Palladium heteroannulation process for synthesis of substituted pyrrolo [2,3-b]pyridin-3-ones

被引:51
|
作者
Desarbre, E [1 ]
Merour, JY [1 ]
机构
[1] UNIV ORLEANS,CNRS,INST CHIM ORGAN & ANALYT,F-45067 ORLEANS 2,FRANCE
关键词
D O I
10.1016/0040-4039(95)02079-9
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Substituted-3H-pyrrolo[2,3-b]pyridin-3-ones 7b-d were prepared from 2-amino-3-iodopyridine derivatives 3b-d by palladium carboannulation process with allenic compounds and then oxidative cleavage of the exocyclic carbon-carbon double bond.
引用
收藏
页码:43 / 46
页数:4
相关论文
共 50 条
  • [21] Synthesis and unexpected reactions of 2-hydroxy-3-pyridinylacetic hydrazides. Formation of 2H-pyrrolo[2,3-b]pyridin-2-ones
    Teleha, CA
    Greenberg, RA
    Chorvat, RJ
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 1998, 35 (01) : 145 - 149
  • [22] SYNTHESIS OF PYRROLO[2,3-B]PYRROLE DERIVATIVES
    BLANTON, CD
    WIDBY, JF
    BRIGGS, FH
    JOURNAL OF ORGANIC CHEMISTRY, 1971, 36 (25): : 3929 - &
  • [23] One-pot synthesis of 1,2-disubstituted pyrrolo[2,3-b]quinoxalines via palladium-catalyzed heteroannulation in water
    Keivanloo, Ali
    Bakherad, Mohammad
    Rahimi, Amin
    Taheri, Sayed Ali Naghi
    TETRAHEDRON LETTERS, 2010, 51 (18) : 2409 - 2412
  • [24] Synthesis and Biological Evaluation of 5′-Arylspiro[piperidine-4,3′-pyrrolo-[2,3-b]pyridin] Analogues
    Mudasani, Gopal
    Paidikondala, Kalyani
    Gundla, Rambabu
    Joseph Maddirala, Shambabu
    Das, Viswanath
    CHEMISTRYSELECT, 2021, 6 (14): : 3378 - 3381
  • [25] PYRROLO[2,3-B]PYRIDINES
    ZIMMERMANN, W
    EGER, K
    ROTH, HJ
    ARCHIV DER PHARMAZIE, 1976, 309 (07) : 597 - 600
  • [26] SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF PYRROLO(2,3-B) QUINOLINE, PYRIDO(2,3-B) QUINOLINE AND AZEPINO(2,3-B) QUINOLINE DERIVATIVES
    ZHIDKOVA, AM
    GRANIK, VG
    GLUSHKOV, RG
    POLEZHAEVA, AI
    MASHKOVSKII, MD
    KHIMIKO-FARMATSEVTICHESKII ZHURNAL, 1976, 10 (05): : 18 - 22
  • [27] 6-Substituted-5H-pyrrolo[2,3-b]pyrazines via palladium-catalyzed heteroannulation from N-(3-chloropyrazin-2-yl)methanesulfonamide and alkynes
    Hopkins, CR
    Collar, N
    TETRAHEDRON LETTERS, 2004, 45 (43) : 8087 - 8090
  • [28] SYNTHESIS OF PYRROLO 2,3-B!PYRROLE DERIVATIVES - ORGN
    DEWITTBL.C
    WHIDBY, JF
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1970, (SEP): : 78 - &
  • [29] Facile Synthesis of Fluorinated Pyrrolo[2,3-b]pyridines
    Groth, Ulrich
    Iaroshenko, Viktor O.
    Wang, Yan
    Wesch, Thornas
    SYNLETT, 2009, (03) : 456 - 460
  • [30] New method for the synthesis of pyrrolo[2,3-b]dihydroquinolines
    Syniugin, Anatolii R.
    Chekanov, Maksym O.
    Savitskiy, Pavel V.
    Pashenko, Alexander E.
    Zhuk, Tatyana S.
    Yarmoluk, Sergiy M.
    Fokin, Andrey A.
    TETRAHEDRON LETTERS, 2016, 57 (02) : 213 - 215