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- [21] Discovery and structure - activity relationship exploration of pyrazolo [1,5-a]pyrimidine derivatives as potent FLT3-ITD inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY, 2021, 48Chen, Yun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China China Pharmaceut Univ, Ctr Drug Discovery, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaBai, Gang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaLi, Yan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaNing, Yi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaCao, Sufen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaZhou, Jinpei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Med Chem, 24 Tongjiaxiang, Nanjing 210009, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaDing, Jian论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaZhang, Huibin论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Ctr Drug Discovery, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaXie, Hua论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Inst Drug Discovery & Dev, Zhongshan 528400, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R ChinaDuan, Wenhu论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Div Small Mol Drug Res Ctr, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China
- [22] Highly selective C3-sulfenylation and C3-selenylation of 3-iodo-5-arylpyrazolo[1,5-a]pyrimidin-7-amine in waterJOURNAL OF MOLECULAR STRUCTURE, 2023, 1292Sang, Tian论文数: 0 引用数: 0 h-index: 0机构: Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R China Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R ChinaJia, Fan论文数: 0 引用数: 0 h-index: 0机构: Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R China Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R ChinaHe, Jing论文数: 0 引用数: 0 h-index: 0机构: Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R China Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R ChinaLiu, Yan论文数: 0 引用数: 0 h-index: 0机构: Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R China Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R ChinaLiu, Jichang论文数: 0 引用数: 0 h-index: 0机构: Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R China Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R ChinaLiu, Ping论文数: 0 引用数: 0 h-index: 0机构: Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R China Shihezi Univ, Sch Chem & Chem Engn, Key Lab Green Proc Chem Engn Xinjiang Bingtuan, Shihezi 832004, Peoples R China
- [23] Efficacy and Tolerability of Pyrazolo[1,5-a]pyrimidine RET Kinase Inhibitors for the Treatment of Lung AdenocarcinomaACS MEDICINAL CHEMISTRY LETTERS, 2020, 11 (04): : 558 - 565Mathison, Casey J. N.论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAChianelli, Donatella论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USARucker, Paul V.论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USANelson, John论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USARoland, Jason论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAHuang, Zhihong论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAYang, Yang论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAJiang, Jiqing论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAXie, Yun Feng论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAEpple, Robert论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USABursulaya, Badry论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USALee, Christian论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAGao, Mu-Yun论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAShaffer, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USABriones, Sergio论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USASarkisova, Yelena论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAGalkin, Anna论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USALi, Lintong论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USALi, Nanxin论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USALi, Chun论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAHua, Su论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAKasibhatla, Shailaja论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAKinyamu-Akunda, Jacqueline论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAKikkawa, Rie论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAMolteni, Valentina论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USATellew, John E.论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA
- [24] Advances in pyrazolo[1,5-a]pyrimidines: synthesis and their role as protein kinase inhibitors in cancer treatmentRSC ADVANCES, 2025, 15 (05) : 3756 - 3828Iorkula, Terungwa H.论文数: 0 引用数: 0 h-index: 0机构: Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAJude-Kelly Osayawe, Osasere论文数: 0 引用数: 0 h-index: 0机构: Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAOdogwu, Daniel A.论文数: 0 引用数: 0 h-index: 0机构: Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAGaniyu, Latifat Oluwatobi论文数: 0 引用数: 0 h-index: 0机构: Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAFaderin, Emmanuel论文数: 0 引用数: 0 h-index: 0机构: Southern Illinois Univ, Dept Pharmaceut Sci, 1Harirpin Dr, Edwardsville, IL 62026 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAAwoyemi, Raymond Femi论文数: 0 引用数: 0 h-index: 0机构: Mississippi State Univ, Dept Chem, Mississippi, MS 39762 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAAkodu, Busayo Odunayo论文数: 0 引用数: 0 h-index: 0机构: Southern Illinois Univ, Dept Pharmaceut Sci, 1Harirpin Dr, Edwardsville, IL 62026 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAIfijen, Ikhazuagbe Hilary论文数: 0 引用数: 0 h-index: 0机构: Rubber Res Inst Nigeria, Dept Res Outreach, Benini City, Nigeria Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAAworinde, Omowunmi Rebecca论文数: 0 引用数: 0 h-index: 0机构: Michigan Technol Univ, Dept Chem, 1400 Townsend Dr, Houghton, MI 49931 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAAgyemang, Peter论文数: 0 引用数: 0 h-index: 0机构: Michigan Technol Univ, Dept Chem, 1400 Townsend Dr, Houghton, MI 49931 USA Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USAOnyinyechi, Odo Lovelyn论文数: 0 引用数: 0 h-index: 0机构: Univ Nigeria, Fac Pharmaceut Sci, Nsukka, Nigeria Brigham Young Univ, Dept Chem & Biochem, Provo, UT 84602 USA
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- [30] Discovery of 3-pyrazolyl-substituted pyrazolo[1,5-a]pyrimidine derivatives as potent TRK inhibitors to overcome clinically acquired resistanceEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 241Gong, Yi论文数: 0 引用数: 0 h-index: 0机构: Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R China Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R ChinaWu, Feng-Xu论文数: 0 引用数: 0 h-index: 0机构: Hubei Univ Med, Sch Pharmaceut Sci, Hubei Key Lab Wudang Local Chinese Med Res, Hubei 442000, Peoples R China Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R ChinaWang, Ming-Shu论文数: 0 引用数: 0 h-index: 0机构: Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R China Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R ChinaXu, Hong-Chuang论文数: 0 引用数: 0 h-index: 0机构: Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R China Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R ChinaZhuo, Lin-Sheng论文数: 0 引用数: 0 h-index: 0机构: Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R China Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R ChinaYang, Guang-Fu论文数: 0 引用数: 0 h-index: 0机构: Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R China Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R ChinaHuang, Wei论文数: 0 引用数: 0 h-index: 0机构: Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R China Cent China Normal Univ, Key Lab Pesticide & Chem Biol, Int Joint Res Ctr Intelligent Biosensor Technol &, Coll Chem,Minist Educ, Wuhan 430079, Peoples R China