Design and discovery of macrocyclic diaminopropanes as potent inhibitors of BACE1

被引：0

作者：

Marcin, Lawrence R. ^{[1
]}

Thompson, Lorin A. ^{[1
]}

Higgins, Mendi A. ^{[1
]}

Shi, JianLiang ^{[1
]}

Boy, Kenneth M. ^{[1
]}

Olson, Richard E. ^{[1
]}

Good, Andrew C. ^{[2
]}

Burton, Catherine R. ^{[3
]}

Barten, Donna M. ^{[4
]}

Muckelbauer, Jodi K. ^{[5
]}

Calambur, Deepa ^{[5
]}

Camac, Daniel M. ^{[5
]}

Chang, ChiehYing ^{[5
]}

Toyn, Jeremy H. ^{[3
]}

Lentz, Kimberley A. ^{[6
]}

Grace, James E. ^{[6
]}

Herbst, Grace John J. ^{[7
]}

Marino, Anthony M. ^{[6
]}

Meredith, Jere E. ^{[3
]}

Albright, Charlie F. ^{[3
]}

Macor, John E. ^{[8
]}

机构：

[1] Bristol Myers Squibb Res & Dev, Neurosci Discovery Chem, Wallingford, CT 06492 USA

[2] Genzyme Corp, Cambridge, MA USA

[3] Bristol Myers Squibb Co, Neurosci Biol, New York, NY 10154 USA

[4] Bristol Myers Squibb Co, Neurosci Discovery Biol, New York, NY 10154 USA

[5] Bristol Myers Squibb Co, Macromol Crystallog, New York, NY 10154 USA

[6] Bristol Myers Squibb Co, Pharmaceut Candidate Optimizat, New York, NY 10154 USA

[7] Bristol Myers Squibb Co, Lead Profiling, New York, NY 10154 USA

[8] Bristol Myers Squibb Res & Dev, Neurosci Chem, Wallingford, CT 06492 USA

来源：

ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2009年 / 238卷

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

212-MEDI

引用

页数：1

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