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- [31] Discovery of CX-6258. A Potent, Selective, and Orally Efficacious pan-Pim Kinases InhibitorACS MEDICINAL CHEMISTRY LETTERS, 2012, 3 (02): : 135 - 139Haddach, Mustapha论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAMichaux, Jerome论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USASchwaebe, Michael K.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAPierre, Fabrice论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAO'Brien, Sean E.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USABorsan, Cosmin论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USATran, Joe论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USARaffaele, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USARavula, Suchitra论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USADrygin, Denis论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USASiddiqui-Jain, Adam论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USADarjania, Levan论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAStansfield, Ryan论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAProffitt, Chris论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAMacalino, Diwata论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAStreiner, Nicole论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USABliesath, Joshua论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAOmori, May论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAWhitten, Jeffrey P.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USAAnderes, Kenna论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USARice, William G.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USARyckman, David M.论文数: 0 引用数: 0 h-index: 0机构: Cylene Pharmaceut Inc, San Diego, CA 92121 USA Cylene Pharmaceut Inc, San Diego, CA 92121 USA
- [32] Discovery of EBI-1051: A novel and orally efficacious MEK inhibitor with benzofuran scaffoldBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (03) : 581 - 589Lu, Biao论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaHuang, Song论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaCao, Jingsong论文数: 0 引用数: 0 h-index: 0机构: Etern Biosci Inc, 6 Cedarbrook Dr, Cranbury, NJ 08512 USA Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaHu, Qiyue论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaShen, Ru论文数: 0 引用数: 0 h-index: 0机构: Etern Biosci Inc, 6 Cedarbrook Dr, Cranbury, NJ 08512 USA Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaWan, Hong论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaWang, Dan论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaYuan, Jijun论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Etern Biosci Inc, 6 Cedarbrook Dr, Cranbury, NJ 08512 USA Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaZhang, Lei论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Etern Biosci Inc, 6 Cedarbrook Dr, Cranbury, NJ 08512 USA Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaZhang, Jiayin论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaZhang, Minsheng论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaTao, Weikang论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R ChinaZhang, Lianshan论文数: 0 引用数: 0 h-index: 0机构: Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China Shanghai Hengrui Pharmaceut Co Ltd, 279 Wenjing Rd, Shanghai 200245, Peoples R China
- [33] Discovery of an Orally Efficacious Inhibitor of Anaplastic Lymphoma KinaseJOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (10) : 4580 - 4593Gingrich, Diane E.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USALisko, Joseph G.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USACurry, Matthew A.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USACheng, Mangeng论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAQuail, Matthew论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USALu, Lihui论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAWan, Weihua论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAAlbom, Mark S.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAAngeles, Thelma S.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAAimone, Lisa D.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAHaltiwanger, R. Curtis论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAWells-Knecht, Kevin论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAOtt, Gregory R.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAGhose, Arup K.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USAAtor, Mark A.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USARuggeri, Bruce论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USADorsey, Bruce D.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA Cephalon Inc, Worldwide Discovery Res, W Chester, PA 19380 USA
- [34] Discovery of novel and potent sulfonamide derivatives as orally available drug for psoriasisBIOORGANIC CHEMISTRY, 2024, 153Qi, Liang论文数: 0 引用数: 0 h-index: 0机构: Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R China Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R ChinaPing, Yi-Nuo论文数: 0 引用数: 0 h-index: 0机构: Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R China Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R ChinaSun, Shang-Shang论文数: 0 引用数: 0 h-index: 0机构: Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R China Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R ChinaXu, Ran论文数: 0 引用数: 0 h-index: 0机构: Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R China Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R ChinaZhou, Xin-Ru论文数: 0 引用数: 0 h-index: 0机构: Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R China Jiangsu Med Coll, Sch Pharm, Yancheng 224005, Jiangsu, Peoples R China
- [35] Discovery of novel, potent and orally available MAT2A inhibitorsCANCER RESEARCH, 2023, 83 (07)Chen, Xuxing论文数: 0 引用数: 0 h-index: 0Li, Jing论文数: 0 引用数: 0 h-index: 0Chen, Yanhong论文数: 0 引用数: 0 h-index: 0
- [36] Discovery of tetrahydroindazoles as a novel class of potent and in vivo efficacious gamma secretase modulatorsBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (12) : 3227 - 3241Gerlach, Kai论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, GermanyHobson, Scott论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Cent Nervous Syst Dis Res, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, GermanyEickmeier, Christian论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, GermanyGross, Ulrike论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, GermanyBraun, Clemens论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Drug Discovery Sci, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, GermanySieger, Peter论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Drug Discovery Sci, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, GermanyGarneau, Michel论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Drug Discovery Sci, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, GermanyHoerer, Stefan论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, GermanyHeine, Niklas论文数: 0 引用数: 0 h-index: 0机构: Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, Germany Boehringer Ingelheim Pharma GmbH & Co KG, Med Chem, Birkendorfer Str 65, D-88397 Biberach, Germany
- [37] Discovery of novel, potent and orally bioavailable CRTH2 antagonistsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241Terasaka, Tadashi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanIto, Shinji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanZenkoh, Tatsuya论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanHayashida, Hisashi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanMatsuda, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanMiyata, Junji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanNagata, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanTakasuna, Yuji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanKobayashi, Miki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanTakeuchi, Makoto论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, JapanOhta, Mitsuaki论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, Tsukuba, Ibaraki, Japan
- [38] Discovery of a novel sulfonamide-pyrazolopiperidine series as potent and Efficacious γ-Secretase InhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (07) : 2195 - 2199Ye, Xiaocong M.论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USAKonradi, Andrei W.论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USASmith, Jenifer论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USAXu, Ying-Zi论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USADressen, Darren论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USAGarofalo, Albert W.论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USAMarugg, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USASham, Hing L.论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USATruong, Anh P.论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USAJagodzinski, Jacek论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Proc & Analyt Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USAPleiss, Michael论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USAZhang, Hongbin论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Lead Discovery & Optimizat, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USAGoldbach, Erich论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Lead Discovery & Optimizat, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USASauer, John-Michael论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Lead Discovery & Optimizat, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USABrigham, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Vivo Pharmacol, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USABova, Michael论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Biol, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USABasi, Guriqbal S.论文数: 0 引用数: 0 h-index: 0机构: Elan Pharmaceut, Dept Biol, San Francisco, CA 94080 USA Elan Pharmaceut, Dept Med Chem, San Francisco, CA 94080 USA
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