Synthesis and characterization of novel 1,2,3-triazole-linked theophylline and coumarin s-triazines

被引：0

作者：

Joshi, Penny ^{[1
,2
]}

Tripathi, Mohit ^{[1
]}

Rawat, Diwan S. ^{[1
]}

机构：

[1] Univ Delhi, Dept Chem, Delhi 110007, India

[2] Kumaun Univ, Dept Chem, Naini Tal 263001, India

来源：

INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2014年 / 53卷 / 03期

关键词：

s-Triazine; dendrimer; triazole; theophylline; coumarin; VITRO ANTIMALARIAL ACTIVITY; IMPROVED IN-VITRO; ANTIBACTERIAL ACTIVITY; DRUG-DELIVERY; DERIVATIVES; HYBRIDS; CYTOTOXICITY; DENDRIMERS; ANALOGS; DESIGN;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of novel s-triazine-1,2,3-triazole-theophylline and s-triazine-1,2,3-triazole-coumarin generation-0 dendrimers has been synthesized and characterized by FT-IR, H-1 and C-13 NMR, and mass-spectral methods. Some 'selected compounds have been evaluated for antibacterial and antifungal activity against a variety of strains and for anti-cancer activity against 60 human cancer cell lines.

引用

页码：311 / 318

页数：8

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