Synthesis and pharmacological screening of some substituted benzothiazole derivatives of thioquinazolinone

被引：0
|
作者：
Patel, HH [1 ]
Khedekar, PB [1 ]
Bhusari, KP [1 ]
机构：
[1] Sharad Pawar Coll Pharm, Nagpur 441110, Maharashtra, India
来源：
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2006年 / 15卷 / 03期
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D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Various substituted 2-amino-N-(2-benzothiazolyl) benzamides (IIIa-n) and 2-thio-3-(2-benzothiazolyl-4-(3H)-quinazolines (IVa-n) containing different functional groups have been synthesized by condensing substituted anthranilic acids (I) with substituted 2-aminobenzothiazoles (II) in dry pyridine. The identity of compounds III and IV were confirmed on the basis of their spectral (UV, IR, and H-1 NMR) data. Further, they have been screened for their anticonvulsant activity.
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页码：217 / 220
页数：4
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