Pyridazines .81. A novel 1,2-diazine containing tricyclic system: Synthesis of pyridazino[3,4-b][1,5]benzodiazepin-5-ones as potential HIV-1 reverse transcriptase inhibitors

被引：0

作者：

Heinisch, G ^{[1
]}

Matuszczak, B ^{[1
]}

Mereiter, K ^{[1
]}

机构：

[1] TECH UNIV VIENNA, INST MINERAL CRYSTALLOG & STRUCT CHEM, A-1060 VIENNA, AUSTRIA

来源：

HETEROCYCLES | 1997年 / 45卷 / 04期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Ring closure reactions of 3-alkylamino-6-chloro-N-phenylpyridazine-4-carboxamides (7, 10, 13) bearing a halogen function in ortho position of the carbocyclic moiety were shown to provide convenient access to the pyridazino[3,4-b][1,5]benzodiazepin-5-one system.

引用

页码：673 / 682

页数：10

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