydroxycoumarins and 4-hydroxy-2-pyrones as potent non-peptidic inhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (12) : 2400 - 2410Thaisrivongs, SJanakiraman, MNChong, KTTomich, PKDolak, LATurner, SRStrohbach, JWLynn, JCHorng, MMHinshaw, RRWatenpaugh, KD
- [2] Structure-based design of HIV protease inhibitors: 5,6-dihydro-4-hydroxy-2-pyrones as effective, nonpeptidic inhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (23) : 4630 - 4642Thaisrivongs, SRomero, DLTommasi, RAJanakiraman, MNStrohbach, JWTurner, SRBiles, CMorge, RRJohnson, PDAristoff, PATomich, PKLynn, JCHorng, MMChong, KTHinshaw, RRHowe, WJFinzel, BCWatenpaugh, KD
- [3] Structure-based design of sulfonamide-substituted non-peptidic HIV protease inhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (26) : 4968 - 4971Skulnick, HIJohnson, PDHowe, WJTomich, PKChong, KTWatenpaugh, KDJanakiraman, MNDolak, LAMcGrath, JPLynn, JCHorng, MMHinshaw, RRZipp, GLRuwart, MJSchwende, FJZhong, WZPadbury, GEDalga, RJShiou, LHPossert, PLRush, BDWilkinson, KFHoward, GMToth, LNWilliams, MGKakuk, TJCole, SLZaya, RMLovasz, KDMorris, JKRomines, KRThaisrivongs, SAristoff, PA
- [4] Synthesis of 5,6-dihydro-4-hydroxy-2-pyrones as HIV-1 protease inhibitors: The profound effect of polarity on antiviral activityJOURNAL OF MEDICINAL CHEMISTRY, 1997, 40 (23) : 3707 - 3711Hagen, SEPrasad, JVNVBoyer, FEDomagala, JMEllsworth, ELGajda, CHamilton, HWMarkoski, LJSteinbaugh, BATait, BDLunney, EATummino, PJFerguson, DHupe, DNouhan, CGracheck, SJSaunders, JMVanderRoest, S
- [5] Non-peptidic hn protease inhibitors: Structure-based drug design of bis-sulfonamide dihydropyrones.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1996, 212 : 207 - MEDIJanakiraman, MNWatenpaugh, KDTomich, PKChong, KTThaisrivongs, SStrohbach, JW
- [6] STRUCTURE-BASED DESIGN OF HIV PROTEASE INHIBITORS - 4-HYDROXYCOUMARINS AND 4-HYDROXY-2-PYRONES AS NONPEPTIDIC INHIBITORSJOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (20) : 3200 - 3204THAISRIVONGS, STOMICH, PKWATENPAUGH, KDCHONG, KTHOWE, WJYANG, CPSTROHBACH, JWTURNER, SRMCGRATH, JPBOHANON, MJLYNN, JCMULICHAK, AMSPINELLI, PAHINSHAW, RRPAGANO, PJMOON, JBRUWART, MJWILKINSON, KFRUSH, BDZIPP, GLDALGA, RJSCHWENDE, FJHOWARD, GMPADBURY, GETOTH, LNZHAO, ZYKOEPLINGER, KAKAKUK, TJCOLE, SLZAYA, RMPIPER, RCJEFFREY, P
- [7] STRUCTURE-BASED DESIGN OF NONPEPTIDIC HIV PROTEASE INHIBITORS - CARBOXAMIDE-CONTAINING 4-HYDROXYCOUMARINS AND 4-HYDROXY-2-PYRONESABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1995, 209 : 239 - MEDITHAISRIVONGS, SSTROHBACH, JWTURNER, SRTOMICH, PKWATENPAUGH, KDCHONG, KTHOWE, WJRUWART, MJZIPP, GLSCHWENDE, FJPADBURY, GE
- [8] Non-peptidic HIV protease inhibitors:: C2-symmetry-based design of bis-sulfonamide dihydropyronesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1998, 8 (10) : 1237 - 1242Janakiraman, MNWatenpaugh, KDTomich, PKChong, KTTurner, SRTommasi, RAThaisrivongs, SStrohbach, JW
- [9] Iterative structure-based design of achiral, non-peptidic anthranilamide and benzamide-containing HIV protease inhibitors as antiviral agents.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1996, 211 : 14 - MEDIRandad, RSLubkowska, LBhat, TNSilva, AGulnik, SYu, BErickson, JW
- [10] STRUCTURE-BASED DESIGN OF NOVEL HIV PROTEASE INHIBITORS - CARBOXAMIDE-CONTAINING 4-HYDROXYCOUMARINS AND 4-HYDROXY-2-PYRONES AS POTENT NONPEPTIDIC INHIBITORSJOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (18) : 3624 - 3637THAISRIVONGS, SWATENPAUGH, KDHOWE, WJTOMICH, PKDOLAK, LACHONG, KTTOMICH, CSCTOMASSELLI, AGTURNER, SRSTROHBACH, JWMULICHAK, AMJANAKIRAMAN, MNMOON, JBLYNN, JCHORNG, MMHINSHAW, RRCURRY, KAROTHROCK, DJ