Multicomponent eco-friendly synthesis of 3,4-dihydropyrimidine-2-(1H)-ones using an organocatalyst Lactic acid

被引：30
|
作者：
Suresh [1 ]
Saini, Anil [1 ]
Kumar, Dhruva [1 ]
Sandhu, Jagir S. [1 ]
机构：
[1] Punjabi Univ, Dept Chem, Patiala 147002, Punjab, India
来源：
GREEN CHEMISTRY LETTERS AND REVIEWS | 2009年 / 2卷 / 01期
关键词：
aldehyde; 1,3-dicarbonyl compound; urea; Lactic acid; CALCIUM-CHANNEL BLOCKERS; ONE-POT SYNTHESIS; SOLVENT-FREE CONDITIONS; BIGINELLI REACTION; CONDENSATION REACTION; LITHIUM BROMIDE; CATALYST; 3,4-DIHYDROPYRIMIDIN-2(1H)-ONES; ESTERS; WATER;
D O I：
10.1080/17518250902973833
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Biginelli compounds 3,4-dihydropyrimidine-2-(1H)-ones are synthesized in high yields via eco-friendly simple reaction procedure using Lactic acid: organocatalyst. The new method reported herein is green and is free of formation of any hazardous by products. The process has significant advantages over other reported methods. [GRAPHICS] .
引用
收藏
页码：29 / 33
页数：5
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