Synthetic inhibitors of yeast cyclin-dependent kinase-activating kinases as antifungal agents

被引：0
|
作者：
不详
机构：
来源：
EXPERT OPINION ON THERAPEUTIC PATENTS | 2003年 / 13卷 / 06期
关键词：
antifungal; cyclin-dependent kinase (CDK); cyclin-dependent kinase-activating kinase (CAK); indolizines; kinase inhibitors;
D O I：
暂无
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
The Vertex application discloses an indeterminate number of indolizine and related heterocyclic derivatives that are claimed to be inhibitors of cyclin-dependent kinase (CDK)-activating kinases (CAKs), useful as antifungal agents. The GPC Biotech application discloses an, indeterminate number of compounds with a phenethylazaryl 'portion' linked to various substituents; all claimed to be inhibitors of various fungal enzymes, particularly prenyltransferases and CAK.
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页码：925 / 927
页数：3
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