New class TRPM8 antagonist, voacangine is the first natural competitive antagonist for menthol receptor, TRPM8

被引：0
|
作者：
Terada, Yuko [1 ]
Horie, Syunji [2 ]
Takayama, Hiromitsu [3 ]
Watanabe, Tatsuo [1 ]
机构：
[1] Univ Shizuoka, Dept Nutr & Environm Sci, Shizuoka 4228526, Japan
[2] Josai Int Univ, Dept Pharmaceut Sci, Togane, Chiba 2838555, Japan
[3] Chiba Univ, Dept Biofunct Mol Chem, Yayoi, Chiba 2638522, Japan
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2013年 / 245卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
384-MEDI
引用
收藏
页数：1
相关论文
共 50 条
  • [31] Antitussive Effect of (-) Menthol: the Role of Nasal Trigeminal Trpm8 Receptors
    Plevkova, J.
    Surdenikova, L.
    Poliacek, I
    Tatar, M.
    Kollarik, M.
    Canning, B. J.
    LUNG, 2012, 190 (01) : 64 - 65
  • [32] The menthol and cold sensation receptor TRPM8 in normal human nasal mucosa and rhinitis
    Keh, Siew M.
    Facer, Paul
    Yehia, Ahmed
    Sandhu, Guri
    Saleh, Hesham A.
    Anand, Praveen
    RHINOLOGY, 2011, 49 (04) : 453 - 457
  • [33] Design and optimization of benzimidazole-containing cold menthol receptor (TRPM8) antagonists
    Parks, Daniel J.
    Calvo, Raul R.
    Parsons, William H.
    Meegalla, Sanath
    Ballentine, Shelley K.
    Chen, Jinsheng
    Illig, Carl R.
    Stone, Dennis J.
    Qin, Ning
    Hutchinson, Tasha L.
    Lubin, Mary Lou
    Liu, Yi
    Baker, Judith
    Colburn, Raymond W.
    Flores, Christopher M.
    Player, Mark R.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240
  • [34] Modeling the Menthol Binding Pocket Within TRPM8 Ion Channel
    Replogle, Jessica
    Cutforth, Siena
    Dobelhoff, Katie
    Moran, Elizabeth
    Suder, Karen
    FASEB JOURNAL, 2021, 35
  • [35] Effects of the TRPM8 Agonist Menthol on Corneal Sensitivity and Tear Secretion
    Belmonte, J.
    Alfaro, S.
    Berenguer, T. B.
    Costa, J. M.
    Cuquerella, V.
    Acosta, M. C.
    Belmonte, C.
    Gallar, J.
    INVESTIGATIVE OPHTHALMOLOGY & VISUAL SCIENCE, 2010, 51 (13)
  • [36] Identification of the cold receptor TRPM8 in the nasal mucosa
    Liu, Shao-Cheng
    Lu, Hsuan-Hsuan
    Cheng, Li-Hsiang
    Chu, Yueng-Hsiang
    Lee, Fei-Peng
    Wu, Chi-Chung
    Wang, Hsing-Won
    AMERICAN JOURNAL OF RHINOLOGY & ALLERGY, 2015, 29 (04) : E112 - E116
  • [37] Discovery of a Selective TRPM8 Antagonist with Clinical Efficacy in Cold-Related Pain
    Andrews, Mark D.
    af Forselles, Kerry
    Beaumont, Kevin
    Galan, Sebastien R. G.
    Glossop, Paul A.
    Grenie, Mathilde
    Jessiman, Alan
    Kenyon, Amy S.
    Lunn, Graham
    Maw, Graham
    Owen, Robert M.
    Pryde, David C.
    Roberts, Dannielle
    Thien Duc Tran
    ACS MEDICINAL CHEMISTRY LETTERS, 2015, 6 (04): : 419 - 424
  • [38] Distribution of transient receptor potential melastatin type-8 (TRPM8) and effects of TRPM8 agonists in mouse lower gastrointestinal tract
    Hosoya, Takuji
    JOURNAL OF PHARMACOLOGICAL SCIENCES, 2010, 112 : 52P - 52P
  • [39] Trigeminal Neuralgia TRPM8 Mutation
    Gualdani, Roberta
    Yuan, Jun-Hui
    Effraim, Philip R.
    Di Stefano, Giulia
    Truini, Andrea
    Cruccu, Giorgio
    Dib-Hajj, Sulayman D.
    Gailly, Philippe
    Waxman, Stephen G.
    NEUROLOGY-GENETICS, 2021, 7 (01)
  • [40] TRPM8的研究现状
    关荣华
    林小娥
    科学技术创新, 2017, (26) : 4 - 5
12345