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- [42] Novel pyrazolo[1,5-a]pyrimidines as c-Src kinase inhibitors that reduce IKr channel blockadeBIOORGANIC & MEDICINAL CHEMISTRY, 2008, 16 (02) : 909 - 921Mukalyama, Harunobu论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, JapanNishimura, Toshihiro论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, JapanKobayashi, Satoko论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, JapanKomatsu, Yoshimitsu论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, JapanKikuchi, Shinji论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, JapanOzawa, Tomonaga论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, JapanKamada, Noboru论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, JapanOhnota, Hideki论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, Nagano 3998304, Japan
- [43] Discovery of novel pyrazole and pyrazolo[1,5-a]pyrimidine derivatives as cyclooxygenase inhibitors (COX-1 and COX-2) using molecular modeling simulationARCHIV DER PHARMAZIE, 2023, 356 (02)论文数: 引用数: h-index:机构:Radwan, A. M.论文数: 0 引用数: 0 h-index: 0机构: Al Azhar Univ, Fac Sci Girls, Dept Chem, Cairo 11754, Egypt Al Azhar Univ, Fac Sci Girls, Dept Chem, Cairo 11754, EgyptElmetwally, Amira M.论文数: 0 引用数: 0 h-index: 0机构: Egyptian Drug Author EDA, Dept Raw Mat, Giza, Egypt Al Azhar Univ, Fac Sci Girls, Dept Chem, Cairo 11754, EgyptAmmar, Yousry A.论文数: 0 引用数: 0 h-index: 0机构: Al Azhar Univ, Fac Sci Boys, Dept Chem, Cairo 11884, Egypt Al Azhar Univ, Fac Sci Girls, Dept Chem, Cairo 11754, Egypt论文数: 引用数: h-index:机构:
- [44] Surrogating and redirection of pyrazolo[1,5-a]pyrimidin-7(4H)-one core, a novel class of potent and selective DPP-4 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (04) : 903 - 912Deng, Xinxian论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China China State Inst Pharmaceut Ind, 285 Gebaini Rd, Shanghai 201203, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaShen, Jian论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Viva Biotech Ltd Shanghai, 334 Aidisheng Rd, Shanghai 201203, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaZhu, Hui论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Shanghai Peoples Hosp 9, Dept Endocrinol, Sch Med, 369 Zhizaoju Rd, Shanghai 200011, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaXiao, Jia论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaSun, Ran论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaXie, Fangzhou论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaLam, Celine论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaWang, Juntao论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaQiao, Yixue论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China论文数: 引用数: h-index:机构:Hu, Yang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaDue, Yi论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Med, Xinhua Hosp, 1665 Kongjiang Rd, Shanghai 200092, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaLi, Jianqi论文数: 0 引用数: 0 h-index: 0机构: China State Inst Pharmaceut Ind, 285 Gebaini Rd, Shanghai 201203, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaFu, Lei论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R ChinaJiang, Faqin论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China Shanghai Jiao Tong Univ, Sch Pharm, 800 Dongchuan Rd, Shanghai 200240, Peoples R China
- [45] Discovery of novel pyrazolo[1,5-a]pyrimidine derivatives as selective ROCK2 inhibitors with anti-breast cancer migration and invasion activitiesBIOORGANIC CHEMISTRY, 2024, 151Cao, Zhi论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaWei, Xiujian论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaXing, Shuming论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaZhang, Jiahao论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaWang, Shuqi论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaYue, Lingfeng论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaZhang, Jiahe论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaJiang, Nan论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R ChinaZhai, Xin论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China
- [46] Discovery of Pyrazolo[1,5-a]pyrimidine TTK Inhibitors: CFI-402257 is a Potent, Selective, Bioavailable Anticancer AgentACS MEDICINAL CHEMISTRY LETTERS, 2016, 7 (07): : 671 - 675Liu, Yong论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Campbell Family Inst Breast Canc Res, MaRS Ctr, TMDT East Tower,101 Coll St, Toronto, ON M5G 1L7, Canada Univ Hlth Network, Campbell Family Inst Breast Canc Res, MaRS Ctr, TMDT East Tower,101 Coll St, Toronto, ON M5G 1L7, CanadaLaufer, Radoslaw论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Campbell Family Inst Breast Canc Res, MaRS Ctr, TMDT East Tower,101 Coll St, Toronto, ON M5G 1L7, Canada Univ Hlth Network, Campbell Family Inst Breast Canc Res, MaRS Ctr, TMDT East Tower,101 Coll St, Toronto, ON M5G 1L7, CanadaPatel, Narendra Kumar论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Campbell Family Inst Breast Canc Res, MaRS Ctr, TMDT East Tower,101 Coll St, Toronto, ON M5G 1L7, Canada Univ Hlth Network, Campbell Family Inst Breast Canc Res, MaRS Ctr, 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Canada Univ Hlth Network, Campbell Family Inst Breast Canc Res, MaRS Ctr, TMDT East Tower,101 Coll St, Toronto, ON M5G 1L7, Canada
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- [49] Discovery of Pyrazolo[1,5-a]pyrimidine B-Cell Lymphoma 6 (BCL6) Binders and Optimization to High Affinity Macrocyclic InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2017, 60 (10) : 4386 - 4402McCoull, William论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Oncol & Discovery Sci, 310 Cambridge Sci Pk,Milton Rd, Cambridge CB4 0WG, England AstraZeneca, IMED Oncol & Discovery Sci, 310 Cambridge Sci Pk,Milton Rd, Cambridge CB4 0WG, EnglandAbrams, Roman D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Oncol, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, IMED Oncol & Discovery Sci, 310 Cambridge Sci Pk,Milton Rd, Cambridge CB4 0WG, EnglandAnderson, Erica论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Oncol & Discovery Sci, Gatehouse Pk, Waltham, MA 02451 USA AstraZeneca, IMED Oncol & Discovery Sci, 310 Cambridge Sci Pk,Milton Rd, Cambridge CB4 0WG, EnglandBlades, Kevin论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, IMED Oncol, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England 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