IODINE MEDIATED ONE-POT SYNTHESIS OF IMIDAZO[1,5-a]AZINES FROM DITHIOESTERS

被引：0
|
作者：
Ramesh, Ajjahalli B. [1 ]
Sandhya, N. C. [1 ]
Swarup, H. A. [1 ]
Mantelingu, Kempegowda [1 ]
Rangappa, Kanchugarakoppal S. [1 ]
机构：
[1] Univ Mysore, Chem, Mysore 570006, Karnataka, India
来源：
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2015年 / 24卷 / 04期
关键词：
RECEPTOR ANTAGONISTS; DERIVATIVES; CYCLIZATION; INHIBITOR; DISCOVERY;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Iodine mediated desulfuritive cyclization of insitu generated thioamides serves as efficient and versatile method for the synthesis of imidazo[1,5-a]azines with excellent yields. Substrates such as 2-methylanninoquinoline and pyrazin-2-ylmethanannine also undergoes the corresponding reactions at room temperature. This method has the advantages of mild conditions, short reaction time and high yields.
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页码：465 / 472
页数：8
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