Pyridazines .81. A novel 1,2-diazine containing tricyclic system: Synthesis of pyridazino[3,4-b][1,5]benzodiazepin-5-ones as potential HIV-1 reverse transcriptase inhibitors

被引：0
|
作者：
Heinisch, G [1 ]
Matuszczak, B [1 ]
Mereiter, K [1 ]
机构：
[1] TECH UNIV VIENNA, INST MINERAL CRYSTALLOG & STRUCT CHEM, A-1060 VIENNA, AUSTRIA
来源：
HETEROCYCLES | 1997年 / 45卷 / 04期
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D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Ring closure reactions of 3-alkylamino-6-chloro-N-phenylpyridazine-4-carboxamides (7, 10, 13) bearing a halogen function in ortho position of the carbocyclic moiety were shown to provide convenient access to the pyridazino[3,4-b][1,5]benzodiazepin-5-one system.
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页码：673 / 682
页数：10
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