Quinolone analogues 8.: Synthesis of 3-aminopyridazino[3,4-b]quinoxalin-4(1H)-one

被引：7
|
作者：
Kurasawa, Y [1 ]
Kawase, A
Takizawa, J
Maesaki, Y
Kaji, E
Okamoto, Y
Kim, HS
机构：
[1] Kitasato Univ, Sch Pharmaceut Sci, Minato Ku, Tokyo 1088641, Japan
[2] Kitasato Univ, Ctr Nat Sci, Sagamihara, Kanagawa 2288555, Japan
[3] Catholic Univ Taegu, Dept Chem, Gyongsan 712702, South Korea
来源：
JOURNAL OF HETEROCYCLIC CHEMISTRY | 2005年 / 42卷 / 04期
关键词：
D O I：
10.1002/jhet.5570420412
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The 3-amino-1-methylpyridazino[3,4-b]quinoxalin-4(1H)-one 6 and N-(1,4-dihydro-1-methyl-4-oxopyridazino[3,4-b]quinoxalin-3-yl)carbamates 17a,b were synthesized from the 1,4-dihydro-1-methyl-4-oxopyridazino[3,4-b]quinoxaline-3-carboxylate 1b via the 1,5-dihydro-4-hydroxy-1-methylpyridazino[3,4-b]quinoxaline-3-carbohydrazide 13b and then 1,4-dihydro-1-methyl-4-oxopyridazino[3,4-b]quinoxaline-3-carboxazide 8. Heating of compound 13b and arylaldehydes afforded the 1,4-dihydro-1-methyl-4-oxopyridazino[3,4-b]quinoxaline-3-carbo(2-arylmethylene)hydrazides 14a-d.
引用
收藏
页码：551 / 556
页数：6
相关论文
共 50 条
  • [41] [3+2] Cyclization of Azidotrimethylsilane with Quinoxalin-2(1H)-Ones to Synthesize Tetrazolo[1,5-a]quinoxalin-4(5H)-Ones
    Yang, Qiming
    Zhang, Yuecheng
    Sun, Qian
    Shang, Kun
    Zhang, Hong-Yu
    Zhao, Jiquan
    ADVANCED SYNTHESIS & CATALYSIS, 2018, 360 (23) : 4509 - 4514
  • [42] Synthesis of bis-4H-furo[3,4-b]indoles
    McGowan, Meredeth A.
    Perreault, Denise M.
    Thornton, Nancy B.
    Garaas, Sarah D.
    Gribble, Gordon W.
    ARKIVOC, 2018, : 334 - 347
  • [43] 4H-1-BENZOTHIOPYRAN-4-ONE-3-CARBOXYLIC ACIDS AND 3,4-DIHYDRO-2H-ISOTHIAZOLO[5,4-B][1]BENZOTHIOPYRAN-3,4-DIONES AS QUINOLONE ANTIBACTERIAL ANALOGS
    CECCHETTI, V
    FRAVOLINI, A
    FRINGUELLI, R
    SCHIAFFELLA, F
    LORENZINI, MC
    TABARRINI, O
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 1993, 30 (04) : 1143 - 1148
  • [44] A NOVEL ONE-STEP SYNTHESIS OF 4H-FURO[3,4-B]PYRANS AND A TRANSFORMATION INTO A DIFURO[3,4-B-3',4'-E]PYRIDINE
    MARTIN, N
    SEGURA, JL
    SEOANE, C
    SOTO, JL
    MORALES, M
    SUAREZ, M
    LIEBIGS ANNALEN DER CHEMIE, 1991, (08): : 827 - 830
  • [45] Facile One-Pot Synthesis of [1,2,4]Triazolo[3,4-b][1,3,4]thiadiazines and 3,7-Dimethyl-4H-[1,2,4]triazino[3,4-b][1,3,4]thiadiazin-6-one Using Heteropolyacid Catalysts
    Motamedi, Radineh
    Monfared, Aazam
    Nezamabadi, Zohre Ghahghai
    Bamoharram, Fatemeh F.
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2011, 48 (03) : 604 - 607
  • [46] INTRAMOLECULARLY HYDROGEN-BONDED 3-PHENACYL-1H-PYRIDO[3,4-B]-PYRAZIN-2-ONE AND 2-PHENACYL-4H-PYRIDO[3,4-B]PYRAZIN-3-ONE
    SEKI, T
    IWANAMI, Y
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 1994, 31 (04) : 1065 - 1067
  • [47] Synthetic investigations of 3,4-dihydroquinoxalin-2(1H)-one and quinoxalin-2(1H)-one under varied experimental conditions
    Kurttila, Jaclyn
    Emery, Todd
    Kellen-Yuen, Cynthia
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250
  • [48] Facile Synthesis of Hydrazine Derivatives of 5H-Pyrrolo[3,4-b]pyrazine and 1H-Pyrrolo[3,4-b]quinoxaline
    Hordiyenko, Olga V.
    Rudenko, Igor V.
    Zamkova, Irina A.
    Denisenko, Oleksandr V.
    Biitseva, Angelina V.
    Arrault, Axelle
    Tolmachev, Andrei A.
    SYNTHESIS-STUTTGART, 2013, 45 (24): : 3375 - 3382
  • [49] SELENIUM HETEROCYCLES .33. SYNTHESIS OF THIENO[3,4-B]FURAN, SELENO[3,4-B]FURAN, THIENO[3,4-B]INDOLE AND SELENO[3,4-B]INDOLE - 4 NOVEL HETEROCYCLES
    SHAFIEE, A
    SATTARI, S
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 1982, 19 (02) : 227 - 231
  • [50] Novel one-pot synthesis of pyrazolo[3,4-b][1,4]oxazines
    Raslan, MA
    Abd El Latif, FM
    Otto, HH
    Sadek, KU
    JOURNAL OF THE CHINESE CHEMICAL SOCIETY, 2000, 47 (4B) : 947 - 949
12345