Synthesis and in vitro anti-bacterial evaluation of tetracyclic-ortho-fused 4H-naphtho[1′,2′-5,6]pyrano[3,4-d](1,2,3)selenadiazole and its derivatives

被引：49

作者：

Karnik, A. V. ^{[1
]}

Kulkarni, A. M. ^{[1
]}

Malviya, N. J. ^{[1
]}

Mourya, B. R. ^{[2
]}

Jadhav, B. L. ^{[2
]}

机构：

[1] Univ Bombay, Dept Chem, Bombay 400098, Maharashtra, India

[2] Univ Bombay, Dept Life Sci, Bombay 400098, Maharashtra, India

来源：

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 2008年 / 43卷 / 11期

关键词：

Anti-bacterial activity; Semicarbazones; Annulation; 1,2,3-Selenadiazole; Naphthopyran;

D O I：

10.1016/j.ejmech.2008.01.026

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Synthesis of new heterocyclic compounds 3a-e containing naphthopyran and selenadiazole as the heterocyclic sub-units in the molecule is achieved using high yielding synthetic protocol. These molecules 3a-e have shown moderate anti-bacterial activity against some gram-positive and grain-negative bacterias. (C) 2008 Elsevier Masson SAS. All rights reserved.

引用

页码：2615 / 2617

页数：3

共 50 条

[21] Synthesis and inhibition of protoporphyrinogen oxidase activity of 3H-pyrazolo[3,4-d][1,2,3]triazin-4-one derivatives
Li, Hua Bin
Xu, Han
Li, Zheng-Ming
Yang, Hua Zheng
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248
[22] SYNTHESIS OF N-ALKYL-N'-(4-DIAZO-5-PYRAZOLYL)UREAS AND THEIR CONVERSION INTO PYRAZOLO[3,4-D][1,2,3]TRIAZOLE AND PYRAZOLO[3,4-D]OXAZOLE DERIVATIVES
VICENTINI, CB
VERONESE, AC
POLI, T
GUARNERI, M
GIORI, P
HETEROCYCLES, 1991, 32 (04) : 727 - 734
[23] SYNTHESIS OF SOME NOVEL ANTIMICROBIAL AND ANTIOXIDANT AGENTS OF FUNCTIONALIZED PYRAZOLO[4′,3′:5,6]PYRANO[3,2-d]-[1,2] AZAPHOSPHOLES AND PYRAZOLO [4′,3′:5,6]PYRANO [2,3-d]-[1,3,2]DIAZAPHOSPHININES
Hassanin, Noha M.
Ali, Tarik E.
El-Shaaer, Hafez M.
Abdel-Kariem, Somaia M.
El-Edfawy, Somaya M.
Abdel-Monem, Wafaa R.
HETEROCYCLES, 2020, 100 (11) : 1902 - 1913
[24] Synthesis and Pharmacological Studies of Unprecedented Fused Pyridazino[3′,4′:5,6][1,2,4]triazino[3,4-b][1,3,4]thiadiazine Derivatives
Ali, Rania S.
Saad, Hosam A.
MOLECULES, 2018, 23 (05):
[25] CHEMISTRY OF 1,2,3-THIADIAZOLE .4. SYNTHESIS OF [1]BENZOXEPINO-[3,4-D][1,2,3]THIADIAZOLE, [1]BENZOTHIEPINO-[3,4-D][1,2,3]THIADIAZOLE, [1]BENZOTHIEPINO[4,3-D][1,2,3]THIADIAZOLE, [1]BENZOXEPINO[4,3-D]OXAZOLE AND [1]BENZOXEPINO[4,3-D]OXAZOLE - 4 NOVEL HETEROCYCLES
SHAFIEE, A
KIAEAY, G
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1981, 18 (05) : 899 - 903
[26] SYNTHESIS OF 5,7-DIHYDRO-6H-NAPHTHO-[1',2'/5,6]PYRANO[3,2-C]QUINOLIN-6-ONES
GUPTA, MCLN
DARBARWAR, M
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1994, 33 (11): : 1080 - 1082
[27] Efficient synthesis of 5-fluoroalkylated 1H-1,2,3-triazoles and application of the bromodifluoromethylated triazole to the synthesis of novel bicyclic gem-difluorinated 1H-pyrano[3,4-d] [1,2,3]-triazol-4-one compounds
Peng, WM
Zhu, SZ
TETRAHEDRON, 2003, 59 (24) : 4395 - 4404
[28] Synthesis and Neurotropic Activity of 1-Substituted 4H-[1]Benzopyrano[3,4-d][1,2,3]triazol-4-ones
V. L. Savel'ev
O. L. Samsonova
V. P. Lezina
V. S. Troitskaya
I. I. Kozlovskii
A. Beshimov
M. M. Kozlovskaya
Pharmaceutical Chemistry Journal, 2003, 37 (9) : 476 - 481
[29] BICYCLIC COMPOUNDS WITH POTENTIAL ANTIULCER AND OR ANTISECRETORY ACTIVITY .2. 1(OR 3),4,6,7-TETRAHYDRO-1(3)H-PYRANO[3,4-D]IMIDAZOLES AND 1(OR 3),4,6,7-TETRAHYDRO-1(3)H-THIOPYRANO[3,4-D]IMIDAZOLES
SCARPONI, U
CIMASCHI, R
ARCARI, G
TOTI, D
BALLABIO, M
GANDINI, E
DECASTIGLIONE, R
FARMACO-EDIZIONE SCIENTIFICA, 1986, 41 (01): : 23 - 40
[30] SYNTHESIS AND SPECTRAL PROPERTIES OF PYRROLO[3',4'-5,6]-4H-PYRANO[2,3-D]PYRIMIDINE DERIVATIVES
MARCHALIN, S
PAVLIKOVA, F
ILAVSKY, D
COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS, 1989, 54 (05) : 1336 - 1345

← 1 2 3 4 5 →