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- [1] Discovery of a potent, highly selective, and orally efficacious small-molecule activator of the insulin receptorJOURNAL OF MEDICINAL CHEMISTRY, 2000, 43 (19) : 3487 - 3494Liu, K论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAXu, LB论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USASzalkowski, D论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USALi, ZH论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USADing, V论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAKwei, G论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAHuskey, S论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAMoller, DE论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAHeck, JV论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAZhang, BB论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USAJones, AB论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Rahway, NJ 07065 USA Merck Res Labs, Rahway, NJ 07065 USA
- [2] Discovery of structurally novel, potent and orally efficacious GPR119 agonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (10) : 2383 - 2387Alper, Phil论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAAzimioara, Mihai论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USACow, Christopher论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAMutnick, Daniel论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USANikulin, Victor论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAMichellys, Pierre-Yves论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAWang, Zhiliang论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAReding, Esther论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAPaliotti, Michael论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USALi, Jing论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USABao, Dingjiu论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAZoll, Jocelyn论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAKim, Young论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAZimmerman, Matthew论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAGroessel, Todd论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USATuntland, Tove论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAJoseph, Sean B.论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAMcNamara, Peter论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USASeidel, H. Martin论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USAEpple, Robert论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA
- [3] Discovery of a Potent and Orally Efficacious TGR5 Receptor AgonistACS MEDICINAL CHEMISTRY LETTERS, 2016, 7 (01): : 51 - 55Agarwal, Sameer论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaPatil, Amit论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaAware, Umesh论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaDeshmukh, Prashant论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaDarji, Brijesh论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaSasane, Santosh论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaSairam, Kalapatapu V. V. M.论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaPriyadarsiny, Priyanka论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaGiri, Poonam论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaPatel, Harilal论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaGiri, Suresh论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaJain, Mukul论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, IndiaDesai, Ranjit C.论文数: 0 引用数: 0 h-index: 0机构: Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India Cadila Healthcare Ltd, Zydus Res Ctr, Sarkhej Bavla NH 8 A, Ahmadabad 382210, Gujarat, India
- [4] Discovery of DNP-60502, a novel, potent AMPK activator for the treatment of metabolic syndromeABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 237Okano, Koji论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, JapanHashimoto, Masakazu论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Pharmacol, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, JapanKodama, Tomohiro论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, JapanIwata, Mitsutaka论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, JapanKohayakawa, Chie论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Pharmacol, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, JapanTanaka, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, JapanYano, Akihiro论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Pharmacol, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, JapanTsuji, Jun-ichi论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Pharmacol, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, JapanSato, Fuminori论文数: 0 引用数: 0 h-index: 0机构: Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, Japan Dainippon Sumitomo Pharma Co Ltd, Dept Chem, Konohana Ku, Osaka 5540022, Japan
- [5] Discovery of CLPP-1071 as an Exceptionally Potent and Orally Efficacious Human ClpP Activator with Strong In Vivo Antitumor ActivityJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (23) : 21009 - 21029Chen, Beijing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Guizhou Med Univ, Sch Pharm, Guiyang 550014, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaSun, Mingyang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaZhang, Chun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Zunyi Med Univ, Sch Pharm, Zunyi 563000, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaHuang, Qi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Fudan Univ, Sch Pharm, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaTeng, Dan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaHu, Linghao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Chinese Acad Sci, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaMa, Huicong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Zunyi Med Univ, Sch Pharm, Zunyi 563000, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaLin, Xinyi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Southern Med Univ, Sch Pharmaceut Sci, Guangzhou 510515, Guangdong, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaHuang, Zan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaGui, Renzhao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaHu, Xiaobei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaXu, Lei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaZheng, Mingyue论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Design Ctr, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaZhou, Yubo论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Chinese Acad Sci, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaLi, Jia论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Guizhou Med Univ, Sch Pharm, Guiyang 550014, Peoples R China Chinese Acad Sci, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, State Key Lab Chem Biol, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R ChinaWang, Mingliang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China Zunyi Med Univ, Sch Pharm, Zunyi 563000, Peoples R China Chinese Acad Sci, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Zhongshan Inst Drug Discovery, Shanghai Inst Mat Med, Zhongshan 528400, Guangdong, Peoples R China
- [6] Discovery of potent, highly selective and orally efficacious SMARCA2 degradersCANCER RESEARCH, 2024, 84 (06)Leng, Lingying论文数: 0 引用数: 0 h-index: 0Yang, Lin论文数: 0 引用数: 0 h-index: 0Tu, Wenbin论文数: 0 引用数: 0 h-index: 0Rej, Rohan论文数: 0 引用数: 0 h-index: 0Allu, Srinivasa Rao论文数: 0 引用数: 0 h-index: 0Huang, Liyue论文数: 0 引用数: 0 h-index: 0Jiang, Wei论文数: 0 引用数: 0 h-index: 0Wang, Yu论文数: 0 引用数: 0 h-index: 0Stuckey, Jeanne论文数: 0 引用数: 0 h-index: 0Sarkari, Farzad R.论文数: 0 引用数: 0 h-index: 0Wang, Meilin论文数: 0 引用数: 0 h-index: 0Wang, Lu论文数: 0 引用数: 0 h-index: 0Wen, Bo论文数: 0 引用数: 0 h-index: 0Sun, Duxin论文数: 0 引用数: 0 h-index: 0Wang, Shaomeng论文数: 0 引用数: 0 h-index: 0
- [7] The discovery of BMS-275183: An orally efficacious novel taxaneBIOORGANIC & MEDICINAL CHEMISTRY, 2003, 11 (20) : 4315 - 4323Mastalerz, H论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USACook, D论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAFairchild, CR论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAHansel, S论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAJohnson, W论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAKadow, JF论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USALong, BH论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USARose, WC论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USATarrant, J论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAWu, MJ论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAMay, QF论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAZhang, GF论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAZoeckler, M论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USAVyas, DM论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Wallingford, CT 06492 USA
- [8] Discovery of YS-363 as a highly potent, selective, and orally efficacious EGFR inhibitorBIOMEDICINE & PHARMACOTHERAPY, 2023, 167He, Pengxing论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaJing, Jing论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaDu, Linna论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaZhang, Xuyang论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaRen, Yufei论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaYang, Han论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaYu, Bin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R ChinaLiu, Hongmin论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China
- [9] The discovery of a potent orally efficacious indole androgen receptor antagonist through in vivo screeningBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (01) : 123 - 126Lanter, James C.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USAFiordeliso, James J.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USAJiang, Weiqin论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USAAllan, George F.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USALai, Muh-Tsann论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USALinton, Olivia论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USAHahn, Do Won论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USALundeen, Scott G.论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USASui, Zhihua论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA Johnson & Johnson Pharmaceut Res & Dev LLC, Exton, PA 19341 USA
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