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- [31] Discovery of G2019S-Selective Leucine Rich Repeat Protein Kinase 2 inhibitors with in vivo efficacyEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 229Lesniak, Robert K.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USANichols, R. Jeremy论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Dept Pathol, 300 Pasteur Dr, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USASchonemann, Marcus论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Dept Pathol, 300 Pasteur Dr, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USAZhao, Jing论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Dept Pathol, 300 Pasteur Dr, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USAGajera, Chandresh R.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Dept Pathol, 300 Pasteur Dr, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USAFitch, William L.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Sch Med, Div Gastroenterol & Hepatol, Dept Med, Stanford, CA 94305 USA Stanford Univ, Sch Med, Div Gastroenterol & Hepatol, Dept Microbiol & Immunol, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USALam, Grace论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Sch Med, Div Gastroenterol & Hepatol, Dept Med, Stanford, CA 94305 USA Stanford Univ, Sch Med, Div Gastroenterol & Hepatol, Dept Microbiol & Immunol, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USANguyen, Khanh C.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Sch Med, Div Gastroenterol & Hepatol, Dept Med, Stanford, CA 94305 USA Stanford Univ, Sch Med, Div Gastroenterol & Hepatol, Dept Microbiol & Immunol, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USASmith, Mark论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USAMontine, Thomas J.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Dept Pathol, 300 Pasteur Dr, Stanford, CA 94305 USA Stanford Univ, Med Chem Knowledge Ctr, Stanford ChEM H, Stanford, CA 94305 USA
- [32] Sphingosine Kinase 2 Inhibitors: Rigid Aliphatic Tail Derivatives Deliver Potent and Selective AnaloguesACS BIO & MED CHEM AU, 2022, 2 (05): : 469 - 489Pashikanti, Srinath论文数: 0 引用数: 0 h-index: 0机构: Virginia Tech, Dept Chem, Blacksburg, VA 24060 USA Idaho State Univ, Dept Biomed & Pharmaceut Sci, Pocatello, ID 83209 USA Virginia Tech, Dept Chem, Blacksburg, VA 24060 USAFoster, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: Virginia Tech, Dept Chem, Blacksburg, VA 24060 USA Virginia Tech, Dept Chem, Blacksburg, VA 24060 USA论文数: 引用数: h-index:机构:Brown, Anne M.论文数: 0 引用数: 0 h-index: 0机构: Virginia Tech, Virginia Tech Ctr Drug Discovery, Blacksburg, VA 24060 USA Virginia Tech, Dept Biochem, Blacksburg, VA 24060 USA Virginia Tech, Dept Chem, Blacksburg, VA 24060 USABevan, David R.论文数: 0 引用数: 0 h-index: 0机构: Virginia Tech, Virginia Tech Ctr Drug Discovery, Blacksburg, VA 24060 USA Virginia Tech, Dept Biochem, Blacksburg, VA 24060 USA Virginia Tech, Dept Chem, Blacksburg, VA 24060 USALynch, Kevin R.论文数: 0 引用数: 0 h-index: 0机构: Univ Virginia, Dept Pharmacol, Charlottesville, VA 22908 USA Virginia Tech, Dept Chem, Blacksburg, VA 24060 USASantos, Webster L.论文数: 0 引用数: 0 h-index: 0机构: Virginia Tech, Dept Chem, Blacksburg, VA 24060 USA Virginia Tech, Virginia Tech Ctr Drug Discovery, Blacksburg, VA 24060 USA Virginia Tech, Dept Chem, Blacksburg, VA 24060 USA
- [33] Synthesis and biological evaluation of sphingosine kinase 2 inhibitors with anti-inflammatory activityARCHIV DER PHARMAZIE, 2019, 352 (03)Vettorazzi, Marcela论文数: 0 引用数: 0 h-index: 0机构: Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, Argentina Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaVila, Laura论文数: 0 引用数: 0 h-index: 0机构: Univ Valencia, Dept Pharmacol, Valencia, Spain Univ Clin Hosp Valencia, INCLIVA, Inst Hlth Res, Valencia, Spain Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaLima, Santiago论文数: 0 引用数: 0 h-index: 0机构: Virginia Commonwealth Univ, Dept Biol, Richmond, VA 23284 USA Virginia Commonwealth Univ, Dept Biochem & Mol Biol, Sch Med, Richmond, VA USA Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaAcosta, Lina论文数: 0 引用数: 0 h-index: 0机构: Univ Ind Santander, Escuela Quim, Lab Sintesis Organ, Bucaramanga, Colombia Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaYepes, Felipe论文数: 0 引用数: 0 h-index: 0机构: Univ Ind Santander, Escuela Quim, Lab Sintesis Organ, Bucaramanga, Colombia Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaPalma, Alirio论文数: 0 引用数: 0 h-index: 0机构: Univ Ind Santander, Escuela Quim, Lab Sintesis Organ, Bucaramanga, Colombia Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaCobo, Justo论文数: 0 引用数: 0 h-index: 0机构: Univ Jaen, Inorgan & Organ Dept, Jaen, Spain Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaTengler, Jan论文数: 0 引用数: 0 h-index: 0机构: Medis Int As, Bolatice, Czech Republic Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaMalik, Ivan论文数: 0 引用数: 0 h-index: 0机构: Comenius Univ, Dept Pharmaceut Chem, Fac Pharm, Bratislava, Slovakia Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaAlvarez, Sergio论文数: 0 引用数: 0 h-index: 0机构: Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, Argentina Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaMarques, Patrice论文数: 0 引用数: 0 h-index: 0机构: Univ Valencia, Dept Pharmacol, Valencia, Spain Univ Clin Hosp Valencia, INCLIVA, Inst Hlth Res, Valencia, Spain Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaCabedo, Nuria论文数: 0 引用数: 0 h-index: 0机构: Univ Valencia, Dept Pharmacol, Valencia, Spain Univ Clin Hosp Valencia, INCLIVA, Inst Hlth Res, Valencia, Spain Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, ArgentinaSanz, Maria J.论文数: 0 引用数: 0 h-index: 0机构: Univ Valencia, Dept Pharmacol, Valencia, Spain Univ Clin Hosp Valencia, INCLIVA, Inst Hlth Res, Valencia, Spain Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, Argentina论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Enriz, Ricardo D.论文数: 0 引用数: 0 h-index: 0机构: Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, Argentina Univ Nacl San Luis, Inst Multidisciplinario Invest Biol IMIBIO SL, Fac Quim Bioquim & Farm, Chacabuco 915, RA-5700 San Luis, Argentina
- [34] Structure-Guided Discovery of Selective USP7 Inhibitors with In Vivo ActivityJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (21) : 18993 - 19009Vasas, Attila论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryIvanschitz, Lisa论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-91190 Gif Sur Yvette, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryMolnar, Balazs论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryKiss, Arpad论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryBaker, Lisa论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryFiumana, Andrea论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryMacias, Alba论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryMurray, James B.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungarySanders, Emma论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryWhitehead, Neil论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryHubbard, Roderick E.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungarySaunier, Carine论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-91190 Gif Sur Yvette, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryMonceau, Elodie论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-91190 Gif Sur Yvette, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryGirard, Anne Marie论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-91190 Gif Sur Yvette, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryRousseau, Marion论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-91190 Gif Sur Yvette, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryChanrion, Maia论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-91190 Gif Sur Yvette, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryDemarles, Didier论文数: 0 引用数: 0 h-index: 0机构: Technol Servier, F-45000 Orleans, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryGeneste, Olivier论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-91190 Gif Sur Yvette, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryWeber, Csaba论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryLewkowicz, Elodie论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-91190 Gif Sur Yvette, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryKotschy, Andras论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, Hungary
- [35] Discovery of potent and selective focal adhesion kinase inhibitorsEJC SUPPLEMENTS, 2008, 6 (12): : 43 - 43Kawahara, E.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanMiyake, T.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanMatsuura, N.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanUmemura, I.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanMasuya, K.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanKanazawa, T.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanMeyer, T.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanMestan, J.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanHatakeyama, S.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, JapanOhmori, O.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki, Japan
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