Synthesis of indole-2-carboxylic acid esters

被引：4
|
作者：
Allen, DA [1 ]
机构：
[1] Roche Biosci, Palo Alto, CA 94304 USA
来源：
SYNTHETIC COMMUNICATIONS | 1999年 / 29卷 / 03期
关键词：
D O I：
10.1080/00397919908085787
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The title compounds were prepared via lateral lithiation of N-Boc protected toluidines with sec-BuLi, quench with diethyl oxalate, followed by dehydration in TFA/CH2Cl2.
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页码：447 / 455
页数：9
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