New class TRPM8 antagonist, voacangine is the first natural competitive antagonist for menthol receptor, TRPM8

被引:0
|
作者
Terada, Yuko [1 ]
Horie, Syunji [2 ]
Takayama, Hiromitsu [3 ]
Watanabe, Tatsuo [1 ]
机构
[1] Univ Shizuoka, Dept Nutr & Environm Sci, Shizuoka 4228526, Japan
[2] Josai Int Univ, Dept Pharmaceut Sci, Togane, Chiba 2838555, Japan
[3] Chiba Univ, Dept Biofunct Mol Chem, Yayoi, Chiba 2638522, Japan
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
384-MEDI
引用
收藏
页数:1
相关论文
共 50 条
  • [41] Identification of a Potent Tryptophan-Based TRPM8 Antagonist With in Vivo Analgesic Activity
    Bertamino, Alessia
    Iraci, Nunzio
    Ostacolo, Carmine
    Arnbrosino, Paolo
    Musella, Simona
    Di Sarno, Veronica
    Ciaglia, Tania
    Pepe, Giacomo
    Sala, Marina
    Soldovier, Maria Virginia
    Mosca, Ilaria
    Gonzalez-Rodriguez, Sara
    Fernandez-Carvajal, Asia
    Ferrer-Montiel, Antonio
    Novellino, Ettore
    Taglialatela, Maurizio
    Campiglia, Pietro
    Gomez-Monterrey, Isabel
    JOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (14) : 6140 - 6152
  • [42] TRPM8 Biology and Medicinal Chemistry
    DeFalco, Jeff
    Duncton, Matthew A. J.
    Emerling, Daniel
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2011, 11 (17) : 2237 - 2252
  • [43] TRPM8 and prostate: a cold case?
    Noyer, Lucile
    Grolez, Guillaume P.
    Prevarskaya, Natalia
    Gkika, Dimitra
    Lemonnier, Loic
    PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 2018, 470 (10): : 1419 - 1429
  • [44] Molecular mechanism of desensitization of TRPM8
    Hosokawa, Hiroshi
    Abe, Junji
    Yamanaka, Keiji
    Matsumura, Kiyoshi
    Kobayashi, Shigeo
    NEUROSCIENCE RESEARCH, 2006, 55 : S140 - S140
  • [45] Discovery of AMG 333: A potent, orally bioavailable TRPM8 antagonist for the treatment of migraine
    Horne, Daniel
    Biswas, Kaustav
    Brown, James
    Gore, Vijay
    Harried, Scott
    Kaller, Matthew
    Ma, Vu
    Monenschein, Holger
    Nguyen, Thomas
    Zhong, Wenge
    Bartberger, Michael
    Davis, Carl
    Rose, Mark
    Horner, Michelle
    Wu, Tian
    Sandrock, Robert
    Lehto, Sonya
    Rao, Sara
    Youngblood, Beth
    Zhang, Maosheng
    Zhu, Dawn
    Gavva, Narender
    Chen, Jian
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250
  • [46] TRPM8 influences bladder filling
    Peter Sidaway
    Nature Reviews Urology, 2015, 12 (9) : 476 - 476
  • [47] Cooling the Itch via TRPM8
    Liu, Boyi
    Jordt, Sven-Eric
    JOURNAL OF INVESTIGATIVE DERMATOLOGY, 2018, 138 (06) : 1254 - 1256
  • [48] Structure of human TRPM8 channel
    Sergii Palchevskyi
    Mariusz Czarnocki-Cieciura
    Giulio Vistoli
    Silvia Gervasoni
    Elżbieta Nowak
    Andrea R. Beccari
    Marcin Nowotny
    Carmine Talarico
    Communications Biology, 6
  • [49] Regulation of TRPM8 channel activity
    Yudin, Yevgen
    Rohacs, Tibor
    MOLECULAR AND CELLULAR ENDOCRINOLOGY, 2012, 353 (1-2) : 68 - 74
  • [50] Structure of human TRPM8 channel
    Palchevskyi, Sergii
    Czarnocki-Cieciura, Mariusz
    Vistoli, Giulio
    Gervasoni, Silvia
    Nowak, Elzbieta
    Beccari, Andrea R.
    Nowotny, Marcin
    Talarico, Carmine
    COMMUNICATIONS BIOLOGY, 2023, 6 (01)