Solution- and Solid-Phase Synthesis of Bis-Benzamide Libraries as α-Helix Mimetics and Their Evaluation on Inhibitory Activity to Prostate Cancer

被引:0
|
作者
Lee, Tae-Kyung [1 ]
Ravindranathan, Preethi [2 ]
Raj, Ganesh V. [2 ]
Ahn, Jung-Mo [1 ]
机构
[1] Univ Texas Dallas, Dept Chem, Richardson, TX 75080 USA
[2] Univ Texas SW Med Ctr Dallas, Dept Urol, Dallas, TX 75390 USA
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:460 / 460
页数:1
相关论文
共 50 条
  • [1] Solution- and solid-phase synthesis of isoxazole/isoxazoline containing phenolic libraries.
    Kurth, MJ
    Sammelson, RE
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 219 : U121 - U121
  • [2] Synthesis and Biological Evaluation of Bis-Benzamide-Based α-Helix Mimetics as Inhibitors of Androgen Receptor-Coactivator Interaction in Prostate Cancer
    Lee, Tae-Kyung
    Ravindranathan, Preethi
    Raj, Ganesh V.
    Ahn, Jung-Mo
    BIOPOLYMERS, 2011, 96 (04) : 460 - 460
  • [3] Solid-Phase Synthesis of Tris-Benzamides as α-Helix Mimetics
    Lee, Tae-Kyung
    Ahn, Jung-Mo
    ACS COMBINATORIAL SCIENCE, 2011, 13 (02) : 107 - 111
  • [4] Advances in Solution- and Solid-Phase Synthesis toward the Generation of Natural Product-like Libraries
    Nandy, Jyoti P.
    Prakesch, Michael
    Khadem, Shahriar
    Reddy, P. Thirupathi
    Sharma, Utpal
    Arya, Prabhat
    CHEMICAL REVIEWS, 2009, 109 (05) : 1999 - 2060
  • [5] Solution- and solid-phase synthesis of combinatorial libraries of trisubstituted 1,3,5-triazines
    Masquelin, T
    Meunier, N
    Gerber, F
    Rossé, G
    HETEROCYCLES, 1998, 48 (12) : 2489 - 2505
  • [6] Solution and solid-phase synthesis of trifluoromethyl peptides and mimetics
    Bravo, P
    Bruché, L
    Pesenti, C
    Viani, F
    Volonterio, A
    Zanda, M
    JOURNAL OF FLUORINE CHEMISTRY, 2001, 112 (01) : 153 - 162
  • [7] Solution- and solid-phase synthesis of radicicol (monorden) and pochonin C
    Barluenga, S
    Moulin, E
    Lopez, P
    Winssinger, N
    CHEMISTRY-A EUROPEAN JOURNAL, 2005, 11 (17) : 4935 - 4952
  • [8] Acyclic and cyclic thioenamino peptides: solution- and solid-phase synthesis
    Goren, Lee
    Pappo, Doron
    Goldberg, Israel
    Kashman, Yoel
    TETRAHEDRON LETTERS, 2009, 50 (09) : 1048 - 1050
  • [9] Modular Solid-Phase Synthesis of Teroxazoles as a Class of a-Helix Mimetics
    Gomes, Cristiano Pinto
    Metz, Alexander
    Bats, Jan W.
    Gohlke, Holger
    Goebel, Michael W.
    EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2012, 2012 (17) : 3270 - 3277
  • [10] Solution- and solid-phase synthesis of potential anticancer HDAC inhibitors
    Blum, Travis R.
    Shah, Heli K.
    Zang, Xiaoyu
    Korn, Ariella R.
    Wholly, Deirdre M.
    Miller, Justin S.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240